EA202191984A1 - Фармацевтическая композиция, содержащая ингибитор flt3 и гипометилирующий агент, для лечения острого миелолейкоза - Google Patents
Фармацевтическая композиция, содержащая ингибитор flt3 и гипометилирующий агент, для лечения острого миелолейкозаInfo
- Publication number
- EA202191984A1 EA202191984A1 EA202191984A EA202191984A EA202191984A1 EA 202191984 A1 EA202191984 A1 EA 202191984A1 EA 202191984 A EA202191984 A EA 202191984A EA 202191984 A EA202191984 A EA 202191984A EA 202191984 A1 EA202191984 A1 EA 202191984A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- treatment
- pharmaceutical composition
- acute
- agent
- myeloleukosis
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Hematology (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Предложены фармацевтическая композиция для лечения острого миелолейкоза (AML) и способ лечения острого миелолейкоза с ее использованием, где композиция содержит ингибитор Fms-подобной тирозинкиназы-3 (FLT3) или его фармацевтически приемлемые соль или сольват и гипометилирующий агент (НМА) или его фармацевтически приемлемые соль или сольват в терапевтически эффективной комбинации.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
KR20190021228 | 2019-02-22 | ||
KR1020200021502A KR20200102949A (ko) | 2019-02-22 | 2020-02-21 | Flt3 저해제 및 저메틸화제를 포함하는 급성 골수성 백혈병의 치료를 위한 약학적 조성물 |
PCT/KR2020/002536 WO2020171646A1 (ko) | 2019-02-22 | 2020-02-21 | Flt3 저해제 및 저메틸화제를 포함하는 급성 골수성 백혈병의 치료를 위한 약학적 조성물 |
Publications (1)
Publication Number | Publication Date |
---|---|
EA202191984A1 true EA202191984A1 (ru) | 2021-11-19 |
Family
ID=72470030
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA202191984A EA202191984A1 (ru) | 2019-02-22 | 2020-02-21 | Фармацевтическая композиция, содержащая ингибитор flt3 и гипометилирующий агент, для лечения острого миелолейкоза |
Country Status (8)
Country | Link |
---|---|
EP (1) | EP3928780A4 (ru) |
KR (1) | KR20200102949A (ru) |
CN (1) | CN113490497A (ru) |
AU (1) | AU2020226111A1 (ru) |
CA (1) | CA3130244A1 (ru) |
EA (1) | EA202191984A1 (ru) |
IL (1) | IL285628A (ru) |
SG (1) | SG11202108867VA (ru) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN114650823A (zh) * | 2019-06-27 | 2022-06-21 | 韩美药品株式会社 | 用于治疗急性髓系白血病的含有flt3抑制剂和化疗剂的药物组合物 |
EP4370127A2 (en) * | 2021-07-12 | 2024-05-22 | Quteba Ebrahem | A method of treating cancer or a blood disorder |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MX2009005621A (es) | 2006-11-28 | 2009-06-12 | Novartis Ag | Combinacion de inhibidores de iap e inhibidores de flt3. |
KR20180124055A (ko) | 2016-03-29 | 2018-11-20 | 아스테라스 세이야쿠 가부시키가이샤 | 급성 골수성 백혈병의 치료를 위한 병용 요법 |
PT3514153T (pt) * | 2017-01-26 | 2021-09-22 | Hanmi Pharm Ind Co Ltd | Composto de pirimidina e utilização farmacêutica do mesmo |
-
2020
- 2020-02-21 CN CN202080015594.7A patent/CN113490497A/zh active Pending
- 2020-02-21 CA CA3130244A patent/CA3130244A1/en active Pending
- 2020-02-21 AU AU2020226111A patent/AU2020226111A1/en active Pending
- 2020-02-21 KR KR1020200021502A patent/KR20200102949A/ko unknown
- 2020-02-21 SG SG11202108867VA patent/SG11202108867VA/en unknown
- 2020-02-21 EA EA202191984A patent/EA202191984A1/ru unknown
- 2020-02-21 EP EP20759712.1A patent/EP3928780A4/en active Pending
-
2021
- 2021-08-15 IL IL285628A patent/IL285628A/en unknown
Also Published As
Publication number | Publication date |
---|---|
KR20200102949A (ko) | 2020-09-01 |
EP3928780A4 (en) | 2022-12-07 |
SG11202108867VA (en) | 2021-09-29 |
CN113490497A (zh) | 2021-10-08 |
AU2020226111A1 (en) | 2021-09-09 |
EP3928780A1 (en) | 2021-12-29 |
IL285628A (en) | 2021-09-30 |
CA3130244A1 (en) | 2020-08-27 |
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