ES2160161T3 - Composiciones farmaceuticas derivadas de geles basados en microemulsiones, metodo para su preparacion y nuevos geles basados en microemulsiones. - Google Patents

Composiciones farmaceuticas derivadas de geles basados en microemulsiones, metodo para su preparacion y nuevos geles basados en microemulsiones.

Info

Publication number
ES2160161T3
ES2160161T3 ES95916686T ES95916686T ES2160161T3 ES 2160161 T3 ES2160161 T3 ES 2160161T3 ES 95916686 T ES95916686 T ES 95916686T ES 95916686 T ES95916686 T ES 95916686T ES 2160161 T3 ES2160161 T3 ES 2160161T3
Authority
ES
Spain
Prior art keywords
microemulsion
component
hydrophilic
lipophilic
pct
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES95916686T
Other languages
English (en)
Inventor
Sune Backlund
Folke Eriksson
Maria Rantala
Pertti Rantala
Kari Varho
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer Oy
Original Assignee
Leiras Oy
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Leiras Oy filed Critical Leiras Oy
Application granted granted Critical
Publication of ES2160161T3 publication Critical patent/ES2160161T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/06Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Dispersion Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Colloid Chemistry (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

LA INVENCION HACE REFERENCIA A UNA COMPOSICION FARMACEUTICA QUE INCLUYE UNA MICROEMULSION HECHA DE UN COMPONENTE HIDROFILICO, UN COMPONENTE LIPOFILICO, UN SURFACTANTE Y UN MEDICAMENTO, DE FORMA QUE EL COMPONENTE HIDROFILICO, EL COMPONENTE LIPOFILICO, Y EL SURFACTANTE FORMAN, CUANDO SE EXAMINAN EN UNA ESCALA MACROSCOPICA, UNA SOLUCION DE UNA FASE. EL COMPONENTE HIDROFILICO SE DISPERSA COMO GOTITAS COLOIDALES EN EL COMPONENTE LIPOFILICO, O EL COMPONENTE LIPOFILICO SE DISPERSA COMO GOTITAS COLOIDALES EN EL COMPONENTE HIDROFILICO. EN OTRA ALTERNATIVA LOS COMPONENTES HIDROFILICOS Y LIPOFILICOS FORMAN UNA MICROEMULSION CON ESTRUCTURA BICONTINUA DE FORMA QUE DICHOS COMPONENTES FORMAN CANALES ADYACENTES ALARGADOS. EL MEDICAMENTO SE DISUELVE EN EL COMPONENTE DISPERSADO O, EN EL CASO DE UNA MICROEMULSION CON UN ESTRUCTURA BICONTINUA, EN EL COMPONENTE HIDROFILICO O LIPOFILICO. LA MICROEMULSION SE ESTABILIZA MEDIANTE EL SURFACTANTE. ES CARACTERISTICO AÑADIR UN GELIFICADOR Y AGUA A LA EMULSION DANDOLE ASI A ESTA LA FORMA DE GEL.
ES95916686T 1994-05-24 1995-04-28 Composiciones farmaceuticas derivadas de geles basados en microemulsiones, metodo para su preparacion y nuevos geles basados en microemulsiones. Expired - Lifetime ES2160161T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FI942387A FI100692B (fi) 1994-05-24 1994-05-24 Menetelmä farmaseuttisten koostumusten valmistamiseksi, jolloin koostu mukset pohjautuvat mikroemulsiogeeleihin sekä uusia mikroemulsioihin p ohjautuvia geelejä

Publications (1)

Publication Number Publication Date
ES2160161T3 true ES2160161T3 (es) 2001-11-01

Family

ID=8540757

Family Applications (1)

Application Number Title Priority Date Filing Date
ES95916686T Expired - Lifetime ES2160161T3 (es) 1994-05-24 1995-04-28 Composiciones farmaceuticas derivadas de geles basados en microemulsiones, metodo para su preparacion y nuevos geles basados en microemulsiones.

Country Status (13)

Country Link
US (1) US6004580A (es)
EP (1) EP0760651B1 (es)
JP (1) JPH10500675A (es)
AT (1) ATE202699T1 (es)
AU (1) AU2309195A (es)
CA (1) CA2190869A1 (es)
DE (1) DE69521611T2 (es)
DK (1) DK0760651T3 (es)
ES (1) ES2160161T3 (es)
FI (1) FI100692B (es)
GR (1) GR3036681T3 (es)
PT (1) PT760651E (es)
WO (1) WO1995031969A1 (es)

Families Citing this family (34)

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GB2305603A (en) * 1995-09-26 1997-04-16 Allied Medical Group Topical cooling gels for reducing excess body fat
GB9601120D0 (en) * 1996-01-19 1996-03-20 Sandoz Ltd Organic compounds
US5858401A (en) 1996-01-22 1999-01-12 Sidmak Laboratories, Inc. Pharmaceutical composition for cyclosporines
US5686133A (en) * 1996-01-31 1997-11-11 Port Systems, L.L.C. Water soluble pharmaceutical coating and method for producing coated pharmaceuticals
GR1002706B (el) * 1996-05-22 1997-05-26 Μικρογαλακτωματα λεκιθινης περιεχοντα πρωτεολυτικα ενζυμα α-χυμοθρυψινης η θρυψινη και μεθοδος μονιμης ενζυμικης αποτριχωσης.
DE19641672A1 (de) * 1996-10-10 1998-04-16 Beiersdorf Ag Kosmetische oder dermatologische Zubereitungen auf der Basis von ethylenoxidfreien und propylenoxidfreien Emulgatoren zur Herstellung von Mikroemulsionsgelen
DE19810655A1 (de) * 1998-03-12 1999-09-16 Univ Eberhard Karls Arzneimittel mit einem Gehalt an Ciclosporin
US7064114B2 (en) 1999-03-19 2006-06-20 Parker Hughes Institute Gel-microemulsion formulations
JP2002540080A (ja) * 1999-03-19 2002-11-26 パーカー ヒューズ インスティテュート ゲルミクロ乳濁液製剤
US7919113B2 (en) * 1999-12-30 2011-04-05 Yissum Research Development Company Of The Hebrew University Of Jerusalem Dispersible concentrate lipospheres for delivery of active agents
US7732404B2 (en) 1999-12-30 2010-06-08 Dexcel Ltd Pro-nanodispersion for the delivery of cyclosporin
WO2003032949A1 (en) * 2001-10-19 2003-04-24 Isotechnika Inc. Novel cyclosporin analog microemulsion preconcentrates
US20030113366A1 (en) * 2001-12-14 2003-06-19 Macgregor Alexander Reverse-micellar delivery system for controlled transportation and enhanced absorption of agents
US6858666B2 (en) * 2002-03-04 2005-02-22 Aveka, Inc. Organogel particles
US20040018237A1 (en) * 2002-05-31 2004-01-29 Perricone Nicholas V. Topical drug delivery using phosphatidylcholine
US8642079B2 (en) 2004-02-23 2014-02-04 Hormos Medical Corporation Solid formulations of ospemifene
US20050232974A1 (en) * 2004-04-19 2005-10-20 Gore Makarand P System and a method for pharmaceutical dosage preparation using jettable microemulsions
SI2275098T1 (sl) 2004-05-04 2012-12-31 Hormos Medical Ltd. Nove oralne formulacije ospemifena
US8758821B2 (en) 2004-05-04 2014-06-24 Hormos Medical Ltd. Oral formulations of ospemifene
US7862552B2 (en) 2005-05-09 2011-01-04 Boston Scientific Scimed, Inc. Medical devices for treating urological and uterine conditions
GB2464393B (en) * 2006-11-29 2011-05-18 Malvern Cosmeceutics Ltd Solubilised peptide or protein formulations using molecular assemblies comprising a surfactant and a lipid
GB0623838D0 (en) 2006-11-29 2007-01-10 Malvern Cosmeceutics Ltd Novel compositions
ES2590262T3 (es) 2007-02-14 2016-11-21 Hormos Medical Ltd. Método para la preparación de derivados de trifenilbuteno con valor terapéutico
US7504530B2 (en) 2007-02-14 2009-03-17 Hormos Medical Ltd. Methods for the preparation of fispemifene from ospemifene
FR2917976B1 (fr) * 2007-06-29 2010-05-28 Galderma Sa Composition dermatologique comprenant des vehicules lipidiques de calcitriol, son procede de preparation et son utilisation
MX2011003207A (es) * 2008-09-27 2011-11-04 Jina Pharmaceuticals Inc Preparaciones farmaceuticas a base de lipidos para la aplicacion oral y topica; sus composiciones, metodos y usos.
EP2355803A4 (en) * 2008-11-14 2012-04-25 Archer Daniels Midland Co COMPOSITIONS AND METHODS FOR ORGANOGEL PRODUCTION
JP5901617B2 (ja) * 2010-05-14 2016-04-13 アーチャー−ダニエルズ−ミッドランド カンパニー オルガノゲルを含む食品組成物
WO2014060639A1 (en) 2012-10-19 2014-04-24 Fermion Oy A process for the preparation of ospemifene
WO2014063761A1 (en) * 2012-10-26 2014-05-01 Services Petroliers Schlumberger Compositions and methods for completing subterranean wells
WO2015164657A1 (en) * 2014-04-23 2015-10-29 Bcs Business Consulting Services Pte Ltd Incorporation of water soluble component(s) into anhydrous formulations
WO2016128235A1 (en) * 2015-02-11 2016-08-18 Nestec S.A. Vitamin a composition
CN106963725A (zh) * 2017-04-19 2017-07-21 赵艳霞 一种地塞米松纳米凝胶及其制备方法
JP6815497B2 (ja) 2017-05-18 2021-01-20 キユーピー株式会社 自己乳化性を有する組成物、及びその製造方法、並びにナノエマルション、及びその製造方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT370721B (de) * 1981-02-24 1983-04-25 Ciba Geigy Ag Verfahren zur herstellung von neuen salzen der 2- (2,6-dichloranilino)-phenylessigsaeure, der
CH662944A5 (it) * 1984-10-18 1987-11-13 Pier Luigi Prof Dr Luisi Procedimento per la preparazione di biocompatibili di micelle inverse di biocompatibili e loro utilizzazione.
US5294249A (en) * 1987-03-27 1994-03-15 Luisi Pier L Blendpolymers
US5342625A (en) * 1988-09-16 1994-08-30 Sandoz Ltd. Pharmaceutical compositions comprising cyclosporins
KR0148748B1 (ko) * 1988-09-16 1998-08-17 장 크라메르, 한스 루돌프 하우스 사이클로스포린을 함유하는 약학조성물
US5206219A (en) * 1991-11-25 1993-04-27 Applied Analytical Industries, Inc. Oral compositions of proteinaceous medicaments

Also Published As

Publication number Publication date
DE69521611D1 (de) 2001-08-09
JPH10500675A (ja) 1998-01-20
DK0760651T3 (da) 2001-10-22
EP0760651A1 (en) 1997-03-12
FI942387A0 (fi) 1994-05-24
FI942387A (fi) 1995-11-25
ATE202699T1 (de) 2001-07-15
PT760651E (pt) 2001-11-30
WO1995031969A1 (en) 1995-11-30
FI100692B (fi) 1998-02-13
EP0760651B1 (en) 2001-07-04
CA2190869A1 (en) 1995-11-30
GR3036681T3 (en) 2001-12-31
AU2309195A (en) 1995-12-18
DE69521611T2 (de) 2001-10-18
US6004580A (en) 1999-12-21

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