AU3894800A - Solid phase synthesis of benzodiazepine diones - Google Patents

Solid phase synthesis of benzodiazepine diones

Info

Publication number
AU3894800A
AU3894800A AU38948/00A AU3894800A AU3894800A AU 3894800 A AU3894800 A AU 3894800A AU 38948/00 A AU38948/00 A AU 38948/00A AU 3894800 A AU3894800 A AU 3894800A AU 3894800 A AU3894800 A AU 3894800A
Authority
AU
Australia
Prior art keywords
diones
benzodiazepine
solid phase
phase synthesis
synthesis
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU38948/00A
Inventor
Jeffrey Mark Dener
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Axys Pharmaceuticals Inc
Original Assignee
Axys Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Axys Pharmaceuticals Inc filed Critical Axys Pharmaceuticals Inc
Publication of AU3894800A publication Critical patent/AU3894800A/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06—Esters of carbamic acids
    • C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
    • C07C271/26—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atom of at least one of the carbamate groups bound to a carbon atom of a six-membered aromatic ring
    • C07C271/28—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atom of at least one of the carbamate groups bound to a carbon atom of a six-membered aromatic ring to a carbon atom of a non-condensed six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/16—Systems containing only non-condensed rings with a six-membered ring the ring being unsaturated
    • C—CHEMISTRY; METALLURGY
    • C40—COMBINATORIAL TECHNOLOGY
    • C40B—COMBINATORIAL CHEMISTRY; LIBRARIES, e.g. CHEMICAL LIBRARIES
    • C40B40/00—Libraries per se, e.g. arrays, mixtures

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU38948/00A 1999-03-23 2000-03-16 Solid phase synthesis of benzodiazepine diones Abandoned AU3894800A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US12568499P 1999-03-23 1999-03-23
US60125684 1999-03-23
PCT/US2000/007117 WO2000056721A1 (en) 1999-03-23 2000-03-16 Solid phase synthesis of benzodiazepine diones

Publications (1)

Publication Number Publication Date
AU3894800A true AU3894800A (en) 2000-10-09

Family

ID=22420923

Family Applications (1)

Application Number Title Priority Date Filing Date
AU38948/00A Abandoned AU3894800A (en) 1999-03-23 2000-03-16 Solid phase synthesis of benzodiazepine diones

Country Status (2)

Country Link
AU (1) AU3894800A (en)
WO (1) WO2000056721A1 (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN100365633C (en) 2000-09-30 2008-01-30 世嘉股份有限公司 Service ticket issuing system and service ticket issuing service
AU2002340464B2 (en) 2001-11-13 2008-03-13 3-Dimensional Pharmaceuticals, Inc. Substituted 1,4-benzodiazepines and uses thereof for the treatment of cancer
AU2005272627A1 (en) 2004-08-13 2006-02-23 Amgen Inc. Substituted benzofused heterocycles

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA924760B (en) * 1991-06-28 1993-03-31 Smithkline Beecham Corp Bicyclic fibrinogen antagonists
US5288514A (en) * 1992-09-14 1994-02-22 The Regents Of The University Of California Solid phase and combinatorial synthesis of benzodiazepine compounds on a solid support
US5702672A (en) * 1992-10-08 1997-12-30 Warner-Lambert Company Apparatus and method for multiple simultaneous synthesis
US5817751A (en) * 1994-06-23 1998-10-06 Affymax Technologies N.V. Method for synthesis of diketopiperazine and diketomorpholine derivatives
CN1173946C (en) * 1998-01-29 2004-11-03 阿温蒂斯药物公司 Method for preparing an N-[(aliphatic or aromatic) carbonyl]-2-aminoacetamide compound and a cyclyzed compound

Also Published As

Publication number Publication date
WO2000056721A1 (en) 2000-09-28

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Legal Events

Date Code Title Description
MK6 Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase