ECSP077208A - Inhibidores de los canales de potasio - Google Patents

Inhibidores de los canales de potasio

Info

Publication number
ECSP077208A
ECSP077208A EC2007007208A ECSP077208A ECSP077208A EC SP077208 A ECSP077208 A EC SP077208A EC 2007007208 A EC2007007208 A EC 2007007208A EC SP077208 A ECSP077208 A EC SP077208A EC SP077208 A ECSP077208 A EC SP077208A
Authority
EC
Ecuador
Prior art keywords
potassium channel
channel inhibitors
inhibitors
compounds
relates
Prior art date
Application number
EC2007007208A
Other languages
English (en)
Inventor
Mark T Bilodeau
Zhicai Wu
John Hartnett
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of ECSP077208A publication Critical patent/ECSP077208A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/18Sulfonamides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente invención se refiere a compuestos que tienen la estructura útiles como inhibidores del canal de potasio para tratar arritmias cardíacas y afecciones similares.
EC2007007208A 2004-07-29 2007-01-26 Inhibidores de los canales de potasio ECSP077208A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US59218104P 2004-07-29 2004-07-29

Publications (1)

Publication Number Publication Date
ECSP077208A true ECSP077208A (es) 2007-02-28

Family

ID=35613661

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2007007208A ECSP077208A (es) 2004-07-29 2007-01-26 Inhibidores de los canales de potasio

Country Status (15)

Country Link
KR (1) KR20070043985A (es)
AR (1) AR049847A1 (es)
BR (1) BRPI0513793A (es)
CR (1) CR8876A (es)
EC (1) ECSP077208A (es)
IL (1) IL180846A0 (es)
MA (1) MA28980B1 (es)
MX (1) MX2007001188A (es)
NO (1) NO20071107L (es)
PE (1) PE20060382A1 (es)
RU (1) RU2344134C2 (es)
TW (1) TW200607493A (es)
UA (1) UA88018C2 (es)
WO (1) WO2006028590A1 (es)
ZA (1) ZA200700477B (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN105311003A (zh) * 2009-03-18 2016-02-10 麦迪库瑞国际公司 替罗非班的透皮药物制剂和给药
ES2675314T3 (es) 2012-06-11 2018-07-10 Bristol-Myers Squibb Company Profármacos de ácido fosforamídico de 5-[5-fenil-4-(piridin-2-ilmetilamino) quinazolin-2-il] piridin-3-sulfonamida

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1911740B1 (en) * 2002-01-04 2013-02-27 NeuroSearch A/S Potassium channel modulators

Also Published As

Publication number Publication date
BRPI0513793A (pt) 2008-05-13
IL180846A0 (en) 2007-06-03
TW200607493A (en) 2006-03-01
NO20071107L (no) 2007-04-19
PE20060382A1 (es) 2006-05-15
MX2007001188A (es) 2007-03-21
ZA200700477B (en) 2009-08-26
MA28980B1 (fr) 2007-11-01
UA88018C2 (ru) 2009-09-10
KR20070043985A (ko) 2007-04-26
RU2007107408A (ru) 2008-09-10
WO2006028590A1 (en) 2006-03-16
RU2344134C2 (ru) 2009-01-20
AR049847A1 (es) 2006-09-06
CR8876A (es) 2007-08-28

Similar Documents

Publication Publication Date Title
ECSP088676A (es) Pirazolquinolonas como potentes inhibidores de parp
UY32730A (es) Inhibidores de cyp17
DOP2010000225A (es) Arilpirrolinas insecticidas
CO6511220A2 (es) Quinazolinas como inhibidores de los canales iónicos de potasio
ECSP10010344A (es) Azolilmetiloxiranos, su uso y agentes que los contienen
TR201901649T4 (tr) Nematodların ve toprak kaynaklı hastalıkların kontrolüne yönelik bileşimler ve yöntemler.
ECSP088221A (es) Agonistas adrenoreceptores alfa2c
EA200970737A1 (ru) Оксабициклогептаны и оксабициклогептены, их получение и применение
ATE510822T1 (de) Kaliumkanalinhibitoren
PA8667201A1 (es) Nuevos compuestos farmaceuticos
DOP2011000134A (es) Lactamas como inhibidores de beta secretasa
UY31560A1 (es) Azolilmetiloxiranos, su uso y agentes que los contienen
UY31688A1 (es) Plaguicidas
CL2008000202A1 (es) Compuestos derivados de n-aril-acetamida, antagonista trpv1;composicion farmaceutica que los comprende, utiles en el tratamiento del dolor.
CO6361894A2 (es) Composiciones aclaradoras de la piel con inhibidores de acetilcolinesterasa
UY29668A1 (es) Nuevos derivados de heptaazafenaleno, procedimientos para su obtencinn, ase como utilizacinn de estos como agentes protectores contra la radicacinn uv.-
UA106889C2 (uk) Похідні n1-ацил-5-фторпіримідинону
CR20120117A (es) Métodos para la propagación vegetativa de gramíneas
ECSP099738A (es) Derivados de pirazolona como inhibidores de pde4
EA201170201A1 (ru) Предотвращение и лечение радиационного поражения
BRPI0820698A2 (pt) 4-imidazolidinonas como inibidores de canal de potássio kv1.5
ECSP077208A (es) Inhibidores de los canales de potasio
BRPI0821394A2 (pt) 4-imidazolidinonas como inibidores de canal de potássio kv1.5
DOP2005000144A (es) Inhibidores de los canales de potasio
MA33932B1 (fr) Dérivés de 2-aldoximino-5-fluoropyrimidine