ES2335664T3 - Derivados de 8-aza-biciclo(3.2.1)octano y su uso como inhibidores de la reabsorcion de neurotransmisores de monoaminas. - Google Patents
Derivados de 8-aza-biciclo(3.2.1)octano y su uso como inhibidores de la reabsorcion de neurotransmisores de monoaminas. Download PDFInfo
- Publication number
- ES2335664T3 ES2335664T3 ES04709633T ES04709633T ES2335664T3 ES 2335664 T3 ES2335664 T3 ES 2335664T3 ES 04709633 T ES04709633 T ES 04709633T ES 04709633 T ES04709633 T ES 04709633T ES 2335664 T3 ES2335664 T3 ES 2335664T3
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- Prior art keywords
- aza
- bicyclo
- octane
- methyl
- thienyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
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Classifications
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Landscapes
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- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
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- Medicinal Chemistry (AREA)
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Applications Claiming Priority (4)
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| US44810603P | 2003-02-20 | 2003-02-20 | |
| US448106P | 2003-02-20 |
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| EP1779851A1 (en) * | 2005-10-31 | 2007-05-02 | Boehringer Ingelheim Pharma GmbH & Co.KG | Treatment of diabetes |
| JP5194607B2 (ja) * | 2006-07-26 | 2013-05-08 | 大正製薬株式会社 | ソーシャルインターラクションの低下予防・改善剤 |
| DE102007046887A1 (de) * | 2007-09-28 | 2009-04-09 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Verfahren zur Herstellung von (1R,5S)-Anhydroecgoninestersalzen |
| WO2009065845A1 (en) * | 2007-11-20 | 2009-05-28 | Neurosearch A/S | A method for treating over-eating disorders |
| US8101642B2 (en) | 2008-06-05 | 2012-01-24 | Sk Biopharmaceuticals Co., Ltd. | 3-substituted propanamine compounds |
| US8546576B2 (en) | 2008-06-06 | 2013-10-01 | Sk Biopharmaceuticals Co., Ltd. | 3 or 4-substituted piperidine compounds |
| WO2010086612A1 (en) | 2009-01-29 | 2010-08-05 | Cambrex Karlskoga Ab | Process for preparing enantiomerically enriched alkaloids |
| WO2014130910A1 (en) | 2013-02-22 | 2014-08-28 | Baylor College Of Medicine | Treatment for substance use disorders and stress disorders |
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| FI111367B (fi) * | 1991-02-04 | 2003-07-15 | Aventis Pharma Inc | Menetelmä terapeuttisesti käyttökelpoisten N-(aryylioksialkyyli)heteroaryyli-8-atsabisyklo[3.2.1]oktaanijohdannaisten valmistamiseksi ja menetelmässä käytetyt välituotteet |
| AU672052B2 (en) * | 1992-12-23 | 1996-09-19 | Neurosearch A/S | Antidepressant and antiparkinsonian compounds |
| CZ285571B6 (cs) | 1995-11-02 | 1999-09-15 | Neurosearch A/S | Kondenzované tropanové deriváty, způsob jejich výroby, farmaceutické prostředky, které je obsahují a jejich použití k léčení |
| TR199801641T2 (xx) | 1996-02-22 | 1998-11-23 | Neurosearch A/S | Tropan t�revleri bunlar�n haz�rlanmas� ve kullan�m� |
| AU4819099A (en) | 1998-06-19 | 2000-01-05 | Eli Lilly And Company | Inhibition of serotonin reuptake |
| AU9543601A (en) * | 2000-10-13 | 2002-04-22 | Neurosearch As | Treatment of affective disorders by the combined action of a nicotinic receptor agonist and a monoaminergic substance |
| AU2002306848A1 (en) * | 2001-03-23 | 2002-10-08 | Elan Pharmaceuticals, Inc. | Methods of treating alzheimer's disease with piperidin derivates |
| JP2005508872A (ja) * | 2001-05-23 | 2005-04-07 | ニューロサーチ、アクティーゼルスカブ | トロパン誘導体及びこれをモノアミン神経伝達物質再取り込み阻害剤として使用する方法 |
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Also Published As
| Publication number | Publication date |
|---|---|
| US7247643B2 (en) | 2007-07-24 |
| US20060122218A1 (en) | 2006-06-08 |
| DE602004024033D1 (de) | 2009-12-24 |
| EP1594868A1 (en) | 2005-11-16 |
| EP1594868B1 (en) | 2009-11-11 |
| MXPA05008314A (es) | 2005-10-05 |
| NZ541249A (en) | 2008-04-30 |
| WO2004072071A1 (en) | 2004-08-26 |
| AU2004212166A1 (en) | 2004-08-26 |
| ATE448223T1 (de) | 2009-11-15 |
| CA2515584A1 (en) | 2004-08-26 |
| AU2004212166B2 (en) | 2010-07-29 |
| JP2006517568A (ja) | 2006-07-27 |
| DK1594868T3 (da) | 2010-03-15 |
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