ES2115608T3 - Procedimiento para preparar derivados lactamicos. - Google Patents

Procedimiento para preparar derivados lactamicos.

Info

Publication number
ES2115608T3
ES2115608T3 ES91304642T ES91304642T ES2115608T3 ES 2115608 T3 ES2115608 T3 ES 2115608T3 ES 91304642 T ES91304642 T ES 91304642T ES 91304642 T ES91304642 T ES 91304642T ES 2115608 T3 ES2115608 T3 ES 2115608T3
Authority
ES
Spain
Prior art keywords
compound
formula
lactamic
derivatives
preparing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES91304642T
Other languages
English (en)
Inventor
John William Frank Whitehead
Keith Mills
Ian Harold Coates
Alexander William Oxford
Peter Charles North
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Glaxo Group Ltd
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10676385&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ES2115608(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Application granted granted Critical
Publication of ES2115608T3 publication Critical patent/ES2115608T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/80—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D211/84—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen directly attached to ring carbon atoms
    • C07D211/86—Oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Cephalosporin Compounds (AREA)
  • Physical Or Chemical Processes And Apparatus (AREA)

Abstract

LA INVENCION SE REFIERE A UN PROCESO PARA LA PREPARACION DE UN COMPUESTO DE FORMULA (I) DONDE R REPRESENTA UN ATOMO DE HIDROGENO O UN GRUPO METILO O ETILO, QUE INCLUYE LA CICLACION DE UN COMPUESTO DE FORMULA (IV) DONDE R REPRESENTA UN ATOMO DE HIDROGENO, EL COMPUESTO DE FORMULA (IV) PUEDE ALQUILARSE OPCIONALMENTE PARA PRODUCIR UN COMPUESTO EN EL QUE R SEA METILO O ETILO. EL COMPUESTO DE FORMULA (I) ES UTIL COMO INTERMEDIO EN LA PREPARACION DE 2, 3, 4, 5-TETRAHIDRO-2-[(IMIDAZOL-4(OR5)-IL)METIL]-1H-PIRIDO [4,3-B]INDOL-1-ONAS QUE TIENEN ACTIVIDAD ANTAGONISTA DE 5-HT SUB 3.
ES91304642T 1990-05-23 1991-05-22 Procedimiento para preparar derivados lactamicos. Expired - Lifetime ES2115608T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB909011469A GB9011469D0 (en) 1990-05-23 1990-05-23 Chemical process

Publications (1)

Publication Number Publication Date
ES2115608T3 true ES2115608T3 (es) 1998-07-01

Family

ID=10676385

Family Applications (1)

Application Number Title Priority Date Filing Date
ES91304642T Expired - Lifetime ES2115608T3 (es) 1990-05-23 1991-05-22 Procedimiento para preparar derivados lactamicos.

Country Status (10)

Country Link
US (1) US5196534A (es)
EP (1) EP0458624B1 (es)
JP (1) JP3148281B2 (es)
AT (1) ATE164581T1 (es)
DE (1) DE69129165T2 (es)
DK (1) DK0458624T3 (es)
ES (1) ES2115608T3 (es)
GB (1) GB9011469D0 (es)
HK (1) HK1009647A1 (es)
SG (1) SG43894A1 (es)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH11279040A (ja) * 1998-03-27 1999-10-12 Kao Corp 皮膚外用剤
US6375948B1 (en) 1999-07-12 2002-04-23 Kao Corporation Treating method for suppressing hair growth
CN102617408B (zh) * 2008-07-02 2013-11-27 重庆华邦制药有限公司 氨基酸苄酯衍生物及其中间体
CN101619041B (zh) * 2008-07-02 2012-07-04 重庆华邦制药股份有限公司 一种二酮基含氮环化合物的合成方法及其中间体
US11589583B2 (en) 2013-12-03 2023-02-28 Fmc Corporation Pyrrolidinones herbicides
EP3294743B1 (en) 2015-05-12 2019-08-21 FMC Corporation Aryl substituted bicyclic compounds as herbicides
JP6869192B2 (ja) 2015-05-29 2021-05-12 エフ エム シー コーポレーションＦｍｃ Ｃｏｒｐｏｒａｔｉｏｎ 除草剤としての置換環状アミド
WO2016196593A1 (en) 2015-06-02 2016-12-08 E I Du Pont De Nemours And Company Substituted cyclic amides and their use as herbicides
JP7325328B2 (ja) 2016-12-21 2023-08-14 エフ エム シー コーポレーション ニトロン除草剤
KR102620213B1 (ko) * 2017-03-21 2024-01-03 에프엠씨 코포레이션 피롤리디논 및 이의 제조 방법
WO2018175231A1 (en) 2017-03-21 2018-09-27 Fmc Corporation Herbicidal mixture, composition and method
AR111839A1 (es) 2017-05-30 2019-08-21 Fmc Corp Lactamas 3-sustituidas herbicidas
AR111967A1 (es) 2017-05-30 2019-09-04 Fmc Corp Amidas herbicidas

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3316271A (en) * 1962-10-16 1967-04-25 Hoffmann La Roche 2-methyl-7-alkoxy-1, 2, 3, 4-tetrahydro-5h-pyrid[4, 3-b]indoles and a method for their preparation
DE1695644A1 (de) * 1967-08-08 1971-04-22 Ravensburg Gmbh Chem Fab Verfahren zur Herstellung substituierter 2,4-Dioxopiperidinverbindungen und deren Derivate
US4870180A (en) * 1986-03-17 1989-09-26 Sanofi And Centre National De La Recherche Scientifique 1,2-dihydro-4-methyl-1-oxo-5H-pyrido(4,3-b)indoles and the process for their synthesis
GB2209335B (en) * 1987-09-03 1991-05-29 Glaxo Group Ltd Lactam derivatives
EP0339959A3 (en) * 1988-04-27 1991-03-20 Glaxo Group Limited Lactam derivatives
FI92067C (fi) * 1988-08-02 1994-09-26 Glaxo Group Ltd Menetelmä valmistaa terapeuttisesti aktiivisia mono- tai disubstituoituja (imidatsol-4-yyli)metyylipyrido/4,3-b/indol- ja atsepino/4,3-b/indol-1-oneja
HU204049B (en) * 1989-02-28 1991-11-28 Glaxo Group Ltd Process for producing lactam derivatives and pharmaceutical compositions comprising same

Also Published As

Publication number Publication date
JP3148281B2 (ja) 2001-03-19
HK1009647A1 (en) 1999-06-04
EP0458624B1 (en) 1998-04-01
ATE164581T1 (de) 1998-04-15
US5196534A (en) 1993-03-23
EP0458624A1 (en) 1991-11-27
JPH05117272A (ja) 1993-05-14
DK0458624T3 (da) 1998-10-19
SG43894A1 (en) 1997-11-14
GB9011469D0 (en) 1990-07-11
DE69129165D1 (de) 1998-05-07
DE69129165T2 (de) 1998-07-30

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