EP1206463A4 - FATTY ACID SYNTHASE INHIBITORS - Google Patents
FATTY ACID SYNTHASE INHIBITORSInfo
- Publication number
- EP1206463A4 EP1206463A4 EP00957681A EP00957681A EP1206463A4 EP 1206463 A4 EP1206463 A4 EP 1206463A4 EP 00957681 A EP00957681 A EP 00957681A EP 00957681 A EP00957681 A EP 00957681A EP 1206463 A4 EP1206463 A4 EP 1206463A4
- Authority
- EP
- European Patent Office
- Prior art keywords
- fatty acid
- acid synthase
- synthase inhibitors
- inhibitors
- fatty
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
- C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
- C07D317/62—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to atoms of the carbocyclic ring
- C07D317/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US15027699P | 1999-08-23 | 1999-08-23 | |
PCT/US2000/023073 WO2001014362A1 (en) | 1999-08-23 | 2000-08-23 | Fatty acid synthase inhibitors |
US150276P | 2009-02-05 |
Publications (2)
Publication Number | Publication Date |
---|---|
EP1206463A1 EP1206463A1 (en) | 2002-05-22 |
EP1206463A4 true EP1206463A4 (en) | 2003-01-29 |
Family
ID=22533807
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EP00957681A Withdrawn EP1206463A4 (en) | 1999-08-23 | 2000-08-23 | FATTY ACID SYNTHASE INHIBITORS |
Country Status (4)
Country | Link |
---|---|
EP (1) | EP1206463A4 (ja) |
JP (1) | JP2003507467A (ja) |
AU (1) | AU6926500A (ja) |
WO (1) | WO2001014362A1 (ja) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2002014262A1 (fr) * | 2000-08-11 | 2002-02-21 | Kaken Pharmaceutical Co.,Ltd. | Derives de l'acide 2,3-diphenylpropionique ou leurs sels, medicaments ou inhibiteurs d'adhesion cellulaire en contenant, et leur utilisation |
PT2968316T (pt) | 2013-03-13 | 2019-10-29 | Forma Therapeutics Inc | Derivados de 2-hidroxi-1-{4-[(4-fenilfenil)carbonil]piperazin-1-il}etano-1-ona e compostos relacionados como inibidores da sintase de ácidos gordos (fasn) para o tratamento do cancro |
CN103539668B (zh) * | 2013-10-22 | 2015-07-01 | 山西省化工研究所(有限公司) | 合成对苯二亚甲基双丙二酸二乙酯紫外线吸收剂的工艺 |
TWI767148B (zh) | 2018-10-10 | 2022-06-11 | 美商弗瑪治療公司 | 抑制脂肪酸合成酶(fasn) |
CN113382633A (zh) | 2018-10-29 | 2021-09-10 | 福马治疗股份有限公司 | (4-(2-氟-4-(1-甲基-1H-苯并[d]咪唑-5-基)苯甲酰基)哌嗪-1-基)(1-羟基环丙基)甲酮的固体形式 |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3528977A (en) * | 1966-12-14 | 1970-09-15 | Colgate Palmolive Co | Substituted t-aminophenylalanines |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2137211B1 (ja) * | 1971-05-17 | 1974-08-02 | Bouchara Emile | |
IT1177966B (it) * | 1984-08-14 | 1987-09-03 | Medosan Ind Biochimi | Derivati amidici dell'acido 2-(p-aminobenzil)butirrico e relativi e-steri provvisti di attivita' ipolipidemizzante |
JPH04120040A (ja) * | 1990-09-11 | 1992-04-21 | Sumitomo Chem Co Ltd | 光学活性なフェノール誘導体およびその製造法 |
JPH04124158A (ja) * | 1990-09-12 | 1992-04-24 | Sumitomo Chem Co Ltd | 光学活性なフェノール誘導体およびその製造法 |
US5614551A (en) * | 1994-01-24 | 1997-03-25 | The Johns Hopkins University | Inhibitors of fatty acid synthesis as antimicrobial agents |
-
2000
- 2000-08-23 WO PCT/US2000/023073 patent/WO2001014362A1/en not_active Application Discontinuation
- 2000-08-23 AU AU69265/00A patent/AU6926500A/en not_active Abandoned
- 2000-08-23 EP EP00957681A patent/EP1206463A4/en not_active Withdrawn
- 2000-08-23 JP JP2001518449A patent/JP2003507467A/ja not_active Withdrawn
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3528977A (en) * | 1966-12-14 | 1970-09-15 | Colgate Palmolive Co | Substituted t-aminophenylalanines |
Non-Patent Citations (1)
Title |
---|
See also references of WO0114362A1 * |
Also Published As
Publication number | Publication date |
---|---|
JP2003507467A (ja) | 2003-02-25 |
AU6926500A (en) | 2001-03-19 |
WO2001014362A1 (en) | 2001-03-01 |
EP1206463A1 (en) | 2002-05-22 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PUAI | Public reference made under article 153(3) epc to a published international application that has entered the european phase |
Free format text: ORIGINAL CODE: 0009012 |
|
17P | Request for examination filed |
Effective date: 20020304 |
|
AX | Request for extension of the european patent |
Free format text: AL;LT;LV;MK;RO;SI |
|
A4 | Supplementary search report drawn up and despatched |
Effective date: 20021212 |
|
RIC1 | Information provided on ipc code assigned before grant |
Ipc: 7C 07D 315/00 A Ipc: 7C 07D 229/00 B Ipc: 7A 61K 31/19 B Ipc: 7C 07D 317/00 B Ipc: 7C 07D 317/68 B Ipc: 7C 07D 317/14 B |
|
STAA | Information on the status of an ep patent application or granted ep patent |
Free format text: STATUS: THE APPLICATION IS DEEMED TO BE WITHDRAWN |
|
18D | Application deemed to be withdrawn |
Effective date: 20040302 |