EP0649443A4 - Matieres derivees d'oxazolone. - Google Patents
Matieres derivees d'oxazolone.Info
- Publication number
- EP0649443A4 EP0649443A4 EP93916883A EP93916883A EP0649443A4 EP 0649443 A4 EP0649443 A4 EP 0649443A4 EP 93916883 A EP93916883 A EP 93916883A EP 93916883 A EP93916883 A EP 93916883A EP 0649443 A4 EP0649443 A4 EP 0649443A4
- Authority
- EP
- European Patent Office
- Prior art keywords
- oxazolone
- derived materials
- derived
- materials
- oxazolone derived
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H21/00—Compounds containing two or more mononucleotide units having separate phosphate or polyphosphate groups linked by saccharide radicals of nucleoside groups, e.g. nucleic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C229/34—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
- C07C229/36—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings with at least one amino group and one carboxyl group bound to the same carbon atom of the carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
- C07C237/02—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton
- C07C237/22—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton having nitrogen atoms of amino groups bound to the carbon skeleton of the acid part, further acylated
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/36—One oxygen atom
- C07D263/42—One oxygen atom attached in position 5
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/04—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers
- C07K1/047—Simultaneous synthesis of different peptide species; Peptide libraries
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/001—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof by chemical synthesis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/46—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
- C07K14/47—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
- C07K14/4701—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals not used
- C07K14/4702—Regulators; Modulating activity
- C07K14/4703—Inhibitors; Suppressors
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
- C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
- C07K5/0222—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/02—Linear peptides containing at least one abnormal peptide link
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Medicinal Chemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Biophysics (AREA)
- Gastroenterology & Hepatology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Virology (AREA)
- Veterinary Medicine (AREA)
- Oncology (AREA)
- Analytical Chemistry (AREA)
- Biotechnology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Communicable Diseases (AREA)
- Toxicology (AREA)
- Zoology (AREA)
- Engineering & Computer Science (AREA)
- Peptides Or Proteins (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US90675692A | 1992-06-30 | 1992-06-30 | |
US906756 | 1992-06-30 | ||
US4156293A | 1993-04-02 | 1993-04-02 | |
US41562 | 1993-04-02 | ||
PCT/US1993/006240 WO1994000509A1 (fr) | 1992-06-30 | 1993-06-30 | Matieres derivees d'oxazolone |
Publications (2)
Publication Number | Publication Date |
---|---|
EP0649443A1 EP0649443A1 (fr) | 1995-04-26 |
EP0649443A4 true EP0649443A4 (fr) | 1995-11-08 |
Family
ID=26718293
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EP93916883A Ceased EP0649443A4 (fr) | 1992-06-30 | 1993-06-30 | Matieres derivees d'oxazolone. |
Country Status (7)
Country | Link |
---|---|
EP (1) | EP0649443A4 (fr) |
JP (1) | JPH08500576A (fr) |
KR (1) | KR950702216A (fr) |
AU (1) | AU678168B2 (fr) |
BR (1) | BR9306656A (fr) |
CA (1) | CA2139350A1 (fr) |
WO (1) | WO1994000509A1 (fr) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0738155A4 (fr) * | 1993-12-28 | 1997-03-19 | Arqule Partners L P | Structure et synthese modulaire de molecules derivees de l'oxazolone |
JPH09507852A (ja) * | 1994-01-05 | 1997-08-12 | アーキュール,インコーポレーテッド | 特定の性質を有するポリマーの製造方法 |
DE19714343A1 (de) * | 1997-04-08 | 1998-10-15 | Bayer Ag | Chromatographische Enantiomerentrennung von Lactonen |
GB9812675D0 (en) * | 1998-06-11 | 1998-08-12 | Univ Edinburgh | Peptides |
WO2000064845A1 (fr) * | 1999-04-22 | 2000-11-02 | Sankyo Company, Limited | Cetoamides porteurs de resine et leur procede de preparation |
EP2113510A1 (fr) * | 2008-04-30 | 2009-11-04 | Freie Universität Berlin | Dérivés de pepstatine A |
CN112898218B (zh) * | 2020-01-14 | 2022-08-26 | 河南师范大学 | 一锅法合成含三氟甲基噁唑酮类化合物的方法 |
CN112830882A (zh) * | 2020-12-31 | 2021-05-25 | 河南绿园药业有限公司 | 一种对羟基苯甘氨酸甲酯合成方法 |
Citations (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2391191A1 (fr) * | 1977-05-16 | 1978-12-15 | Sandoz Sa | Nouveaux composes polypeptidiques, lyeptidiques, leur preparation et leur application comme medicaments |
EP0008097A2 (fr) * | 1978-08-07 | 1980-02-20 | BASF Aktiengesellschaft | Procédé de préparation d'indolénines |
EP0105665A1 (fr) * | 1982-09-27 | 1984-04-18 | Minnesota Mining And Manufacturing Company | Composés contenant le groupement fonctionnel azlactone et compositions durcissables les contenant |
EP0328340A2 (fr) * | 1988-02-09 | 1989-08-16 | BAUSCH & LOMB INCORPORATED | Polymères hydrophiles perméables à l'oxygène |
EP0433034A2 (fr) * | 1989-12-12 | 1991-06-19 | Minnesota Mining And Manufacturing Company | Méthode impliquant liaisons alpha-amidoacétyles ou béta-amidopropionyles thermosensibles |
EP0449488A1 (fr) * | 1990-03-28 | 1991-10-02 | Minnesota Mining And Manufacturing Company | Produits d'addition Michael des azlactones |
EP0525420A1 (fr) * | 1991-07-01 | 1993-02-03 | Mitsubishi Chemical Corporation | Pseudopeptides et peptides caractérisés par une partie méthyle cétone substituée à la terminaison C comme inhibiteurs de thiol protéase |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4125519A (en) * | 1976-10-13 | 1978-11-14 | Murray Goodman | Polypeptides containing 3,4-dihydroxyphenylalanine |
JPS60215657A (ja) * | 1984-04-10 | 1985-10-29 | Mitsui Toatsu Chem Inc | N−アシルフエニルアラニン類の製造法 |
US4996292A (en) * | 1989-06-30 | 1991-02-26 | Fox Sidney W | Self-sealing artificial skin comprising copoly-alpha-amino acid |
US5039813A (en) * | 1990-06-29 | 1991-08-13 | Polaroid Corporation | 2-(4-alkenylphenyl)-5-oxazolones and polymers thereof |
US5219731A (en) * | 1991-11-01 | 1993-06-15 | Wisconsin Alumni Research Foundation | Method for preparing optically-active amino acid derivatives |
-
1993
- 1993-06-30 BR BR9306656A patent/BR9306656A/pt not_active Application Discontinuation
- 1993-06-30 WO PCT/US1993/006240 patent/WO1994000509A1/fr not_active Application Discontinuation
- 1993-06-30 CA CA002139350A patent/CA2139350A1/fr not_active Abandoned
- 1993-06-30 JP JP6502661A patent/JPH08500576A/ja active Pending
- 1993-06-30 KR KR1019940704824A patent/KR950702216A/ko not_active Application Discontinuation
- 1993-06-30 EP EP93916883A patent/EP0649443A4/fr not_active Ceased
- 1993-06-30 AU AU46591/93A patent/AU678168B2/en not_active Ceased
Patent Citations (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2391191A1 (fr) * | 1977-05-16 | 1978-12-15 | Sandoz Sa | Nouveaux composes polypeptidiques, lyeptidiques, leur preparation et leur application comme medicaments |
EP0008097A2 (fr) * | 1978-08-07 | 1980-02-20 | BASF Aktiengesellschaft | Procédé de préparation d'indolénines |
EP0105665A1 (fr) * | 1982-09-27 | 1984-04-18 | Minnesota Mining And Manufacturing Company | Composés contenant le groupement fonctionnel azlactone et compositions durcissables les contenant |
EP0328340A2 (fr) * | 1988-02-09 | 1989-08-16 | BAUSCH & LOMB INCORPORATED | Polymères hydrophiles perméables à l'oxygène |
EP0433034A2 (fr) * | 1989-12-12 | 1991-06-19 | Minnesota Mining And Manufacturing Company | Méthode impliquant liaisons alpha-amidoacétyles ou béta-amidopropionyles thermosensibles |
EP0449488A1 (fr) * | 1990-03-28 | 1991-10-02 | Minnesota Mining And Manufacturing Company | Produits d'addition Michael des azlactones |
EP0525420A1 (fr) * | 1991-07-01 | 1993-02-03 | Mitsubishi Chemical Corporation | Pseudopeptides et peptides caractérisés par une partie méthyle cétone substituée à la terminaison C comme inhibiteurs de thiol protéase |
Non-Patent Citations (1)
Title |
---|
See also references of WO9400509A1 * |
Also Published As
Publication number | Publication date |
---|---|
AU678168B2 (en) | 1997-05-22 |
JPH08500576A (ja) | 1996-01-23 |
KR950702216A (ko) | 1995-06-19 |
AU4659193A (en) | 1994-01-24 |
CA2139350A1 (fr) | 1994-01-06 |
WO1994000509A1 (fr) | 1994-01-06 |
EP0649443A1 (fr) | 1995-04-26 |
BR9306656A (pt) | 1998-12-08 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
EP0597463A3 (en) | Thermotherapiesonde. | |
EP0580285A3 (fr) | Auto-réenclencheurs. | |
EP0670716A4 (fr) | Substances pharmaceutiques au gout camoufle. | |
GB9311790D0 (en) | Photothermographic materials | |
EP0633771A4 (en) | Compounds. | |
EP0572808A3 (fr) | Système de régulation antiblocage. | |
EP0586828A3 (fr) | Hydrophone. | |
EP0668864A4 (fr) | Biphenylmethylimidazopyridines substituees. | |
EP0649443A4 (fr) | Matieres derivees d'oxazolone. | |
GB2263953B (en) | The radial change multigear | |
ZA929724B (en) | Ballisitc materials. | |
EP0599191A3 (fr) | Circuit de régulation de vitesse d'un moteur. | |
EP0592354A3 (fr) | Centrifugeuse à vide. | |
EP0586706A4 (fr) | Ensemble d'injection. | |
EP0601762A3 (fr) | Matériau de frottement. | |
EP0663819A4 (fr) | Association d'ibuprofene et de cafeine. | |
ZA934353B (en) | Linear peptides. | |
ZA919371B (en) | Containers. | |
ZA935828B (en) | New insobutyl-substituted methanesulphonyl-quinolyl-methoxyphenyl-cycloalkylacetamides. | |
ZA931036B (en) | Containers. | |
GB9221450D0 (en) | The wropod | |
ZA931403B (en) | Sulphonamidocarboxamides. | |
GB9200646D0 (en) | Silicate-carbonate materials | |
GB9200539D0 (en) | Silicate-carbonate materials | |
GB9200286D0 (en) | Silicate-carbonate materials |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
PUAI | Public reference made under article 153(3) epc to a published international application that has entered the european phase |
Free format text: ORIGINAL CODE: 0009012 |
|
17P | Request for examination filed |
Effective date: 19950130 |
|
AK | Designated contracting states |
Kind code of ref document: A1 Designated state(s): AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE |
|
A4 | Supplementary search report drawn up and despatched |
Effective date: 19950922 |
|
AK | Designated contracting states |
Kind code of ref document: A4 Designated state(s): AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE |
|
17Q | First examination report despatched |
Effective date: 19970404 |
|
RAP1 | Party data changed (applicant data changed or rights of an application transferred) |
Owner name: ARQULE PARTNERS, L.P. |
|
RAP1 | Party data changed (applicant data changed or rights of an application transferred) |
Owner name: ARQULE, INC. |
|
STAA | Information on the status of an ep patent application or granted ep patent |
Free format text: STATUS: THE APPLICATION HAS BEEN REFUSED |
|
18R | Application refused |
Effective date: 20001012 |