ES2145142T3 - Compuesto de acido succinamico, procedimiento para su produccion y su uso. - Google Patents

Compuesto de acido succinamico, procedimiento para su produccion y su uso.

Info

Publication number
ES2145142T3
ES2145142T3 ES94921848T ES94921848T ES2145142T3 ES 2145142 T3 ES2145142 T3 ES 2145142T3 ES 94921848 T ES94921848 T ES 94921848T ES 94921848 T ES94921848 T ES 94921848T ES 2145142 T3 ES2145142 T3 ES 2145142T3
Authority
ES
Spain
Prior art keywords
succinamic acid
pharmaceutically acceptable
acceptable salt
acid compound
present
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES94921848T
Other languages
English (en)
Inventor
Hiroshi Hosono
Toshiyuki Nishio
Hiromichi Gurandohait Ishikawa
Yoshiyuki Nakamura
Tetsuo Matsui
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Senju Pharmaceutical Co Ltd
Tanabe Pharma Corp
Original Assignee
Senju Pharmaceutical Co Ltd
Yoshitomi Pharmaceutical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Senju Pharmaceutical Co Ltd, Yoshitomi Pharmaceutical Industries Ltd filed Critical Senju Pharmaceutical Co Ltd
Application granted granted Critical
Publication of ES2145142T3 publication Critical patent/ES2145142T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62Benzothiazoles
    • C07D277/64Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/12Ophthalmic agents for cataracts
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Ophthalmology & Optometry (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Urology & Nephrology (AREA)
  • Reproductive Health (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

SE PRESENTA UN COMPUESTO DE ACIDO SUCCINAMICO DE LA FORMULA (I) EN DONDE R1 ES ALQUILO O ALQUENILO INFERIOR Y R2 ES UN CARBOXILO OPCIONALMENTE ESTERIFICADO, TAMBIEN SE PRESENTA UNA SAL FARMACOLOGICAMENTE ACEPTABLE DEL COMPUESTO, UN AGENTE PARA LA PROFILAXIS Y/O EL TRATAMIENTO DE LAS COMPLICACIONES DE LA DIABETES, QUE COMPRENDE, COMO INGREDIENTE ACTIVO, EL COMPUESTO DE ACIDO SUCCINAMICO O UNA SAL FARMACOLOGICAMENTE ACEPTABLE DEL MISMO, UN INHIBIDOR DE LA REDUCTASA DE ALDOSA, QUE COMPRENDE, COMO INGREDIENTE ACTIVO EL COMPUESTO DE ACIDO SUCCINAMICO O UNA SAL FARMACOLOGICAMENTE ACEPTABLE DEL MISMO, Y UN METODO PARA PRODUCIR EL COMPUESTO DE ACIDO SUCCINAMICO O UNA SAL FARMACOLOGICAMENTE ACEPTABLE DEL MISMO. LOS NUEVOS COMPUESTOS DEL ACIDO SUCCINAMICO DE LA FORMULA (I) DE LA INVENCION Y LAS SALES FARMACOLOGICAMENTE ACEPTABLES DE LOS MISMOS TIENEN UNA POTENTE ACTIVIDAD INHIBIDORA DE LA REDUCTASA DE ALDOSA EN MAMIFEROS TALES COMO LOS HUMANOS, Y MUESTRAN UNA SUPERIOR SEGURIDAD. POR LO TANTO, SON UTILES COMO AGENTES FARMACOLOGICOS PARA EL TRATAMIENTO DE LAS COMPLICACIONES DE LA DIABETES TALES COMO LA UNION DEFECTUOSA DE LESIONES CORNEALES, LAS CATARATAS, LA NEUROSIS, LA RINOPATIA Y LA NEFROPATIA, EN PARTICULAR, LAS CATARATAS Y LA NEUROSIS. DE ACUERDO CON EL METODO DE PRODUCCION DE LA INVENCION, SE SUMINISTRA UN METODO EFICIENTE DE PRODUCCION DE TALES COMPUESTOS DE LA INVENCION.
ES94921848T 1993-09-14 1994-08-01 Compuesto de acido succinamico, procedimiento para su produccion y su uso. Expired - Lifetime ES2145142T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP5250925A JPH0782259A (ja) 1993-09-14 1993-09-14 スクシンアミド酸誘導体及びそれを含有する糖尿病合併症治療剤

Publications (1)

Publication Number Publication Date
ES2145142T3 true ES2145142T3 (es) 2000-07-01

Family

ID=17215069

Family Applications (1)

Application Number Title Priority Date Filing Date
ES94921848T Expired - Lifetime ES2145142T3 (es) 1993-09-14 1994-08-01 Compuesto de acido succinamico, procedimiento para su produccion y su uso.

Country Status (12)

Country Link
US (1) US5688818A (es)
EP (1) EP0719767B1 (es)
JP (1) JPH0782259A (es)
KR (1) KR960704870A (es)
CN (1) CN1134699A (es)
AT (1) ATE192442T1 (es)
AU (1) AU680670B2 (es)
CA (1) CA2171756A1 (es)
DE (1) DE69424295T2 (es)
ES (1) ES2145142T3 (es)
TW (1) TW324719B (es)
WO (1) WO1995007898A1 (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69902738T2 (de) 1998-01-30 2003-02-06 R-Tech Ueno, Ltd. Ophthalmische zubereitung
US20080233053A1 (en) * 2005-02-07 2008-09-25 Pharmalight Inc. Method and Device for Ophthalmic Administration of Active Pharmaceutical Ingredients
TWI266901B (en) 2005-12-26 2006-11-21 Au Optronics Corp Color filter and method for fabricating the same
MA53706A (fr) 2018-09-25 2021-12-29 Antabio Sas Dérivés d'indane destinés à être utilisés dans le traitement d'une infection bactérienne

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4822809A (en) * 1987-11-13 1989-04-18 Abbott Laboratories Benzazole lipoxygenase inhibiting compounds
JP3126541B2 (ja) * 1993-03-26 2001-01-22 千寿製薬株式会社 ベンゾチアゾール誘導体、その製法及びその用途

Also Published As

Publication number Publication date
EP0719767A1 (en) 1996-07-03
EP0719767A4 (en) 1997-01-08
EP0719767B1 (en) 2000-05-03
DE69424295T2 (de) 2000-10-26
WO1995007898A1 (en) 1995-03-23
US5688818A (en) 1997-11-18
CA2171756A1 (en) 1995-03-23
AU680670B2 (en) 1997-08-07
CN1134699A (zh) 1996-10-30
AU7238994A (en) 1995-04-03
DE69424295D1 (de) 2000-06-08
JPH0782259A (ja) 1995-03-28
ATE192442T1 (de) 2000-05-15
KR960704870A (ko) 1996-10-09
TW324719B (en) 1998-01-11

Similar Documents

Publication Publication Date Title
ES2082805T3 (es) Derivados de tiazol, procedimientos para su produccion y composiciones farmaceuticas que comprenden los mismos.
ATE223378T1 (de) Prolineamid-derivate
NO904202L (no) Terapeutisk aktive bifenylmetanderivater og fremgangsmaatefor deres fremstilling.
DE69320405D1 (de) Ophthalmische Zusammensetzungen enthaltend als Wirkstoff Vitamin-E oder Ester davon
ZA200102067B (en) 2,3-Disubstituted pyridine derivatives, process for the preparation thereof, drug composition containing the same and intermediates for the preparation.
ES2145142T3 (es) Compuesto de acido succinamico, procedimiento para su produccion y su uso.
EA199900374A1 (ru) Ингибитор вторичной катаракты
ES2132394T3 (es) Compuesto de benzotiazol, procedimiento para su produccion, y su utilizacion.
AU695907B2 (en) Pharmaceutical composition for prophylaxis and treatment of type I allergic diseases
AU7424394A (en) 3- or 4-glycosyloxybenzopyran derivatives and antiallergic agents containing the derivatives as active ingredients
EP0644194A4 (en) PYRIDOTHIAZINESSIC ACID DERIVATIVES, METHOD FOR THE PRODUCTION AND USE THEREOF.
ES2130403T3 (es) Derivado del acido quinolin-3-acetico, procedimiento para su produccion, y uso del mismo.
ATE235900T1 (de) Hemmer der subepithelialen turbidität
DE69532963D1 (de) Verwendung von 4-acylaminopyridin derivaten zur Herstellung eines Medikaments für die Behandlung von zerebrovaskulären Erkrankungen
EP0738727A4 (en) 1,4-BENZOXAZINE-2-ACETIC ACID COMPOUND, METHOD FOR THE PRODUCTION AND THEIR USE
ES2061579T3 (es) Compuestos cefem y procedimientos para su preparacion.

Legal Events

Date Code Title Description
FG2A Definitive protection

Ref document number: 719767

Country of ref document: ES