ES2063240T3 - Nuevos derivados de acido amino-carboxilico. - Google Patents

Nuevos derivados de acido amino-carboxilico.

Info

Publication number
ES2063240T3
ES2063240T3 ES90200031T ES90200031T ES2063240T3 ES 2063240 T3 ES2063240 T3 ES 2063240T3 ES 90200031 T ES90200031 T ES 90200031T ES 90200031 T ES90200031 T ES 90200031T ES 2063240 T3 ES2063240 T3 ES 2063240T3
Authority
ES
Spain
Prior art keywords
carboxylic acid
amino
new derivatives
group
new
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES90200031T
Other languages
English (en)
Inventor
Jan Verweij
Henri Gerard Julius Hirs
Hendrik Adrianus Witkamp
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Gist Brocades NV
Original Assignee
Gist Brocades NV
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gist Brocades NV filed Critical Gist Brocades NV
Application granted granted Critical
Publication of ES2063240T3 publication Critical patent/ES2063240T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/22—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with radicals containing only hydrogen and carbon atoms, attached in position 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

SE DESCRIBEN NUEVOS DERIVADOS DE ACIDO AMINO CARBOXILICO LOS CUALES COMPRENDEN COMO GRUPO N-TERMINAL, UN GRUPO (CICLO)- ALQUILIDENOAMONICO. TAMBIEN SE DESCUBREN PROCESOS PARA SU PREPARACION Y SU USO COMO PRODUCTOS INTERMEDIOS SINTETICOS.
ES90200031T 1989-01-06 1990-01-04 Nuevos derivados de acido amino-carboxilico. Expired - Lifetime ES2063240T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP89200034 1989-01-06

Publications (1)

Publication Number Publication Date
ES2063240T3 true ES2063240T3 (es) 1995-01-01

Family

ID=8202296

Family Applications (1)

Application Number Title Priority Date Filing Date
ES90200031T Expired - Lifetime ES2063240T3 (es) 1989-01-06 1990-01-04 Nuevos derivados de acido amino-carboxilico.

Country Status (9)

Country Link
EP (1) EP0382268B1 (es)
JP (1) JPH02275885A (es)
KR (1) KR900011777A (es)
AT (1) ATE110385T1 (es)
DE (1) DE69011702T2 (es)
DK (1) DK0382268T3 (es)
ES (1) ES2063240T3 (es)
IE (1) IE65796B1 (es)
TW (1) TW197410B (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103275104B (zh) * 2013-05-15 2015-05-20 苏州明锐医药科技有限公司 头孢托罗及头孢托罗酯的制备方法
CN105601648A (zh) * 2016-03-09 2016-05-25 上海宁瑞生化技术有限公司 一锅法制备头孢吡普的方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3821198A (en) * 1972-05-03 1974-06-28 Squibb & Sons Inc Derivatives of 6-amino penicillanic acid
CA1032533A (en) * 1973-09-07 1978-06-06 William H. Koster Process for the production of cephalosporin compounds
EP0300546B1 (en) * 1987-07-10 1995-08-09 Gist-Brocades N.V. Process for the preparation of cephem compounds and cephalosporin derivatives

Also Published As

Publication number Publication date
EP0382268A1 (en) 1990-08-16
DE69011702D1 (de) 1994-09-29
TW197410B (es) 1993-01-01
KR900011777A (ko) 1990-08-02
IE65796B1 (en) 1995-11-15
DE69011702T2 (de) 1995-04-06
ATE110385T1 (de) 1994-09-15
IE900047L (en) 1990-07-06
EP0382268B1 (en) 1994-08-24
DK0382268T3 (da) 1994-10-24
JPH02275885A (ja) 1990-11-09

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