EP2661260A4 - Benzimidazolformulierungen mit modifizierter freisetzung - Google Patents

Benzimidazolformulierungen mit modifizierter freisetzung

Info

Publication number
EP2661260A4
EP2661260A4 EP11853533.5A EP11853533A EP2661260A4 EP 2661260 A4 EP2661260 A4 EP 2661260A4 EP 11853533 A EP11853533 A EP 11853533A EP 2661260 A4 EP2661260 A4 EP 2661260A4
Authority
EP
European Patent Office
Prior art keywords
modified release
benzimidazole
formulations
benzimidazole formulations
release
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
EP11853533.5A
Other languages
English (en)
French (fr)
Other versions
EP2661260A2 (de
Inventor
Lingam Meka
Srinivasa Almareddy Reddy
Vagisha Sinha
Hitesh Jogia
Srinivas Arutla
Raviraj Pillai
Rahul Sudhakar Gawande
Prasad Vure
Venkateswarlu Vobalaboina
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Dr Reddys Laboratories Ltd
Dr Reddys Laboratories Inc
Original Assignee
Dr Reddys Laboratories Ltd
Dr Reddys Laboratories Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dr Reddys Laboratories Ltd, Dr Reddys Laboratories Inc filed Critical Dr Reddys Laboratories Ltd
Publication of EP2661260A2 publication Critical patent/EP2661260A2/de
Publication of EP2661260A4 publication Critical patent/EP2661260A4/de
Withdrawn legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5026Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5084Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs

Landscapes

  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
EP11853533.5A 2010-12-29 2011-12-29 Benzimidazolformulierungen mit modifizierter freisetzung Withdrawn EP2661260A4 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IN4013CH2010 2010-12-29
US201161447759P 2011-03-01 2011-03-01
PCT/US2011/067868 WO2012092486A2 (en) 2010-12-29 2011-12-29 Modified release benzimidazole formulations

Publications (2)

Publication Number Publication Date
EP2661260A2 EP2661260A2 (de) 2013-11-13
EP2661260A4 true EP2661260A4 (de) 2014-05-14

Family

ID=46383862

Family Applications (1)

Application Number Title Priority Date Filing Date
EP11853533.5A Withdrawn EP2661260A4 (de) 2010-12-29 2011-12-29 Benzimidazolformulierungen mit modifizierter freisetzung

Country Status (7)

Country Link
EP (1) EP2661260A4 (de)
CN (1) CN103402501A (de)
AU (1) AU2011352037A1 (de)
EA (1) EA201390979A1 (de)
NZ (1) NZ613090A (de)
UA (1) UA112855C2 (de)
WO (1) WO2012092486A2 (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112014009580B1 (pt) * 2011-11-02 2022-03-29 Esteve Pharmaceuticals, S.A Composição farmacêutica de omeprazol
CN105120846B (zh) 2013-02-05 2019-10-18 普渡制药公司 抗篡改的药物制剂
US9539265B2 (en) 2013-03-15 2017-01-10 Aihol Corporation Pharmaceutical formulation containing glycosaminoglycan
WO2014142938A1 (en) * 2013-03-15 2014-09-18 Aihol Corporation Pharmaceutical formulation containing glycosaminoglycan
EP3288556A4 (de) 2015-04-29 2018-09-19 Dexcel Pharma Technologies Ltd. Oral zerfallende zusammensetzungen
US10076494B2 (en) 2016-06-16 2018-09-18 Dexcel Pharma Technologies Ltd. Stable orally disintegrating pharmaceutical compositions
CN112336696B (zh) * 2020-12-01 2022-08-05 苏州中化药品工业有限公司 一种长效脉冲制剂及其制备方法

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20060013868A1 (en) * 2002-10-16 2006-01-19 Yohko Akiyama Controlled release preparation
US20080095853A1 (en) * 2004-11-04 2008-04-24 Niclas Clemmensen Modified Release For Proton Pump Inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20050244497A1 (en) * 1997-11-05 2005-11-03 Wockhardt Limited Delayed delivery system for acid-sensitive drugs
JP4541807B2 (ja) * 2004-09-03 2010-09-08 Okiセミコンダクタ株式会社 半導体素子保持装置および半導体素子の搬送方法
FR2891459B1 (fr) * 2005-09-30 2007-12-28 Flamel Technologies Sa Microparticules a liberation modifiee d'au moins un principe actif et forme galenique orale en comprenant
CN101888828A (zh) * 2007-07-27 2010-11-17 蒂宝制药公司 脉冲胃滞留剂型
US20090214599A1 (en) * 2008-02-21 2009-08-27 Agi Therapeutics Plc Proton pump inhibitor formulations, and methods of preparing and using such formulations

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20060013868A1 (en) * 2002-10-16 2006-01-19 Yohko Akiyama Controlled release preparation
US20080095853A1 (en) * 2004-11-04 2008-04-24 Niclas Clemmensen Modified Release For Proton Pump Inhibitors

Also Published As

Publication number Publication date
CN103402501A (zh) 2013-11-20
UA112855C2 (uk) 2016-11-10
EA201390979A1 (ru) 2013-12-30
WO2012092486A3 (en) 2012-11-01
AU2011352037A1 (en) 2013-08-01
EP2661260A2 (de) 2013-11-13
NZ613090A (en) 2015-11-27
WO2012092486A2 (en) 2012-07-05

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Legal Events

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