ECSP088969A - Amino-imidazolones y su uso como medicamento para tratar deficiencias cognitivas, enfermedad de alzheimer, neurodegeneración y demencia - Google Patents
Amino-imidazolones y su uso como medicamento para tratar deficiencias cognitivas, enfermedad de alzheimer, neurodegeneración y demenciaInfo
- Publication number
- ECSP088969A ECSP088969A EC2008008969A ECSP088969A ECSP088969A EC SP088969 A ECSP088969 A EC SP088969A EC 2008008969 A EC2008008969 A EC 2008008969A EC SP088969 A ECSP088969 A EC SP088969A EC SP088969 A ECSP088969 A EC SP088969A
- Authority
- EC
- Ecuador
- Prior art keywords
- neurodegeneration
- dementia
- alzheimer
- disease
- imidazolones
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Abstract
Esta invención se refiere a compuestos nuevos que tienen la fórmula estructural I a continuación y a sus sales, composiciones y métodos de uso farmacéuticamente aceptables. Estos compuestos nuevos proporcionan un tratamiento o la profilaxis de la deficiencia cognitiva, la enfermedad de Alzheimer, la neurodegeneración y la demencia.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US81354906P | 2006-06-14 | 2006-06-14 | |
US86645106P | 2006-11-20 | 2006-11-20 | |
US89698607P | 2007-03-26 | 2007-03-26 |
Publications (1)
Publication Number | Publication Date |
---|---|
ECSP088969A true ECSP088969A (es) | 2009-01-30 |
Family
ID=38831994
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EC2008008969A ECSP088969A (es) | 2006-06-14 | 2008-12-12 | Amino-imidazolones y su uso como medicamento para tratar deficiencias cognitivas, enfermedad de alzheimer, neurodegeneración y demencia |
Country Status (16)
Country | Link |
---|---|
US (1) | US20070299087A1 (es) |
EP (1) | EP2035425A1 (es) |
JP (1) | JP2009539975A (es) |
KR (1) | KR20090031564A (es) |
AR (1) | AR061371A1 (es) |
AU (1) | AU2007259432A1 (es) |
BR (1) | BRPI0712731A2 (es) |
CA (1) | CA2654403A1 (es) |
CL (1) | CL2007001732A1 (es) |
EC (1) | ECSP088969A (es) |
IL (1) | IL195574A0 (es) |
MX (1) | MX2008015587A (es) |
NO (1) | NO20090166L (es) |
TW (1) | TW200808796A (es) |
UY (1) | UY30411A1 (es) |
WO (1) | WO2007145570A1 (es) |
Families Citing this family (25)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7763609B2 (en) | 2003-12-15 | 2010-07-27 | Schering Corporation | Heterocyclic aspartyl protease inhibitors |
US7592348B2 (en) | 2003-12-15 | 2009-09-22 | Schering Corporation | Heterocyclic aspartyl protease inhibitors |
US7700603B2 (en) * | 2003-12-15 | 2010-04-20 | Schering Corporation | Heterocyclic aspartyl protease inhibitors |
ES2306200T3 (es) * | 2004-07-28 | 2008-11-01 | Schering Corporation | Inhibidores macrociclicos de beta-secretasa. |
US7868000B2 (en) * | 2005-06-14 | 2011-01-11 | Schering Corporation | Aspartyl protease inhibitors |
ES2436795T3 (es) * | 2005-06-14 | 2014-01-07 | Merck Sharp & Dohme Corp. | Inhibidores heterocíclicos de aspartil proteasa, preparación y uso de los mismos |
TW200815349A (en) | 2006-06-22 | 2008-04-01 | Astrazeneca Ab | New compounds |
US8093254B2 (en) | 2006-12-12 | 2012-01-10 | Schering Corporation | Aspartyl protease inhibitors |
EP2061771A1 (en) * | 2006-12-12 | 2009-05-27 | Schering Corporation | Aspartyl protease inhibitors containing a tricyclic ring system |
JP2011518225A (ja) * | 2008-04-22 | 2011-06-23 | シェーリング コーポレイション | Bace−1阻害剤としてのフェニル置換2−イミノ−3−メチルピロロピリミジノン化合物、組成物、およびそれらの使用 |
TW201020244A (en) | 2008-11-14 | 2010-06-01 | Astrazeneca Ab | New compounds |
US20100125087A1 (en) * | 2008-11-14 | 2010-05-20 | Astrazeneca Ab | New compounds 575 |
WO2010056194A1 (en) * | 2008-11-14 | 2010-05-20 | Astrazeneca Ab | 5h-pyrrolo [ 3, 4-b] pyridin derivatives and their use |
TW201038265A (en) * | 2009-03-26 | 2010-11-01 | Dainippon Sumitomo Pharma Co | Agent for treatment of cognitive impairment |
WO2011044184A1 (en) | 2009-10-08 | 2011-04-14 | Schering Corporation | Pentafluorosulfur imino heterocyclic compounds as bace-1 inhibitors, compositions, and their use |
UA108363C2 (uk) | 2009-10-08 | 2015-04-27 | Похідні імінотіадіазиндіоксиду як інгібітори bace, композиція на їх основі і їх застосування | |
US8563543B2 (en) | 2009-10-08 | 2013-10-22 | Merck Sharp & Dohme Corp. | Iminothiadiazine dioxide compounds as bace inhibitors, compositions, and their use |
EP2485920B1 (en) | 2009-10-08 | 2016-04-27 | Merck Sharp & Dohme Corp. | Pentafluorosulfur imino heterocyclic compounds as bace-1 inhibitors, compositions, and their use |
US9221839B2 (en) | 2011-04-07 | 2015-12-29 | Merck Sharp & Dohme Corp. | C5-C6 oxacyclic-fused thiadiazine dioxide compounds as BACE inhibitors, compositions, and their use |
EP2694521B1 (en) | 2011-04-07 | 2015-11-25 | Merck Sharp & Dohme Corp. | Pyrrolidine-fused thiadiazine dioxide compounds as bace inhibitors, compositions, and their use |
US9181236B2 (en) | 2011-08-22 | 2015-11-10 | Merck Sharp & Dohme Corp. | 2-spiro-substituted iminothiazines and their mono-and dioxides as bace inhibitors, compositions and their use |
WO2013142370A1 (en) | 2012-03-19 | 2013-09-26 | Varghese John | APP SPECIFIC BACE INHIBITORS (ASBIs) AND USES THEREOF |
US9422277B2 (en) | 2012-10-17 | 2016-08-23 | Merck Sharp & Dohme Corp. | Tricyclic substituted thiadiazine dioxide compounds as BACE inhibitors, compositions and their use |
EP2908824B1 (en) | 2012-10-17 | 2018-05-02 | Merck Sharp & Dohme Corp. | Tricyclic substituted thiadiazine dioxide compounds as bace inhibitors, compositions, and their use |
CN104995176B (zh) | 2013-02-12 | 2019-02-22 | 巴克老龄化研究所 | 调节bace所介导的app加工的乙内酰脲 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR20070026811A (ko) * | 2004-06-16 | 2007-03-08 | 와이어쓰 | 베타-세크리타제 억제제로서의 디페닐이미다조피리미딘 및디페닐이미다졸 아민 |
WO2006076284A2 (en) * | 2005-01-14 | 2006-07-20 | Wyeth | AMINO-IMIDAZOLONES FOR THE INHIBITION OF ß-SECRETASE |
-
2007
- 2007-06-04 TW TW096119991A patent/TW200808796A/zh unknown
- 2007-06-11 US US11/761,131 patent/US20070299087A1/en not_active Abandoned
- 2007-06-12 KR KR1020097000708A patent/KR20090031564A/ko not_active Application Discontinuation
- 2007-06-12 EP EP07748236A patent/EP2035425A1/en not_active Withdrawn
- 2007-06-12 BR BRPI0712731-6A patent/BRPI0712731A2/pt not_active Application Discontinuation
- 2007-06-12 JP JP2009515346A patent/JP2009539975A/ja active Pending
- 2007-06-12 WO PCT/SE2007/000573 patent/WO2007145570A1/en active Application Filing
- 2007-06-12 MX MX2008015587A patent/MX2008015587A/es not_active Application Discontinuation
- 2007-06-12 AU AU2007259432A patent/AU2007259432A1/en not_active Abandoned
- 2007-06-12 CA CA002654403A patent/CA2654403A1/en not_active Abandoned
- 2007-06-13 UY UY30411A patent/UY30411A1/es not_active Application Discontinuation
- 2007-06-13 AR ARP070102596A patent/AR061371A1/es unknown
- 2007-06-13 CL CL2007001732A patent/CL2007001732A1/es unknown
-
2008
- 2008-11-27 IL IL195574A patent/IL195574A0/en unknown
- 2008-12-12 EC EC2008008969A patent/ECSP088969A/es unknown
-
2009
- 2009-01-12 NO NO20090166A patent/NO20090166L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
IL195574A0 (en) | 2009-09-01 |
WO2007145570A9 (en) | 2008-12-11 |
UY30411A1 (es) | 2008-01-31 |
TW200808796A (en) | 2008-02-16 |
AR061371A1 (es) | 2008-08-20 |
EP2035425A1 (en) | 2009-03-18 |
JP2009539975A (ja) | 2009-11-19 |
BRPI0712731A2 (pt) | 2012-10-02 |
US20070299087A1 (en) | 2007-12-27 |
KR20090031564A (ko) | 2009-03-26 |
CL2007001732A1 (es) | 2008-01-25 |
CA2654403A1 (en) | 2007-12-21 |
NO20090166L (no) | 2009-03-12 |
AU2007259432A1 (en) | 2007-12-21 |
MX2008015587A (es) | 2009-01-09 |
WO2007145570A1 (en) | 2007-12-21 |
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