AU2007315943A1 - IKK-beta serine-threonine protein kinase inhibitors - Google Patents
IKK-beta serine-threonine protein kinase inhibitors Download PDFInfo
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- AU2007315943A1 AU2007315943A1 AU2007315943A AU2007315943A AU2007315943A1 AU 2007315943 A1 AU2007315943 A1 AU 2007315943A1 AU 2007315943 A AU2007315943 A AU 2007315943A AU 2007315943 A AU2007315943 A AU 2007315943A AU 2007315943 A1 AU2007315943 A1 AU 2007315943A1
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- cyclopentyl
- carbamoylamino
- carbamoyl
- alkyl
- optionally substituted
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- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Diabetes (AREA)
- Pulmonology (AREA)
- Dermatology (AREA)
- Endocrinology (AREA)
- Transplantation (AREA)
- Obesity (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Hematology (AREA)
- Reproductive Health (AREA)
- Emergency Medicine (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Enzymes And Modification Thereof (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0621720A GB0621720D0 (en) | 2006-11-01 | 2006-11-01 | Inhibitors of ikk- serine-threonine protein kinase |
| GB0621720.2 | 2006-11-01 | ||
| GB0715470A GB0715470D0 (en) | 2007-08-09 | 2007-08-09 | IKK- serine-threonine protein kinase inhibitors |
| GB0715470.1 | 2007-08-09 | ||
| PCT/GB2007/004114 WO2008053182A1 (en) | 2006-11-01 | 2007-10-29 | IKK-β SERINE-THREONINE PROTEIN KINASE INHIBITORS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2007315943A1 true AU2007315943A1 (en) | 2008-05-08 |
Family
ID=39015937
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2007315943A Abandoned AU2007315943A1 (en) | 2006-11-01 | 2007-10-29 | IKK-beta serine-threonine protein kinase inhibitors |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US8003695B2 (enExample) |
| EP (1) | EP2078007B1 (enExample) |
| JP (1) | JP2010508336A (enExample) |
| KR (1) | KR20090077975A (enExample) |
| AT (1) | ATE522516T1 (enExample) |
| AU (1) | AU2007315943A1 (enExample) |
| BR (1) | BRPI0718056A2 (enExample) |
| CA (1) | CA2668338A1 (enExample) |
| DK (1) | DK2078007T3 (enExample) |
| EA (1) | EA200900616A1 (enExample) |
| ES (1) | ES2372707T3 (enExample) |
| IL (1) | IL198267A0 (enExample) |
| MX (1) | MX2009004442A (enExample) |
| NZ (1) | NZ576705A (enExample) |
| WO (1) | WO2008053182A1 (enExample) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0619753D0 (en) | 2006-10-06 | 2006-11-15 | Chroma Therapeutics Ltd | Enzyme inhibitors |
| GB0803747D0 (en) | 2008-02-29 | 2008-04-09 | Martin | Enzyme and receptor modulation |
| MX2010011501A (es) * | 2008-04-23 | 2010-11-30 | Chroma Therapeutics Ltd | Inhibidores de proteina cinasa de serina-treonina ikk-beta. |
| BRPI0911480A2 (pt) * | 2008-04-26 | 2018-04-03 | Chroma Therapeutics Ltd | inibidores de proteínas serina-treonina quinase ikk-beta |
| EP2361245A4 (en) * | 2008-11-26 | 2012-06-13 | Trt Pharma Inc | HYBRID-IONONE AND CURCUMINE MOLECULES AS ANTICREBIALS |
| GB0903480D0 (en) | 2009-02-27 | 2009-04-08 | Chroma Therapeutics Ltd | Enzyme Inhibitors |
| GB0907120D0 (en) * | 2009-04-24 | 2009-06-03 | Chroma Therapeutics Ltd | Inhibitors of IKK-ß serine-threonine protein kinase |
| GB201211310D0 (en) | 2012-06-26 | 2012-08-08 | Chroma Therapeutics Ltd | CSF-1R kinase inhibitors |
| HRP20171320T1 (hr) | 2012-10-17 | 2017-10-20 | Macrophage Pharma Limited | Terc-butil n-[2-{4-[6-amino-5-(2,4-difluorobenzoil)-2-oksopiridin-1(2h)-il]-3,5-difluorofenil}etil]-l-alaninat ili njegova sol, hidrat ili solvat |
| US9809577B2 (en) * | 2013-12-11 | 2017-11-07 | Biogen Ma Inc. | Biaryl inhibitors of Bruton's tyrosine kinase |
| GB201713975D0 (en) | 2017-08-31 | 2017-10-18 | Macrophage Pharma Ltd | Medical use |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE0102616D0 (sv) * | 2001-07-25 | 2001-07-25 | Astrazeneca Ab | Novel compounds |
| SE0300092D0 (sv) | 2003-01-15 | 2003-01-15 | Astrazeneca Ab | Novel compounds |
-
2007
- 2007-10-29 WO PCT/GB2007/004114 patent/WO2008053182A1/en not_active Ceased
- 2007-10-29 AT AT07824358T patent/ATE522516T1/de not_active IP Right Cessation
- 2007-10-29 AU AU2007315943A patent/AU2007315943A1/en not_active Abandoned
- 2007-10-29 JP JP2009535115A patent/JP2010508336A/ja not_active Withdrawn
- 2007-10-29 EA EA200900616A patent/EA200900616A1/ru unknown
- 2007-10-29 US US12/513,206 patent/US8003695B2/en not_active Expired - Fee Related
- 2007-10-29 CA CA002668338A patent/CA2668338A1/en not_active Abandoned
- 2007-10-29 DK DK07824358.1T patent/DK2078007T3/da active
- 2007-10-29 MX MX2009004442A patent/MX2009004442A/es active IP Right Grant
- 2007-10-29 BR BRPI0718056-0A patent/BRPI0718056A2/pt not_active IP Right Cessation
- 2007-10-29 ES ES07824358T patent/ES2372707T3/es active Active
- 2007-10-29 NZ NZ576705A patent/NZ576705A/en not_active IP Right Cessation
- 2007-10-29 KR KR1020097011261A patent/KR20090077975A/ko not_active Withdrawn
- 2007-10-29 EP EP07824358A patent/EP2078007B1/en not_active Not-in-force
-
2009
- 2009-04-21 IL IL198267A patent/IL198267A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NZ576705A (en) | 2011-12-22 |
| EP2078007A1 (en) | 2009-07-15 |
| DK2078007T3 (da) | 2011-12-12 |
| ES2372707T3 (es) | 2012-01-25 |
| US8003695B2 (en) | 2011-08-23 |
| WO2008053182A1 (en) | 2008-05-08 |
| IL198267A0 (en) | 2009-12-24 |
| EA200900616A1 (ru) | 2010-04-30 |
| BRPI0718056A2 (pt) | 2013-11-05 |
| JP2010508336A (ja) | 2010-03-18 |
| EP2078007B1 (en) | 2011-08-31 |
| MX2009004442A (es) | 2009-05-22 |
| CA2668338A1 (en) | 2008-05-08 |
| KR20090077975A (ko) | 2009-07-16 |
| ATE522516T1 (de) | 2011-09-15 |
| US20100087515A1 (en) | 2010-04-08 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK4 | Application lapsed section 142(2)(d) - no continuation fee paid for the application |