ES2173890T3 - Derivados de 17-halogeno-4-azaandrosteno y procedimiento para su preparacion. - Google Patents

Derivados de 17-halogeno-4-azaandrosteno y procedimiento para su preparacion.

Info

Publication number
ES2173890T3
ES2173890T3 ES93913460T ES93913460T ES2173890T3 ES 2173890 T3 ES2173890 T3 ES 2173890T3 ES 93913460 T ES93913460 T ES 93913460T ES 93913460 T ES93913460 T ES 93913460T ES 2173890 T3 ES2173890 T3 ES 2173890T3
Authority
ES
Spain
Prior art keywords
pct
azaandrosteno
halogeno
derivatives
procedure
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES93913460T
Other languages
English (en)
Inventor
Zoltan Tuba
Judit Horvath
Janos Szeles
Marsai Maria Lovasne
Gabor Balogh
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Richter Gedeon Vegyeszeti Gyar Nyrt
Original Assignee
Richter Gedeon Vegyeszeti Gyar RT
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richter Gedeon Vegyeszeti Gyar RT filed Critical Richter Gedeon Vegyeszeti Gyar RT
Application granted granted Critical
Publication of ES2173890T3 publication Critical patent/ES2173890T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/005—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

LA INVENCION SE REFIERE A DERIVADOS DE 4-AZAANDROSTENO NOVEDOSOS DE LA FORMULA GENERAL (I), DONDE R REPRESENTA HIDROGENO O UN GRUPO ALQUIL C{SUB,1-3}; X REPRESENTA CLORO, BROMINA O IODINA, Y LA LINEA DE UNION ----- REPRESENTA UNA UNION SENCILLA O DOBLE.
ES93913460T 1993-06-24 1993-06-24 Derivados de 17-halogeno-4-azaandrosteno y procedimiento para su preparacion. Expired - Lifetime ES2173890T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/HU1993/000040 WO1995000532A1 (en) 1993-06-24 1993-06-24 17-halogeno-4-azaandrostene derivatives and process for the preparation thereof

Publications (1)

Publication Number Publication Date
ES2173890T3 true ES2173890T3 (es) 2002-11-01

Family

ID=10982848

Family Applications (1)

Application Number Title Priority Date Filing Date
ES93913460T Expired - Lifetime ES2173890T3 (es) 1993-06-24 1993-06-24 Derivados de 17-halogeno-4-azaandrosteno y procedimiento para su preparacion.

Country Status (15)

Country Link
US (1) US5583228A (es)
EP (1) EP0705273B1 (es)
JP (1) JP3300359B2 (es)
KR (1) KR100255679B1 (es)
AT (1) ATE215093T1 (es)
AU (1) AU680825B2 (es)
CA (1) CA2166089C (es)
DE (1) DE69331764T2 (es)
DK (1) DK0705273T3 (es)
ES (1) ES2173890T3 (es)
FI (1) FI956235A0 (es)
PT (1) PT705273E (es)
RU (1) RU2103275C1 (es)
UA (1) UA41934C2 (es)
WO (1) WO1995000532A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU212459B (en) * 1992-10-02 1996-06-28 Richter Gedeon Vegyeszet Process for producing new 17-beta-substituted 4-aza-androstane-derivatives and pharmaceutical compositions containing them
CA2524409C (en) * 2003-05-07 2011-12-20 Merck & Co., Inc. Androgen receptor modulators and methods of use thereof
CN102603839A (zh) * 2012-01-13 2012-07-25 宜城市共同药业有限公司 去氢表雄酮的制备方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4377584A (en) * 1978-04-13 1983-03-22 Merck & Co., Inc. 4-Aza-17β-substituted-5α-androstan-3-one-reductase inhibitors
US5359071A (en) * 1993-03-12 1994-10-25 Merck & Co., Inc. 15-substituted 4-azasteroids

Also Published As

Publication number Publication date
AU4352793A (en) 1995-01-17
ATE215093T1 (de) 2002-04-15
AU680825B2 (en) 1997-08-14
DE69331764D1 (de) 2002-05-02
DE69331764T2 (de) 2002-10-02
EP0705273B1 (en) 2002-03-27
JPH08511797A (ja) 1996-12-10
EP0705273A1 (en) 1996-04-10
PT705273E (pt) 2002-07-31
UA41934C2 (uk) 2001-10-15
FI956235A (fi) 1995-12-22
CA2166089A1 (en) 1995-01-05
FI956235A0 (fi) 1995-12-22
US5583228A (en) 1996-12-10
JP3300359B2 (ja) 2002-07-08
WO1995000532A1 (en) 1995-01-05
RU2103275C1 (ru) 1998-01-27
KR100255679B1 (ko) 2000-08-01
DK0705273T3 (da) 2002-06-17
CA2166089C (en) 2004-01-27
KR960703134A (ko) 1996-06-19

Similar Documents

Publication Publication Date Title
AU7116691A (en) Process for the preparation of oxetanones
SG55184A1 (en) New imidazopyridines
BR9407239A (pt) Azadioxacicloalquenos substituídos
FI932229A0 (fi) Azabicykliska bryggderivat
HU9303666D0 (en) Azanorbornane derivatives
DE69428546D1 (en) 3-acylaminobenzazepine
AU2223595A (en) Aziridine derivatives, their production and use
AU8252787A (en) Process for the preparation of thienylethylamines and novel dithienylethylamines
ES2173890T3 (es) Derivados de 17-halogeno-4-azaandrosteno y procedimiento para su preparacion.
AU1193597A (en) Process for the preparation of 2-chloro-5-chloromethyl-thiazole
AU3716093A (en) Dithiolanylglycine-containing HIV protease inhibitors of the hydroxyethylene isostere type
AU4706293A (en) Therapeutic use of phosphoryl-l-serine-n-acyl-sphingosine
AU1600495A (en) Novel indane-2-mercaptoacetylamide disulfide derivatives useful as inhibitors of enkephalinase
GR3029590T3 (en) Crystalline, polymorphic form of (s,s,s)-n-(1- 2-carboxy-3-(n?2 -mesyllysylamino)propyl]-1-cyclopentylcarbonyl)tyrosine
FI963166A (fi) Uusia merkaptoasetyyliamididisulfidijohdannaisia, jotka ovat käyttökelpoisia enkefalinaasin ja ACE:n inhibiittoreina
ES2152982T3 (es) Analogos de la difluoroestatona.
ES2172699T3 (es) Procedimiento para la preparacion de prostaglandina e1.
MX9802000A (es) Sales de adicion de acido de compuestos de 2,3,4,5-tetrahidro-1h-3-benzacepina.

Legal Events

Date Code Title Description
FG2A Definitive protection

Ref document number: 705273

Country of ref document: ES