ATE215093T1 - 17-halogen-4-azaandrosten-derivate und verfahren zu ihrer herstellung - Google Patents

17-halogen-4-azaandrosten-derivate und verfahren zu ihrer herstellung

Info

Publication number
ATE215093T1
ATE215093T1 AT93913460T AT93913460T ATE215093T1 AT E215093 T1 ATE215093 T1 AT E215093T1 AT 93913460 T AT93913460 T AT 93913460T AT 93913460 T AT93913460 T AT 93913460T AT E215093 T1 ATE215093 T1 AT E215093T1
Authority
AT
Austria
Prior art keywords
pct
halogen
production
azaandrostene
sec
Prior art date
Application number
AT93913460T
Other languages
English (en)
Inventor
Zoltan Tuba
Judit Horvath
Janos Szeles
Marsai Maria Lovasne
Gabor Balogh
Original Assignee
Richter Gedeon Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richter Gedeon Vegyeszet filed Critical Richter Gedeon Vegyeszet
Application granted granted Critical
Publication of ATE215093T1 publication Critical patent/ATE215093T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/005—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AT93913460T 1993-06-24 1993-06-24 17-halogen-4-azaandrosten-derivate und verfahren zu ihrer herstellung ATE215093T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/HU1993/000040 WO1995000532A1 (en) 1993-06-24 1993-06-24 17-halogeno-4-azaandrostene derivatives and process for the preparation thereof

Publications (1)

Publication Number Publication Date
ATE215093T1 true ATE215093T1 (de) 2002-04-15

Family

ID=10982848

Family Applications (1)

Application Number Title Priority Date Filing Date
AT93913460T ATE215093T1 (de) 1993-06-24 1993-06-24 17-halogen-4-azaandrosten-derivate und verfahren zu ihrer herstellung

Country Status (15)

Country Link
US (1) US5583228A (de)
EP (1) EP0705273B1 (de)
JP (1) JP3300359B2 (de)
KR (1) KR100255679B1 (de)
AT (1) ATE215093T1 (de)
AU (1) AU680825B2 (de)
CA (1) CA2166089C (de)
DE (1) DE69331764T2 (de)
DK (1) DK0705273T3 (de)
ES (1) ES2173890T3 (de)
FI (1) FI956235A7 (de)
PT (1) PT705273E (de)
RU (1) RU2103275C1 (de)
UA (1) UA41934C2 (de)
WO (1) WO1995000532A1 (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU212459B (en) * 1992-10-02 1996-06-28 Richter Gedeon Vegyeszet Process for producing new 17-beta-substituted 4-aza-androstane-derivatives and pharmaceutical compositions containing them
JP4832303B2 (ja) * 2003-05-07 2011-12-07 メルク・シャープ・エンド・ドーム・コーポレイション アンドロゲン受容体モジュレータおよびこれらの使用
CN102603839A (zh) * 2012-01-13 2012-07-25 宜城市共同药业有限公司 去氢表雄酮的制备方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4377584A (en) * 1978-04-13 1983-03-22 Merck & Co., Inc. 4-Aza-17β-substituted-5α-androstan-3-one-reductase inhibitors
US5359071A (en) * 1993-03-12 1994-10-25 Merck & Co., Inc. 15-substituted 4-azasteroids

Also Published As

Publication number Publication date
EP0705273B1 (de) 2002-03-27
CA2166089A1 (en) 1995-01-05
RU2103275C1 (ru) 1998-01-27
FI956235A0 (fi) 1995-12-22
US5583228A (en) 1996-12-10
FI956235L (fi) 1995-12-22
DK0705273T3 (da) 2002-06-17
AU680825B2 (en) 1997-08-14
KR960703134A (ko) 1996-06-19
AU4352793A (en) 1995-01-17
WO1995000532A1 (en) 1995-01-05
DE69331764D1 (de) 2002-05-02
DE69331764T2 (de) 2002-10-02
UA41934C2 (uk) 2001-10-15
KR100255679B1 (ko) 2000-08-01
CA2166089C (en) 2004-01-27
ES2173890T3 (es) 2002-11-01
FI956235A7 (fi) 1995-12-22
EP0705273A1 (de) 1996-04-10
JP3300359B2 (ja) 2002-07-08
PT705273E (pt) 2002-07-31
JPH08511797A (ja) 1996-12-10

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Legal Events

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