EP0971947A4 - Verbinder auf der basis von rink-chlorid für die synthese von organischen molekülen in der organischen festphase - Google Patents

Verbinder auf der basis von rink-chlorid für die synthese von organischen molekülen in der organischen festphase

Info

Publication number
EP0971947A4
EP0971947A4 EP98913115A EP98913115A EP0971947A4 EP 0971947 A4 EP0971947 A4 EP 0971947A4 EP 98913115 A EP98913115 A EP 98913115A EP 98913115 A EP98913115 A EP 98913115A EP 0971947 A4 EP0971947 A4 EP 0971947A4
Authority
EP
European Patent Office
Prior art keywords
rink
solid phase
organic synthesis
chloride linker
organic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
EP98913115A
Other languages
English (en)
French (fr)
Other versions
EP0971947A2 (de
Inventor
Ravi S Garigipati
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SmithKline Beecham Corp
Original Assignee
SmithKline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by SmithKline Beecham Corp filed Critical SmithKline Beecham Corp
Publication of EP0971947A2 publication Critical patent/EP0971947A2/de
Publication of EP0971947A4 publication Critical patent/EP0971947A4/de
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/04—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers
    • C07K1/045—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers using devices to improve synthesis, e.g. reactors, special vessels

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Analytical Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
  • Peptides Or Proteins (AREA)
  • Other Resins Obtained By Reactions Not Involving Carbon-To-Carbon Unsaturated Bonds (AREA)
EP98913115A 1997-03-28 1998-03-26 Verbinder auf der basis von rink-chlorid für die synthese von organischen molekülen in der organischen festphase Withdrawn EP0971947A4 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US4469697P 1997-03-28 1997-03-28
PCT/US1998/005860 WO1998044329A2 (en) 1997-03-28 1998-03-26 Rink-chloride linker for solid phase organic synthesis of organic molecules
US44696P 2008-04-14

Publications (2)

Publication Number Publication Date
EP0971947A2 EP0971947A2 (de) 2000-01-19
EP0971947A4 true EP0971947A4 (de) 2005-01-26

Family

ID=21933821

Family Applications (1)

Application Number Title Priority Date Filing Date
EP98913115A Withdrawn EP0971947A4 (de) 1997-03-28 1998-03-26 Verbinder auf der basis von rink-chlorid für die synthese von organischen molekülen in der organischen festphase

Country Status (4)

Country Link
EP (1) EP0971947A4 (de)
JP (1) JP2001518946A (de)
CA (1) CA2285175A1 (de)
WO (1) WO1998044329A2 (de)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MXPA03006228A (es) 2001-01-12 2004-12-06 Amersham Plc Haluros de perfluoro sulfonilo y especies relacionadas como modificadores de soporte de polimero.

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH05271332A (ja) * 1992-03-30 1993-10-19 Nippon Steel Chem Co Ltd アミノ基を有するスチレン系ポリマーの製造法
US5268423A (en) * 1992-02-28 1993-12-07 New York University Method for preparation of peptide synthesis resins and peptide synthesis resins
EP0687691A2 (de) * 1990-08-31 1995-12-20 Regents Of The University Of Minnesota Harze für die Feststoff-Peptidsynthese und Verfahren zur Herstellung davon
GB2297551A (en) * 1995-02-04 1996-08-07 Zeneca Ltd Labelled chemical library

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU4779493A (en) * 1992-07-21 1994-02-14 Bunsen Rush Laboratories Inc. Oligomer library formats and methods relating thereto
US5684130A (en) * 1995-06-05 1997-11-04 Solid Phase Sciences Corporation Process for synthesis of organic compounds using magnetic particles

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0687691A2 (de) * 1990-08-31 1995-12-20 Regents Of The University Of Minnesota Harze für die Feststoff-Peptidsynthese und Verfahren zur Herstellung davon
US5268423A (en) * 1992-02-28 1993-12-07 New York University Method for preparation of peptide synthesis resins and peptide synthesis resins
JPH05271332A (ja) * 1992-03-30 1993-10-19 Nippon Steel Chem Co Ltd アミノ基を有するスチレン系ポリマーの製造法
GB2297551A (en) * 1995-02-04 1996-08-07 Zeneca Ltd Labelled chemical library

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
DATABASE WPI Section Ch Week 199346, Derwent World Patents Index; Class A13, AN 1993-365270, XP002308412 *
See also references of WO9844329A3 *

Also Published As

Publication number Publication date
WO1998044329A2 (en) 1998-10-08
JP2001518946A (ja) 2001-10-16
EP0971947A2 (de) 2000-01-19
WO1998044329A3 (en) 1998-12-03
CA2285175A1 (en) 1998-10-08

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