ES2237770T3 - Solucion de irrigacion vascular y metodo de inhibicion del dolor, de la inflamacion, del espasmo y de la restenosis. - Google Patents

Solucion de irrigacion vascular y metodo de inhibicion del dolor, de la inflamacion, del espasmo y de la restenosis.

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Publication number
ES2237770T3
ES2237770T3 ES96923473T ES96923473T ES2237770T3 ES 2237770 T3 ES2237770 T3 ES 2237770T3 ES 96923473 T ES96923473 T ES 96923473T ES 96923473 T ES96923473 T ES 96923473T ES 2237770 T3 ES2237770 T3 ES 2237770T3
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ES
Spain
Prior art keywords
antagonists
nanomolar
inhibitors
receptor
agents
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES96923473T
Other languages
English (en)
Spanish (es)
Inventor
Gregory A. Demopulos
Pamela Anne Pierce
Jeffrey M. Herz
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Omeros Corp
Original Assignee
Omeros Medical Systems Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/US1995/016028 external-priority patent/WO1996019233A2/en
Application filed by Omeros Medical Systems Inc filed Critical Omeros Medical Systems Inc
Application granted granted Critical
Publication of ES2237770T3 publication Critical patent/ES2237770T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/08—Peptides having 5 to 11 amino acids
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404—Indoles, e.g. pindolol
    • A61K31/4045—Indole-alkylamines; Amides thereof, e.g. serotonin, melatonin
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    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
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    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
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ES96923473T 1995-12-12 1996-06-26 Solucion de irrigacion vascular y metodo de inhibicion del dolor, de la inflamacion, del espasmo y de la restenosis. Expired - Lifetime ES2237770T3 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
WOPCT/US95/16028 1995-12-12
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KR100517210B1 (ko) 2006-06-07
KR19980700084A (OSRAM) 1998-03-30
EP0910397B1 (en) 2005-03-02
CN1209066A (zh) 1999-02-24
EP0910397A1 (en) 1999-04-28
DE69634420T2 (de) 2006-02-09
JP2008094855A (ja) 2008-04-24
JP2000501729A (ja) 2000-02-15
AU6397496A (en) 1997-07-03
CN1182869C (zh) 2005-01-05
ATE289822T1 (de) 2005-03-15
CA2240256A1 (en) 1997-06-19
CA2240256C (en) 2009-04-14
DE69634420D1 (de) 2005-04-07
WO1997021445A1 (en) 1997-06-19

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