EA201500913A1 - Противомикробные соединения и способы их получения и применения - Google Patents

Противомикробные соединения и способы их получения и применения

Info

Publication number
EA201500913A1
EA201500913A1 EA201500913A EA201500913A EA201500913A1 EA 201500913 A1 EA201500913 A1 EA 201500913A1 EA 201500913 A EA201500913 A EA 201500913A EA 201500913 A EA201500913 A EA 201500913A EA 201500913 A1 EA201500913 A1 EA 201500913A1
Authority
EA
Eurasian Patent Office
Prior art keywords
methods
production
application
antimicrobial compounds
compounds
Prior art date
Application number
EA201500913A
Other languages
English (en)
Inventor
Эрин М. Даффи
Ашоке Бхаттачарджи
Хардвин О'Доуд
Марко Девиво
Яньмин Ду
Сандра Сиништаж
Юаньцин Тан
Брайан Т. Вимберли
Original Assignee
Мелинта Терапьютикс, Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Мелинта Терапьютикс, Инк. filed Critical Мелинта Терапьютикс, Инк.
Publication of EA201500913A1 publication Critical patent/EA201500913A1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • C07D491/044—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
    • C07D491/048—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring the oxygen-containing ring being five-membered
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Biophysics (AREA)
  • Pathology (AREA)
  • Surgery (AREA)
  • Medical Informatics (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Biomedical Technology (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Physics & Mathematics (AREA)
  • Vascular Medicine (AREA)
  • Ophthalmology & Optometry (AREA)
  • Otolaryngology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Materials For Medical Uses (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Изобретение относится в целом к области противомикробных соединений и к способам их получения и применения. Эти соединения могут быть использованы для лечения, профилактики и уменьшения риска микробных инфекций у человека и животных.
EA201500913A 2009-10-16 2010-10-15 Противомикробные соединения и способы их получения и применения EA201500913A1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US25247809P 2009-10-16 2009-10-16
US31428710P 2010-03-16 2010-03-16
US35820110P 2010-06-24 2010-06-24

Publications (1)

Publication Number Publication Date
EA201500913A1 true EA201500913A1 (ru) 2015-12-30

Family

ID=43876906

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201500913A EA201500913A1 (ru) 2009-10-16 2010-10-15 Противомикробные соединения и способы их получения и применения

Country Status (9)

Country Link
JP (6) JP2016121171A (ru)
KR (3) KR20120101392A (ru)
CN (5) CN107445976A (ru)
AR (3) AR080558A1 (ru)
EA (1) EA201500913A1 (ru)
MY (2) MY161870A (ru)
NZ (2) NZ713357A (ru)
SG (3) SG10201406631TA (ru)
TW (8) TWI612048B (ru)

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BR112012008795A2 (pt) 2009-10-16 2020-09-24 Rib-X Pharmaceuticals, Inc. compostos antimicrobianos e métodos de fabricação e uso dos mesmos.
US9221827B2 (en) * 2011-04-15 2015-12-29 Melinta Therapeutics, Inc. Antimicrobial compounds and methods of making and using the same
EP3039025A4 (en) 2013-09-09 2017-05-31 Melinta Therapeutics, Inc. Antimicrobial compounds and methods of making and using the same
CA2923179A1 (en) 2013-09-09 2015-03-12 Melinta Therapeutics, Inc. Antimicrobial compounds and methods of making and using the same
EA201792006A1 (ru) 2015-03-11 2018-04-30 Мелинта Терапьютикс, Инк. Антимикробные соединения и способы их получения и их применение

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Also Published As

Publication number Publication date
CN104628729A (zh) 2015-05-20
TW201825495A (zh) 2018-07-16
NZ713357A (en) 2017-05-26
JP2018039784A (ja) 2018-03-15
JP2018024653A (ja) 2018-02-15
KR20120099436A (ko) 2012-09-10
TWI612048B (zh) 2018-01-21
TW201124417A (en) 2011-07-16
CN104628729B (zh) 2018-11-06
CN107266470A (zh) 2017-10-20
TW201630914A (zh) 2016-09-01
TWI621439B (zh) 2018-04-21
KR20120101392A (ko) 2012-09-13
TW201125566A (en) 2011-08-01
SG10201406631TA (en) 2014-11-27
CN108456211A (zh) 2018-08-28
AR080559A1 (es) 2012-04-18
TW201731849A (zh) 2017-09-16
TW201622725A (zh) 2016-07-01
CN107445976A (zh) 2017-12-08
KR20120099435A (ko) 2012-09-10
TW201125564A (en) 2011-08-01
AR080617A1 (es) 2012-04-25
MY161870A (en) 2017-05-15
JP2016121171A (ja) 2016-07-07
TWI629277B (zh) 2018-07-11
AR080558A1 (es) 2012-04-18
TWI589294B (zh) 2017-07-01
SG10201406634VA (en) 2014-11-27
TW201726630A (zh) 2017-08-01
JP2016153405A (ja) 2016-08-25
CN105646370A (zh) 2016-06-08
JP2019038808A (ja) 2019-03-14
MY165011A (en) 2018-02-28
KR101857694B1 (ko) 2018-06-19
SG10201406635QA (en) 2014-11-27
JP2016172733A (ja) 2016-09-29
TWI618707B (zh) 2018-03-21
NZ623384A (en) 2016-06-24

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