ES2133153T3 - Nuevos depsipeptidos ciclicos con 18 atomos de anillo, y su empleo para el combate de endoparasitos. - Google Patents

Nuevos depsipeptidos ciclicos con 18 atomos de anillo, y su empleo para el combate de endoparasitos.

Info

Publication number
ES2133153T3
ES2133153T3 ES94119130T ES94119130T ES2133153T3 ES 2133153 T3 ES2133153 T3 ES 2133153T3 ES 94119130 T ES94119130 T ES 94119130T ES 94119130 T ES94119130 T ES 94119130T ES 2133153 T3 ES2133153 T3 ES 2133153T3
Authority
ES
Spain
Prior art keywords
depsipeptides
ring atoms
endoparasites
fight
cyclical
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES94119130T
Other languages
English (en)
Inventor
Dr Peter Jeschke
Dr Jurgen Scherkenbeck
Dr Gerhard Bonse
Dr Erwin Bischoff
Dr Norbert Mencke
Dr Dr Achim Harder
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer AG
Original Assignee
Bayer AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer AG filed Critical Bayer AG
Application granted granted Critical
Publication of ES2133153T3 publication Critical patent/ES2133153T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K11/00—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K11/02—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof cyclic, e.g. valinomycins ; Derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D273/00—Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/15—Depsipeptides; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Genetics & Genomics (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

LA INVENCION SE REFIERE A UN NUEVO DEPSIPEPTIDO CICLICO CON 18 ATOMOS DE ANILLO DE LA FORMULA GENERAL (I) EN DONDE R SIGNIFICA HIDROGENO, ALQUIL DE CADENA RECTA O RAMIFICADA O CICLICA CON HASTA 8 ATOMOS DE CARBONO, ASI COMO SUS ISOMEROS OPTICOS Y RACEMATOS. LA INVENCION SE REFIERE TAMBIEN A SU UTILIZACION EN LA LUCHA CONTRA ENDOPARASITOS EN LA ZONA DE MEDICINA Y UTILIZACION VETERINARIA.
ES94119130T 1993-12-16 1994-12-05 Nuevos depsipeptidos ciclicos con 18 atomos de anillo, y su empleo para el combate de endoparasitos. Expired - Lifetime ES2133153T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4342907A DE4342907A1 (de) 1993-12-16 1993-12-16 Neue cyclische Depsipeptide mit 18 Ringatomen und ihre Verwendung zur Bekämpfung von Endoparasiten

Publications (1)

Publication Number Publication Date
ES2133153T3 true ES2133153T3 (es) 1999-09-01

Family

ID=6505168

Family Applications (1)

Application Number Title Priority Date Filing Date
ES94119130T Expired - Lifetime ES2133153T3 (es) 1993-12-16 1994-12-05 Nuevos depsipeptidos ciclicos con 18 atomos de anillo, y su empleo para el combate de endoparasitos.

Country Status (13)

Country Link
US (1) US5624897A (es)
EP (1) EP0658551B1 (es)
JP (1) JP3600287B2 (es)
KR (1) KR100346799B1 (es)
AT (1) ATE180254T1 (es)
AU (1) AU679585B2 (es)
CA (1) CA2137961C (es)
DE (2) DE4342907A1 (es)
DK (1) DK0658551T3 (es)
ES (1) ES2133153T3 (es)
GR (1) GR3030387T3 (es)
TW (1) TW273555B (es)
ZA (1) ZA9410011B (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6458772B1 (en) 1909-10-07 2002-10-01 Medivir Ab Prodrugs
DE4317458A1 (de) * 1992-06-11 1993-12-16 Bayer Ag Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung
US6080719A (en) * 1996-02-23 2000-06-27 Hoechst Aktiengesellschaft Cyclohexapeptides and their mixtures, a process for preparing them, and their use
DE19962145A1 (de) * 1999-12-22 2001-06-28 Bayer Ag Schädlingsbekämpfungsmittel/Depsipeptide
DE19962147A1 (de) * 1999-12-22 2001-06-28 Bayer Ag Schädlingsbekämpfungsmittel / PF 1022-221
DE102008030764A1 (de) * 2008-06-28 2009-12-31 Bayer Animal Health Gmbh Kombination von Amidin-Derivaten mit cyclischen Depsipeptiden
DE102009012423A1 (de) 2009-03-10 2010-09-16 Bayer Animal Health Gmbh Zubereitung auf Ölbasis
DE102010064245A1 (de) 2010-12-28 2012-06-28 Bayer Animal Health Gmbh Makrocylischen Lactone und deren Verwendung und deren Kombinationen mit anderen Wirkstoffen
WO2012028556A1 (en) 2010-08-31 2012-03-08 Bayer Animal Health Gmbh Macrocyclic lactones and their use and their combinations with other active substances
SG11202003272UA (en) * 2017-11-07 2020-05-28 Bayer Animal Health Gmbh Method for the synthesis of cyclic depsipeptides

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1105131B (it) * 1977-06-08 1985-10-28 Merck & Co Inc Peptidi analoghi della somatostatina dotati di piu' lunga e maggiore attivita' biologica e relativo procedimento di protezione
KR930000029B1 (ko) * 1984-03-14 1993-01-06 제롬 꼬르비에르 N-아실 인돌류 활성성분의 용해방법
DE4317458A1 (de) * 1992-06-11 1993-12-16 Bayer Ag Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung

Also Published As

Publication number Publication date
TW273555B (es) 1996-04-01
EP0658551B1 (de) 1999-05-19
CA2137961C (en) 2005-04-12
GR3030387T3 (en) 1999-09-30
KR100346799B1 (ko) 2003-01-06
DE4342907A1 (de) 1995-06-22
DK0658551T3 (da) 1999-11-08
US5624897A (en) 1997-04-29
AU679585B2 (en) 1997-07-03
DE59408281D1 (de) 1999-06-24
AU8041094A (en) 1995-06-22
JP3600287B2 (ja) 2004-12-15
JPH07196687A (ja) 1995-08-01
EP0658551A1 (de) 1995-06-21
CA2137961A1 (en) 1995-06-17
ATE180254T1 (de) 1999-06-15
ZA9410011B (en) 1995-08-24
KR950018047A (ko) 1995-07-22

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