ES2002723A6 - Un metodo para preparar indoles o derivados del indol - Google Patents

Un metodo para preparar indoles o derivados del indol

Info

Publication number
ES2002723A6
ES2002723A6 ES8601295A ES8601295A ES2002723A6 ES 2002723 A6 ES2002723 A6 ES 2002723A6 ES 8601295 A ES8601295 A ES 8601295A ES 8601295 A ES8601295 A ES 8601295A ES 2002723 A6 ES2002723 A6 ES 2002723A6
Authority
ES
Spain
Prior art keywords
indoles
indole derivatives
well
coupled via
concerned
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES8601295A
Other languages
English (en)
Inventor
Jan Marcussen
Ulvskov Peter Bjarne
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Danske Sukkerfabrikker AS
Original Assignee
Danske Sukkerfabrikker AS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Danske Sukkerfabrikker AS filed Critical Danske Sukkerfabrikker AS
Publication of ES2002723A6 publication Critical patent/ES2002723A6/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Indole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

UN METODO PARA PREPARAR INDOLES O DERIVADOS DE INDOL, COPULADOS POR LA POSICION 4, 5, 6 O 7, HACIENDO REACCIONAR UN COMPUESTO DE INDOL QUE ESTA SUSTITUIDO CON HIDROXILO EN LA POSICION 4, 5, 6 O 7 DE LA FORMULA II EN QUE LOS SIMBOLOS SE EXPLICAN EN LA MEMORIA DESCRIPTIVA CON UN REACTIVO DE ACTIVACION Y A CONTINUACION O SIMULTANEAMENTE INTRODUCIR UN GRUPO NUCLEOFILO, CONVERTIR OPCIONALMENTE EL COMPUESTO RESULTANTE EN UNO DE SUS DERIVADOS ACTIVOS, TAL COMO UN ESTER ACTIVADO O UN DERIVADO DE TOSILO, TRESILO U OTRO DERIVADO, QUE PUEDE SER UNA PARTE DE UNA REACCION DE SUSTITUCION NUCLEOFILA, O INTRODUCIR TEMPORALMENTE ESTE COMO PARTE DE UN GRUPO ELIMINABLE PARA UNIR COVALENTEMENTE EL GRUPO HIDROXILO INDOLICO AL GRUPO FUNCIONAL, QUE HA DE COPULARSE A EL, POR MEDIO DE UN RESIDUO DE COPULACION.
ES8601295A 1985-08-23 1986-08-22 Un metodo para preparar indoles o derivados del indol Expired ES2002723A6 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DK384085A DK158224C (da) 1985-08-23 1985-08-23 Fremgangsmaade til fremstilling af indolderivater

Publications (1)

Publication Number Publication Date
ES2002723A6 true ES2002723A6 (es) 1988-10-01

Family

ID=8127345

Family Applications (2)

Application Number Title Priority Date Filing Date
ES8601295A Expired ES2002723A6 (es) 1985-08-23 1986-08-22 Un metodo para preparar indoles o derivados del indol
ES8802228A Expired ES2007265A6 (es) 1985-08-23 1988-07-15 Un metodo para preparar conjugados de indol-portador biologicamente activos.

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES8802228A Expired ES2007265A6 (es) 1985-08-23 1988-07-15 Un metodo para preparar conjugados de indol-portador biologicamente activos.

Country Status (7)

Country Link
EP (1) EP0216162A3 (es)
JP (1) JPS62103064A (es)
AU (1) AU590603B2 (es)
DE (1) DE216162T1 (es)
DK (1) DK158224C (es)
ES (2) ES2002723A6 (es)
FI (1) FI87560C (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2332893T3 (es) 1996-08-30 2010-02-15 Upfront Chromatography A/S Aislamiento de inmunoglobulinas.
SE9604487D0 (sv) * 1996-12-05 1996-12-05 Pharmacia & Upjohn Ab An antibody, a derivatized diagnostic marker, an immunoassay utilizing the antibody, and diagnostic method
WO1998047870A1 (en) * 1997-04-24 1998-10-29 American Home Products Corporation Process for the synthesis of 4-[6-(hexylcarbamoyloxy) hexylcarbamoyloxy]-piperidine-1- carboxylic acid 4-phenoxyphenyl ester
AUPP405098A0 (en) * 1998-06-12 1998-07-02 Access Pharmaceuticals Australia Pty Limited Novel methods of preparation of vitamin b12 derivatives suitable for conjugation to pharmaceuticals
KR101275770B1 (ko) * 2009-09-11 2013-06-14 숙명여자대학교산학협력단 ＰＰＡＲα/γ/δ 효능제로 작용하는 알콕시 인돌-3-아세트산 유도체, 이의 제조방법 및 이를 유효성분으로 함유하는 약학적 조성물

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH526542A (de) * 1970-03-12 1972-08-15 Sandoz Ag Verfahren zur Herstellung neuer Indolderivate
US4141987A (en) * 1974-06-05 1979-02-27 Imperial Chemical Industries Limited 1-Aryloxy-3-thenamidoalkylamino-2-propanol derivatives

Also Published As

Publication number Publication date
DE216162T1 (de) 1987-11-26
DK158224B (da) 1990-04-16
ES2007265A6 (es) 1989-06-01
EP0216162A3 (en) 1989-03-15
DK384085A (da) 1987-02-24
FI87560B (fi) 1992-10-15
EP0216162A2 (en) 1987-04-01
DK158224C (da) 1990-09-24
FI863417A0 (fi) 1986-08-22
DK384085D0 (da) 1985-08-23
AU590603B2 (en) 1989-11-09
JPS62103064A (ja) 1987-05-13
FI87560C (fi) 1993-01-25
FI863417A (fi) 1987-02-24
AU6174786A (en) 1987-02-26

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 20001204