ES2053580T3 - Derivados de pirido(4,3-d)pirimidina. - Google Patents

Derivados de pirido(4,3-d)pirimidina.

Info

Publication number
ES2053580T3
ES2053580T3 ES87810234T ES87810234T ES2053580T3 ES 2053580 T3 ES2053580 T3 ES 2053580T3 ES 87810234 T ES87810234 T ES 87810234T ES 87810234 T ES87810234 T ES 87810234T ES 2053580 T3 ES2053580 T3 ES 2053580T3
Authority
ES
Spain
Prior art keywords
amino
hydroxy
allergic
alkylamino group
lower alkylamino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES87810234T
Other languages
English (en)
Inventor
Kouichiro Inst Of Bio-Activ Go
Yoshiyuki Inst Of Bio Kurimoto
Norihiko Inst Of Bio- Kitamura
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Nippon Zoki Pharmaceutical Co Ltd
Original Assignee
Nippon Zoki Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nippon Zoki Pharmaceutical Co Ltd filed Critical Nippon Zoki Pharmaceutical Co Ltd
Application granted granted Critical
Publication of ES2053580T3 publication Critical patent/ES2053580T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pulmonology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Immunology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)

Abstract

LA INVENCION SE REFIERE A DERIVADOS DE PIRIDO [4,3-D]PIRIMIDINA QUE TIENEN LA FORMULA GENERAL (I), O A SUS SALES FARMACEUTICAMENTE ACEPTABLES, EN LA QUE R1 Y R2 QUE PUEDEN SER IGUALES O DIFERENTES SON UN GRUPO ALQUILO DE CADENA CORTA; R3 ES H, HALOGENO, OH, AMINO, HIDROXIAMINO, IMINO, HIDRAZINO O UN GRUPO ALQUILAMINO DE CADENA CORTA, QUE PUEDE ESTAR SUSTITUIDO POR OH, AMINO -NH O UN GRUPO ALQUILO DE CADENA CORTA QUE PUEDE ESTAR SUSTITUIDO POR UN GRUPO OH, AMINO O ALQUILAMINO DE CADENA CORTA. ESTOS COMPUESTOS SON UTILES COMO AGENTES ANTIALERGICOS, POR EJEMPLO PARA EL TRATAMIENTO DEL ASMA BRONQUIAL, URTICARIA, RINITIS ALERGICA, DERMATOSIS ALERGICA Y CONJUNTIVITIS ALERGICA.
ES87810234T 1986-04-16 1987-04-10 Derivados de pirido(4,3-d)pirimidina. Expired - Lifetime ES2053580T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP8906586 1986-04-16

Publications (1)

Publication Number Publication Date
ES2053580T3 true ES2053580T3 (es) 1994-08-01

Family

ID=13960451

Family Applications (1)

Application Number Title Priority Date Filing Date
ES87810234T Expired - Lifetime ES2053580T3 (es) 1986-04-16 1987-04-10 Derivados de pirido(4,3-d)pirimidina.

Country Status (6)

Country Link
US (1) US4808618A (es)
EP (1) EP0244352B1 (es)
JP (1) JPH07116188B2 (es)
AT (1) ATE87627T1 (es)
DE (1) DE3785076T2 (es)
ES (1) ES2053580T3 (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9214053D0 (en) * 1992-07-02 1992-08-12 Ici Plc Heterocyclic amides
EP0601322A3 (en) * 1992-10-27 1994-10-12 Nippon Zoki Pharmaceutical Co Adenosine deaminase inhibitor.
EP0958074B1 (de) * 1996-06-07 2001-08-29 SMS Demag AG Giessdüse für dünnbandgiessanlagen
CA3033670A1 (en) * 2016-08-12 2018-02-15 Nanjing Gator Meditech Company, Ltd. Protein kinase regulators
CN109265457A (zh) * 2018-11-01 2019-01-25 中国药科大学 一种利用氧化芳构化构建吡啶并嘧啶二酮骨架的新方法
CN109336884B (zh) * 2018-11-09 2021-02-05 安庆奇创药业有限公司 一种合成曲美替尼关键中间体的方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA762455A (en) * 1962-03-22 1967-07-04 Dr. Karl Thomae Gesellschaft Mit Beschrankter Haftung Pyrido-pyrimidines
JPS5623431B2 (es) * 1973-09-10 1981-05-30
JPS5813550B2 (ja) * 1975-03-15 1983-03-14 ヒサミツセイヤク カブシキガイシヤ シンキナピリド （ ４，３−ｄ ） ピリミジンジオンユウドウタイノセイゾウホウ
JPS5813551B2 (ja) * 1975-03-15 1983-03-14 ヒサミツセイヤク カブシキガイシヤ シンキナピリド （ ４，３−ｄ ） ピリミジンジオンユウドウタイノセイゾウホウ

Also Published As

Publication number Publication date
EP0244352A3 (en) 1989-05-31
JPS6345278A (ja) 1988-02-26
US4808618A (en) 1989-02-28
JPH07116188B2 (ja) 1995-12-13
ATE87627T1 (de) 1993-04-15
EP0244352B1 (en) 1993-03-31
DE3785076D1 (de) 1993-05-06
DE3785076T2 (de) 1993-07-08
EP0244352A2 (en) 1987-11-04

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