EE9400115A - 3- (asendatud tetrasolüül)- 4- okso- 4H- pürido[1,2- a] pürimidiinid, nende soolad, neid sisaldavad farmatseutilised segud ja nende valmistamise protsess - Google Patents

3- (asendatud tetrasolüül)- 4- okso- 4H- pürido[1,2- a] pürimidiinid, nende soolad, neid sisaldavad farmatseutilised segud ja nende valmistamise protsess

Info

Publication number
EE9400115A
EE9400115A EE9400115A EE9400115A EE9400115A EE 9400115 A EE9400115 A EE 9400115A EE 9400115 A EE9400115 A EE 9400115A EE 9400115 A EE9400115 A EE 9400115A EE 9400115 A EE9400115 A EE 9400115A
Authority
EE
Estonia
Prior art keywords
pyrido
pyrimidines
oxo
salts
preparation
Prior art date
Application number
EE9400115A
Other languages
English (en)
Estonian (et)
Inventor
Hermecz István
Knoll József
Sipos Judit
Gyires Klára
Horváth Ágnes
Vasvári Lelle
Tardos László
Balogh Mária
Kapui Zoltán
Papp Ilona
Original Assignee
Chinoin Gyógyszer és Vegyészeti Termékek Gyára Rt.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyógyszer és Vegyészeti Termékek Gyára Rt. filed Critical Chinoin Gyógyszer és Vegyészeti Termékek Gyára Rt.
Publication of EE9400115A publication Critical patent/EE9400115A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
EE9400115A 1990-09-25 1994-08-10 3- (asendatud tetrasolüül)- 4- okso- 4H- pürido[1,2- a] pürimidiinid, nende soolad, neid sisaldavad farmatseutilised segud ja nende valmistamise protsess EE9400115A (et)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU620590A HU209793B (en) 1990-09-25 1990-09-25 Process for the production of pyrido[1,2-a]pyrimidine-derivatives and pharmaceutical compositions containing the same

Publications (1)

Publication Number Publication Date
EE9400115A true EE9400115A (et) 1995-12-15

Family

ID=10971360

Family Applications (1)

Application Number Title Priority Date Filing Date
EE9400115A EE9400115A (et) 1990-09-25 1994-08-10 3- (asendatud tetrasolüül)- 4- okso- 4H- pürido[1,2- a] pürimidiinid, nende soolad, neid sisaldavad farmatseutilised segud ja nende valmistamise protsess

Country Status (19)

Country Link
US (1) US5475000A (zh)
EP (1) EP0641340A1 (zh)
JP (1) JPH06509800A (zh)
CN (1) CN1071925A (zh)
AU (1) AU663886B2 (zh)
BG (1) BG98448A (zh)
CA (1) CA2114145A1 (zh)
CZ (1) CZ27694A3 (zh)
EE (1) EE9400115A (zh)
FI (1) FI940591A0 (zh)
HU (1) HU209793B (zh)
IL (1) IL102788A (zh)
MX (1) MX9204659A (zh)
PT (1) PT100774A (zh)
SI (1) SI9200172A (zh)
SK (1) SK16594A3 (zh)
TW (1) TW222632B (zh)
WO (1) WO1993004065A1 (zh)
YU (1) YU76092A (zh)

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3055911A (en) * 1958-04-29 1962-09-25 William G Finnegan Substituted tetrazoles
US4122274A (en) * 1977-05-25 1978-10-24 Bristol-Myers Company 3-Tetrazolo-5,6,7,8-substituted-pyrido[1,2-a]pyrimidin-4-ones
JPS5536447A (en) * 1978-09-07 1980-03-14 Otsuka Pharmaceut Co Ltd Butyramide derivative
US4474792A (en) * 1979-06-18 1984-10-02 Riker Laboratories, Inc. N-Tetrazolyl benzamides and anti-allergic use thereof
US4432986A (en) * 1979-06-18 1984-02-21 Riker Laboratories, Inc. Tetrazoles bonded to certain polycyclic aromatic systems and anti-allergic use thereof
FI73423C (fi) * 1980-02-29 1987-10-09 Otsuka Pharma Co Ltd Foerfarande foer framstaellning av farmakologiskt verksamma tetrazolderivat.
US4457932A (en) * 1983-07-22 1984-07-03 Bristol-Myers Company Anti-ulcer agents
FR2549831A1 (fr) * 1983-07-27 1985-02-01 Rhone Poulenc Agrochimie Nouveaux derives d'acides aryloxybenzoiques, et leur utilisation comme herbicides
US4845227A (en) * 1984-06-18 1989-07-04 Eli Lilly And Company Aromatase inhibitors from azoles
US5237070A (en) * 1985-07-22 1993-08-17 Riker Laboratories, Inc. Substituted DI-t-butylphenols
US5049572A (en) * 1987-04-06 1991-09-17 Riker Laboratories, Inc. Substituted di-t-butylphenols and anti-allergic use thereof
JP2668259B2 (ja) * 1988-02-18 1997-10-27 塩野義製薬株式会社 複素環化合物および抗潰瘍剤
HUT64064A (en) * 1992-02-13 1993-11-29 Chinoin Gyogyszer Es Vegyeszet Process for producing puyrido/1,2-a/pyrimidine derivatives and pharmaceutical compositions comprising same as active ingredient

Also Published As

Publication number Publication date
AU2462892A (en) 1993-03-16
HU906205D0 (en) 1991-03-28
BG98448A (en) 1994-11-15
CZ27694A3 (en) 1994-08-17
MX9204659A (es) 1993-12-31
HUT64954A (en) 1994-03-28
WO1993004065A1 (en) 1993-03-04
US5475000A (en) 1995-12-12
YU76092A (sr) 1996-01-09
JPH06509800A (ja) 1994-11-02
TW222632B (zh) 1994-04-21
CN1071925A (zh) 1993-05-12
FI940591A (fi) 1994-02-09
FI940591A0 (fi) 1994-02-09
EP0641340A1 (en) 1995-03-08
AU663886B2 (en) 1995-10-26
IL102788A (en) 1996-03-31
HU209793B (en) 1994-11-28
SI9200172A (en) 1993-03-31
SK16594A3 (en) 1994-08-10
CA2114145A1 (en) 1993-03-04
PT100774A (pt) 1993-10-29

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