ECSP17075052A - Tableta de Ribociclib - Google Patents

Tableta de Ribociclib

Info

Publication number
ECSP17075052A
ECSP17075052A ECIEPI201775052A ECPI201775052A ECSP17075052A EC SP17075052 A ECSP17075052 A EC SP17075052A EC IEPI201775052 A ECIEPI201775052 A EC IEPI201775052A EC PI201775052 A ECPI201775052 A EC PI201775052A EC SP17075052 A ECSP17075052 A EC SP17075052A
Authority
EC
Ecuador
Prior art keywords
ribociclib
tablet
coating
present disclosure
coated
Prior art date
Application number
ECIEPI201775052A
Other languages
English (en)
Spanish (es)
Inventor
Grandeury Arnaud
Gururajan Bindhumadhavan
Costa Rui
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=55806565&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ECSP17075052(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of ECSP17075052A publication Critical patent/ECSP17075052A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ECIEPI201775052A 2015-04-16 2017-11-10 Tableta de Ribociclib ECSP17075052A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201562148240P 2015-04-16 2015-04-16

Publications (1)

Publication Number Publication Date
ECSP17075052A true ECSP17075052A (es) 2018-02-28

Family

ID=55806565

Family Applications (1)

Application Number Title Priority Date Filing Date
ECIEPI201775052A ECSP17075052A (es) 2015-04-16 2017-11-10 Tableta de Ribociclib

Country Status (29)

Country Link
US (6) US10799506B2 (cg-RX-API-DMAC7.html)
EP (3) EP4620458A3 (cg-RX-API-DMAC7.html)
JP (1) JP2018514523A (cg-RX-API-DMAC7.html)
KR (2) KR20250009572A (cg-RX-API-DMAC7.html)
CN (2) CN107530292B (cg-RX-API-DMAC7.html)
AR (1) AR104257A1 (cg-RX-API-DMAC7.html)
AU (5) AU2016248017A1 (cg-RX-API-DMAC7.html)
BR (1) BR112017021283A2 (cg-RX-API-DMAC7.html)
CA (1) CA2982425C (cg-RX-API-DMAC7.html)
CL (1) CL2017002593A1 (cg-RX-API-DMAC7.html)
CO (1) CO2017010510A2 (cg-RX-API-DMAC7.html)
DK (1) DK3283058T3 (cg-RX-API-DMAC7.html)
EA (1) EA201792290A1 (cg-RX-API-DMAC7.html)
EC (1) ECSP17075052A (cg-RX-API-DMAC7.html)
ES (1) ES2938261T3 (cg-RX-API-DMAC7.html)
FI (1) FI3283058T3 (cg-RX-API-DMAC7.html)
HR (1) HRP20230053T1 (cg-RX-API-DMAC7.html)
HU (1) HUE061213T2 (cg-RX-API-DMAC7.html)
IL (1) IL254818A0 (cg-RX-API-DMAC7.html)
MX (1) MX2017013350A (cg-RX-API-DMAC7.html)
PE (1) PE20180035A1 (cg-RX-API-DMAC7.html)
PH (1) PH12017501820A1 (cg-RX-API-DMAC7.html)
PL (1) PL3283058T3 (cg-RX-API-DMAC7.html)
PT (1) PT3283058T (cg-RX-API-DMAC7.html)
SG (1) SG11201708084PA (cg-RX-API-DMAC7.html)
SI (1) SI3283058T1 (cg-RX-API-DMAC7.html)
TN (1) TN2017000422A1 (cg-RX-API-DMAC7.html)
TW (1) TW201642864A (cg-RX-API-DMAC7.html)
WO (1) WO2016166703A1 (cg-RX-API-DMAC7.html)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2017013350A (es) * 2015-04-16 2018-01-25 Novartis Ag Comprimido de ribociclib.
CA3048036A1 (en) 2018-07-02 2020-01-02 Apotex Inc Novel crystalline form of ribociclib succinate
AU2020336309A1 (en) 2019-08-26 2022-03-17 Arvinas Operations, Inc. Methods of treating breast cancer with tetrahydronaphthalene derivatives as estrogen receptor degraders
CR20220342A (es) 2019-12-16 2023-01-23 Lunella Biotech Inc Agentes terapéuticos selectivos contra el cáncer inhibidores cdk4/6
US12358920B2 (en) 2019-12-16 2025-07-15 Lunella Biotech, Inc. Substituted pyrrolo[2,3-d]pyrimidines as selective CDK 4/6 inhibitors
BR112023001454A2 (pt) * 2020-08-03 2023-02-14 Natco Pharma Ltd Composição de comprimido de liberação imediata e processo para a preparação da composição
MX2022015336A (es) * 2020-09-29 2023-01-11 Laboratorios Silanes S A De C V Combinaciones farmaceuticas de estatinas y fibratos para el tratamiento y prevencion de hiperlipidemias y enfermedades cardiovasculares.
WO2022162122A1 (en) 2021-01-29 2022-08-04 Biotx.Ai Gmbh Genetically verified netosis inhibitor for use in the treatment of a sars-cov2 infection
AU2022311961A1 (en) 2021-07-16 2023-11-09 Dana-Farber Cancer Institute, Inc. Small molecule cyclin dependent kinase 4/6 (cdk4/6) and ikzf2 (helios) degraders and methods of use thereof
TWI848533B (zh) 2022-01-25 2024-07-11 瑞士商諾華公司 瑞博西尼藥物組成物
JP2025530742A (ja) 2022-08-31 2025-09-17 アルビナス・オペレーションズ・インコーポレイテッド エストロゲン受容体分解物質の投与計画
EP4626890A1 (en) 2022-12-01 2025-10-08 KRKA, d.d., Novo mesto Ribociclib salts and formulations thereof
KR20250163966A (ko) 2023-03-27 2025-11-21 노파르티스 아게 리보시클립과 아로마타제 저해제를 병용하여 초기 유방암을 치료하는 방법
WO2025219830A1 (en) 2024-04-15 2025-10-23 Novartis Ag Pharmaceutical compositions of ribociclib

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5428812A (en) * 1977-08-09 1979-03-03 Yoshitomi Pharmaceut Ind Ltd Preparation of coated tablet
GB9414045D0 (en) 1994-07-12 1994-08-31 Berwind Pharma Service Moisture barrier film coating composition, method, and coated form
AU703933B2 (en) * 1994-07-12 1999-04-01 Berwind Pharmaceutical Services, Inc. Moisture barrier film coating composition, method, and coated form
US6448323B1 (en) * 1999-07-09 2002-09-10 Bpsi Holdings, Inc. Film coatings and film coating compositions based on polyvinyl alcohol
BRPI0917791B1 (pt) 2008-08-22 2022-03-22 Novartis Ag Compostos de pirrolopirimidina como inibidores de cdk, bem como composição farmacêutica e combinação
US8807979B2 (en) * 2009-09-24 2014-08-19 Mcneil-Ppc, Inc. Machine for the manufacture of dosage forms utilizing radiofrequency energy
US20120115878A1 (en) 2010-11-10 2012-05-10 John Vincent Calienni Salt(s) of 7-cyclopentyl-2-(5-piperazin-1-yl-pyridin-2-ylamino)-7h-pyrrolo[2,3-d]pyrimidine-6-carboxylic acid dimethylamide and processes of making thereof
AU2011358840B2 (en) * 2011-02-11 2017-05-04 TauRx Therapeutics Management Ltd Phenothiazine diaminium salts and their use
LT2872482T (lt) * 2012-07-13 2020-12-28 Oncternal Therapeutics, Inc. Krūties vėžių gydymo būdas selektyviu androgeno receptoriaus moduliatoriumi
EP2742940B1 (en) * 2012-12-13 2017-07-26 IP Gesellschaft für Management mbH Fumarate salt of (R)-3-(6-(4-methylphenyl)-pyridin-3-yloxy)-l-aza-bicyclo-[2.2.2]octane for adminstration once daily, twice daily or thrice daily
ES2676177T3 (es) * 2012-12-20 2018-07-17 Novartis Ag Una combinación farmacéutica que comprende binimetinib
AU2014233805B2 (en) * 2013-03-21 2018-10-18 Array Biopharma Inc. Combination therapy comprising a B-Raf inhibitor and a second inhibitor
EP2810644A1 (en) * 2013-06-06 2014-12-10 Ferrer Internacional, S.A. Oral formulation for the treatment of cardiovascular diseases
MX2017013350A (es) * 2015-04-16 2018-01-25 Novartis Ag Comprimido de ribociclib.
CN109953966A (zh) * 2017-12-26 2019-07-02 天津耀辰实业发展有限公司 一种含有瑞博西尼的药物组合物及其制备方法
JP7347388B2 (ja) 2020-09-25 2023-09-20 信越化学工業株式会社 紫外線硬化型有機変性シリコーン組成物および硬化物

Also Published As

Publication number Publication date
CL2017002593A1 (es) 2018-05-18
EP4197530A1 (en) 2023-06-21
AU2020250190A1 (en) 2020-11-05
CA2982425A1 (en) 2016-10-20
JP2018514523A (ja) 2018-06-07
AU2022215155B2 (en) 2024-08-01
CN115554257A (zh) 2023-01-03
PE20180035A1 (es) 2018-01-09
HUE061213T2 (hu) 2023-05-28
TW201642864A (zh) 2016-12-16
BR112017021283A2 (pt) 2018-06-26
PH12017501820A1 (en) 2018-04-23
IL254818A0 (en) 2017-12-31
US12419894B2 (en) 2025-09-23
US20180071292A1 (en) 2018-03-15
EP4620458A3 (en) 2025-10-22
KR102750931B1 (ko) 2025-01-09
HRP20230053T1 (hr) 2023-03-03
PL3283058T3 (pl) 2023-03-20
US20250134893A1 (en) 2025-05-01
US20250090531A1 (en) 2025-03-20
CO2017010510A2 (es) 2018-03-20
SI3283058T1 (sl) 2023-03-31
AR104257A1 (es) 2017-07-05
EP3283058B1 (en) 2022-11-16
CN107530292B (zh) 2022-11-01
KR20170137101A (ko) 2017-12-12
ES2938261T3 (es) 2023-04-05
US12064434B2 (en) 2024-08-20
MX2017013350A (es) 2018-01-25
SG11201708084PA (en) 2017-10-30
EP4197530B1 (en) 2025-11-12
FI3283058T3 (fi) 2023-03-01
PT3283058T (pt) 2023-02-03
CA2982425C (en) 2023-10-31
AU2016248017A1 (en) 2017-10-19
US20230104792A1 (en) 2023-04-06
EP3283058A1 (en) 2018-02-21
AU2022215155A1 (en) 2022-09-01
US20200390771A1 (en) 2020-12-17
EA201792290A1 (ru) 2018-02-28
TN2017000422A1 (en) 2019-01-16
KR20250009572A (ko) 2025-01-17
AU2019201929A1 (en) 2019-04-11
CN107530292A (zh) 2018-01-02
WO2016166703A1 (en) 2016-10-20
AU2019201929B2 (en) 2020-07-09
US20250127785A1 (en) 2025-04-24
DK3283058T3 (da) 2023-02-13
EP4620458A2 (en) 2025-09-24
AU2024227794A1 (en) 2024-11-21
US10799506B2 (en) 2020-10-13

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