ECSP088545A - Composición para prevenir o tratar daños de la mucosa en los conductos gastrointestinales - Google Patents

Composición para prevenir o tratar daños de la mucosa en los conductos gastrointestinales

Info

Publication number
ECSP088545A
ECSP088545A EC2008008545A ECSP088545A ECSP088545A EC SP088545 A ECSP088545 A EC SP088545A EC 2008008545 A EC2008008545 A EC 2008008545A EC SP088545 A ECSP088545 A EC SP088545A EC SP088545 A ECSP088545 A EC SP088545A
Authority
EC
Ecuador
Prior art keywords
composition
prevent
gastrointestinal
mucosa damage
damage
Prior art date
Application number
EC2008008545A
Other languages
English (en)
Inventor
Ki-Baik Hahm
Dong-Kyu Kim
Mi-Sun Kwak
Sang-Aun Joo
Byoung-Seok Moon
Geun-Seog Song
Original Assignee
Yuhan Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Yuhan Corp filed Critical Yuhan Corp
Publication of ECSP088545A publication Critical patent/ECSP088545A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Se provee una composición para prevenir o tratar daños de la mucosa en los conductos gastrointestinales, que incluye el revaprazán o una sal del mismo y un portador farmacéuticamente aceptable. El revaprazán o su sal tienen un excelente efecto preventivo o de tratamiento para daños a la mucosa gastrointestinal, al potenciar un factor defensivo en la mucosa gastrointestinal, y simultáneamente actuar como un antagonista de la bomba de ácido..
EC2008008545A 2005-12-01 2008-06-13 Composición para prevenir o tratar daños de la mucosa en los conductos gastrointestinales ECSP088545A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
KR20050116567 2005-12-01

Publications (1)

Publication Number Publication Date
ECSP088545A true ECSP088545A (es) 2008-08-29

Family

ID=38092428

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2008008545A ECSP088545A (es) 2005-12-01 2008-06-13 Composición para prevenir o tratar daños de la mucosa en los conductos gastrointestinales

Country Status (15)

Country Link
US (1) US7776873B2 (es)
EP (1) EP1954279A4 (es)
JP (1) JP5207974B2 (es)
KR (1) KR100805660B1 (es)
CN (2) CN101316594B (es)
AU (1) AU2006321471B2 (es)
BR (1) BRPI0619081A2 (es)
CA (1) CA2631068C (es)
CR (1) CR10018A (es)
EC (1) ECSP088545A (es)
HK (1) HK1123507A1 (es)
IL (1) IL191680A0 (es)
MY (1) MY145406A (es)
WO (1) WO2007064128A1 (es)
ZA (1) ZA200805747B (es)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10835541B2 (en) 2015-07-30 2020-11-17 Takeda Pharmaceutical Company Limited Tablet

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2007339080B2 (en) * 2006-12-22 2012-09-27 Yuhan Corporation Revaprazan-containing solid dispersion and process for the preparation thereof
JP5802898B2 (ja) 2009-07-09 2015-11-04 ラクオリア創薬株式会社 消化管運動異常が関与する疾患を治療するためのアシッドポンプ拮抗剤
KR101730865B1 (ko) 2011-02-11 2017-04-27 주식회사유한양행 레바프라잔-함유 나노입자를 포함하는 경구투여용 약학 조성물 및 그의 제조방법
KR101739818B1 (ko) * 2011-05-20 2017-05-26 주식회사유한양행 레바프라잔 또는 그의 염을 함유하는 현탁액 형태의 경구투여용 약학 조성물
CN105998688A (zh) * 2016-06-22 2016-10-12 郑亮 一种胃粘膜损伤的抑制方法
KR20180107341A (ko) * 2017-03-16 2018-10-02 차의과학대학교 산학협력단 칼륨 경쟁적 위산분비억제제를 유효성분을 함유하는 장 누수 증후군 치료 및 예방용 조성물

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IN171746B (es) * 1989-11-02 1992-12-26 Mcneil Ppc Inc
DE69530989T2 (de) 1994-08-13 2004-05-19 Yuhan Corp. Neue pyrimidinderivate und verfahren zu ihrer herstellung
JP3160297B2 (ja) * 1996-05-04 2001-04-25 ユーハン・コーポレイション ピリミジン誘導体の製造方法
CN1088706C (zh) * 1996-10-25 2002-08-07 卫福有限公司 新型杂环酰胺化合物及其医药用途
HU226752B1 (en) 1996-10-29 2009-09-28 Yuhan Corp Process for preparation of pyrimidine derivatives
GB0110338D0 (en) * 2001-04-27 2001-06-20 Sb Pharmco Inc Novel processes
US8206741B2 (en) * 2001-06-01 2012-06-26 Pozen Inc. Pharmaceutical compositions for the coordinated delivery of NSAIDs

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10835541B2 (en) 2015-07-30 2020-11-17 Takeda Pharmaceutical Company Limited Tablet

Also Published As

Publication number Publication date
JP2009517462A (ja) 2009-04-30
AU2006321471A1 (en) 2007-06-07
HK1123507A1 (en) 2009-06-19
IL191680A0 (en) 2009-08-03
EP1954279A4 (en) 2009-06-03
KR20070057663A (ko) 2007-06-07
CA2631068C (en) 2011-01-11
CN102309490A (zh) 2012-01-11
CA2631068A1 (en) 2007-06-07
US7776873B2 (en) 2010-08-17
ZA200805747B (en) 2009-11-25
CN101316594B (zh) 2012-07-25
EP1954279A1 (en) 2008-08-13
MY145406A (en) 2012-02-15
BRPI0619081A2 (pt) 2011-09-20
KR100805660B1 (ko) 2008-02-21
WO2007064128A1 (en) 2007-06-07
AU2006321471B2 (en) 2010-07-29
JP5207974B2 (ja) 2013-06-12
US20070129391A1 (en) 2007-06-07
CR10018A (es) 2008-09-02
CN101316594A (zh) 2008-12-03

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