EA201391733A1 - Каннабиноиды, применяемые для лечения невропатической боли - Google Patents
Каннабиноиды, применяемые для лечения невропатической болиInfo
- Publication number
- EA201391733A1 EA201391733A1 EA201391733A EA201391733A EA201391733A1 EA 201391733 A1 EA201391733 A1 EA 201391733A1 EA 201391733 A EA201391733 A EA 201391733A EA 201391733 A EA201391733 A EA 201391733A EA 201391733 A1 EA201391733 A1 EA 201391733A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- cannabinoids
- neuropathic pain
- treatment
- cannabinoids used
- cannabichromen
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
- A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/045—Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
- A61K31/05—Phenols
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pain & Pain Management (AREA)
- Engineering & Computer Science (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Plant Substances (AREA)
Abstract
Настоящее изобретение относится к каннабиноидам, применяемым для лечения невропатической боли. Предпочтительно указанные каннабиноиды представляют собой один или несколько каннабиноидов, выбранных из группы, включающей каннабигерол (CBG), каннабихромен (СВС), каннабидиварин (CBDV) или тетрагидроканнабиварин (THCV). Более предпочтительно указанные каннабиноиды выделяют или получают очисткой из экстрактов растения конопли.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB1108506.5A GB2491118B (en) | 2011-05-20 | 2011-05-20 | Cannabinoids for use in the treatment of neuropathic pain |
PCT/GB2012/051129 WO2012160358A1 (en) | 2011-05-20 | 2012-05-18 | Cannabinoids for use in the treatment of neuropathic pain |
Publications (1)
Publication Number | Publication Date |
---|---|
EA201391733A1 true EA201391733A1 (ru) | 2014-04-30 |
Family
ID=44279366
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201391733A EA201391733A1 (ru) | 2011-05-20 | 2012-05-18 | Каннабиноиды, применяемые для лечения невропатической боли |
Country Status (21)
Country | Link |
---|---|
US (1) | US9895342B2 (ru) |
EP (1) | EP2709604B1 (ru) |
JP (1) | JP6147249B2 (ru) |
KR (1) | KR20140037124A (ru) |
CN (1) | CN103533930A (ru) |
AR (1) | AR086398A1 (ru) |
AU (1) | AU2012260611B2 (ru) |
BR (1) | BR112013029773A2 (ru) |
CA (1) | CA2833099C (ru) |
CO (1) | CO6811867A2 (ru) |
DK (1) | DK2709604T3 (ru) |
EA (1) | EA201391733A1 (ru) |
ES (1) | ES2624308T3 (ru) |
GB (2) | GB2491118B (ru) |
IL (1) | IL229474B (ru) |
MX (1) | MX2013013141A (ru) |
PT (1) | PT2709604T (ru) |
SG (1) | SG194839A1 (ru) |
TW (1) | TW201249425A (ru) |
WO (1) | WO2012160358A1 (ru) |
ZA (1) | ZA201309364B (ru) |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB2530001B (en) | 2014-06-17 | 2019-01-16 | Gw Pharma Ltd | Use of cannabidiol in the reduction of convulsive seizure frequency in treatment-resistant epilepsy |
GB2531282A (en) | 2014-10-14 | 2016-04-20 | Gw Pharma Ltd | Use of cannabinoids in the treatment of epilepsy |
US10499584B2 (en) | 2016-05-27 | 2019-12-10 | New West Genetics | Industrial hemp Cannabis cultivars and seeds with stable cannabinoid profiles |
EP3478307A4 (en) | 2016-06-29 | 2020-02-26 | Cannscience Innovations Inc. | DECARBOXYLATED CANNABIS RESINS, USES AND METHODS OF MAKING |
US10239808B1 (en) | 2016-12-07 | 2019-03-26 | Canopy Holdings, LLC | Cannabis extracts |
WO2018236957A1 (en) * | 2017-06-20 | 2018-12-27 | Nexien Biopharma, Inc. | METHOD AND COMPOSITIONS FOR TREATING REST-FREE LEG SYNDROME |
CN109498606A (zh) * | 2017-09-15 | 2019-03-22 | 汉义生物科技(北京)有限公司 | 一种含有大麻二酚和/或次大麻二酚的组合物及其在治疗痛经中的应用 |
EP3684353A4 (en) * | 2017-09-22 | 2021-06-23 | Inmed Pharmaceuticals Inc. | TOPICAL FORMULATIONS OF CANNABINOIDS AND THEIR USES FOR PAIN TREATMENT |
WO2019147690A1 (en) * | 2018-01-23 | 2019-08-01 | High Sierra Technologies, Inc. | Cannabis products modified by removing volatile organic compounds and adding volatile unsaturated hydrocarbons |
WO2019152736A1 (en) | 2018-01-31 | 2019-08-08 | Canopy Holdings, LLC | Hemp powder |
GB201806953D0 (en) | 2018-04-27 | 2018-06-13 | Gw Res Ltd | Cannabidiol Preparations |
US11040932B2 (en) | 2018-10-10 | 2021-06-22 | Treehouse Biotech, Inc. | Synthesis of cannabigerol |
AU2020268218B2 (en) * | 2019-05-03 | 2022-09-08 | Zyus Life Sciences Inc. | Formulation for pain management |
EP4138813A4 (en) * | 2020-04-24 | 2024-05-15 | Zyus Life Sciences Inc | CANNABICHROMENE FORMULATION FOR PAIN MANAGEMENT |
US11672761B2 (en) | 2020-11-16 | 2023-06-13 | Orcosa Inc. | Rapidly infusing platform and compositions for therapeutic treatment in humans |
CN116648241A (zh) * | 2021-04-14 | 2023-08-25 | 成都百裕制药股份有限公司 | 氘代苯酚衍生物及其制备方法和用途 |
Family Cites Families (26)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EA000976B1 (ru) | 1996-03-25 | 2000-08-28 | Эли Лилли Энд Компани | Композиция для снятия боли и способ снятия боли |
US6949582B1 (en) | 1999-05-27 | 2005-09-27 | Wallace Walter H | Method of relieving analgesia and reducing inflamation using a cannabinoid delivery topical liniment |
US6730330B2 (en) | 2001-02-14 | 2004-05-04 | Gw Pharma Limited | Pharmaceutical formulations |
US7025992B2 (en) | 2001-02-14 | 2006-04-11 | Gw Pharma Limited | Pharmaceutical formulations |
GB2377633A (en) * | 2001-05-11 | 2003-01-22 | Gw Pharmaceuticals Ltd | Pharmaceutical compositions comprising the cannabinoids THC and CBD |
CA2438097C (en) * | 2001-02-14 | 2006-04-25 | Gw Pharma Limited | Cannabinoids pharmaceutical formulations |
US10004684B2 (en) * | 2001-02-14 | 2018-06-26 | Gw Pharma Limited | Pharmaceutical formulations |
GB2381194A (en) * | 2001-09-07 | 2003-04-30 | Gw Pharmaceuticals Ltd | Pharmaceutical formulations |
CH695661A5 (de) | 2001-03-06 | 2006-07-31 | Forsch Hiscia Ver Fuer Krebsfo | Pharmazeutische Zusammensetzung. |
EP1243262B1 (en) | 2001-03-20 | 2006-05-31 | Schwarz Pharma Ag | Novel use of a peptide class of compound for treating non-neuropathic inflammatory pain |
GB2381450B (en) | 2001-10-31 | 2006-05-31 | Gw Pharma Ltd | Compositions for administration of natural or synthetic cannabinoids by vaporisation |
GB2392093B (en) * | 2002-08-14 | 2006-03-08 | Gw Pharma Ltd | Pharmaceutical formulations |
US6946150B2 (en) | 2002-08-14 | 2005-09-20 | Gw Pharma Limited | Pharmaceutical formulation |
KR101008609B1 (ko) | 2002-08-14 | 2011-01-17 | 지더블유 파마 리미티드 | 점막투여용 칸나비노이드 액체 제형 |
GB2391865B (en) | 2002-08-14 | 2005-06-01 | Gw Pharma Ltd | Improvements in the extraction of pharmaceutically active components from plant materials |
GB0222077D0 (en) * | 2002-09-23 | 2002-10-30 | Gw Pharma Ltd | Methods of preparing cannabinoids from plant material |
GB2394894B (en) | 2002-11-04 | 2005-08-31 | G W Pharma Ltd | New use for pharmaceutical composition |
GB2414933B (en) | 2004-06-08 | 2009-07-15 | Gw Pharma Ltd | Cannabinoid compositions for the treatment of disease and/or symptoms in arthritis |
US7968594B2 (en) | 2005-04-27 | 2011-06-28 | Gw Pharma Limited | Pharmaceutical compositions for the treatment of pain |
EP1747786A3 (en) | 2005-07-25 | 2007-04-25 | Perdix Eurogroup S.L. | Natural product in cream with anti-vitiligo therapeutic properties |
US20070036873A1 (en) | 2005-07-27 | 2007-02-15 | Shibnath Ghosal | Method of treatment or management of stress |
CA2517313A1 (en) * | 2005-08-26 | 2007-02-26 | Queen's University At Kingston | Methods and therapies for potentiating therapeutic activities of a cannabinoid receptor agonist via administration of a cannabinoid receptor antagonist |
GB2432312A (en) | 2005-11-01 | 2007-05-23 | Gw Pharma Ltd | Pharmaceutical compositions for the treatment of pain |
GB2439393B (en) * | 2006-06-23 | 2011-05-11 | Gw Pharma Ltd | Cannabinoids for use in the treatment of neuropathic pain |
GB2448535A (en) * | 2007-04-19 | 2008-10-22 | Gw Pharma Ltd | New use for cannabinoid-containing plant extracts |
GB2450493A (en) * | 2007-06-25 | 2008-12-31 | Gw Pharma Ltd | Cannabigerol for use in treatment of diseases benefiting from agonism of CB1 and CB2 cannabinoid receptors |
-
2011
- 2011-05-20 GB GB1108506.5A patent/GB2491118B/en active Active
- 2011-05-20 GB GB1512357.3A patent/GB2524689B/en active Active
-
2012
- 2012-05-09 TW TW101116491A patent/TW201249425A/zh unknown
- 2012-05-14 AR ARP120101707A patent/AR086398A1/es unknown
- 2012-05-18 WO PCT/GB2012/051129 patent/WO2012160358A1/en active Application Filing
- 2012-05-18 DK DK12722495.4T patent/DK2709604T3/en active
- 2012-05-18 KR KR1020137033069A patent/KR20140037124A/ko not_active Application Discontinuation
- 2012-05-18 JP JP2014510885A patent/JP6147249B2/ja active Active
- 2012-05-18 AU AU2012260611A patent/AU2012260611B2/en active Active
- 2012-05-18 CA CA2833099A patent/CA2833099C/en active Active
- 2012-05-18 EP EP12722495.4A patent/EP2709604B1/en active Active
- 2012-05-18 SG SG2013082649A patent/SG194839A1/en unknown
- 2012-05-18 ES ES12722495.4T patent/ES2624308T3/es active Active
- 2012-05-18 US US14/118,563 patent/US9895342B2/en active Active
- 2012-05-18 BR BR112013029773A patent/BR112013029773A2/pt active Search and Examination
- 2012-05-18 MX MX2013013141A patent/MX2013013141A/es not_active Application Discontinuation
- 2012-05-18 PT PT127224954T patent/PT2709604T/pt unknown
- 2012-05-18 EA EA201391733A patent/EA201391733A1/ru unknown
- 2012-05-18 CN CN201280024106.4A patent/CN103533930A/zh active Pending
-
2013
- 2013-11-17 IL IL229474A patent/IL229474B/en active IP Right Grant
- 2013-12-02 CO CO13282297A patent/CO6811867A2/es not_active Application Discontinuation
- 2013-12-11 ZA ZA2013/09364A patent/ZA201309364B/en unknown
Also Published As
Publication number | Publication date |
---|---|
GB2524689A (en) | 2015-09-30 |
WO2012160358A1 (en) | 2012-11-29 |
JP2014513715A (ja) | 2014-06-05 |
GB2524689B (en) | 2016-01-27 |
ZA201309364B (en) | 2015-04-29 |
CA2833099A1 (en) | 2012-11-29 |
ES2624308T3 (es) | 2017-07-13 |
CA2833099C (en) | 2020-11-03 |
AU2012260611A1 (en) | 2013-12-12 |
IL229474B (en) | 2018-11-29 |
JP6147249B2 (ja) | 2017-06-14 |
TW201249425A (en) | 2012-12-16 |
IL229474A0 (en) | 2014-01-30 |
US20140378539A9 (en) | 2014-12-25 |
AR086398A1 (es) | 2013-12-11 |
DK2709604T3 (en) | 2017-05-15 |
GB201108506D0 (en) | 2011-07-06 |
CO6811867A2 (es) | 2013-12-16 |
US20140107192A1 (en) | 2014-04-17 |
EP2709604A1 (en) | 2014-03-26 |
CN103533930A (zh) | 2014-01-22 |
NZ618246A (en) | 2016-01-29 |
SG194839A1 (en) | 2013-12-30 |
BR112013029773A2 (pt) | 2017-01-17 |
AU2012260611B2 (en) | 2017-06-15 |
KR20140037124A (ko) | 2014-03-26 |
EP2709604B1 (en) | 2017-02-01 |
MX2013013141A (es) | 2014-02-17 |
GB2491118A (en) | 2012-11-28 |
GB2491118B (en) | 2015-12-30 |
PT2709604T (pt) | 2017-05-17 |
GB201512357D0 (en) | 2015-08-19 |
US9895342B2 (en) | 2018-02-20 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
EA201391733A1 (ru) | Каннабиноиды, применяемые для лечения невропатической боли | |
EA201490711A1 (ru) | Фармацевтическая композиция, содержащая фитоканнабиноиды каннабидиварин (cbdv) и каннабидиол (cbd) | |
CO2017008437A2 (es) | Métodos de purificación de cannabinoides, composiciones y kits de los mismos | |
UA108852C2 (ru) | Применение одного или комбинации фито каннабиноидов для лечения эпилепсии | |
NZ602925A (en) | Use of the phytocannabinoid cannabidivarin (cbdv) in the treatment of epilepsy | |
CO2019014279A2 (es) | Proceso para la purificación y separación de cannabinoides a partir de cáñamo seco y hojas de cannabis | |
FI3743053T3 (fi) | Kannabinoidien käyttö epilepsian hoidossa | |
GT200900183A (es) | Derivados de isoquinolina e isoquinolinona sustituidos con cicloalquilamina | |
CL2015001667A1 (es) | Derivados de manosa para tratar infecciones bacterianas. | |
CO2020009747A2 (es) | Métodos para purificar cannabinoides usando cromatografía líquido-líquido | |
AU2016255707A8 (en) | Uses of cannabidiol for treatment of infantile spasms | |
BR112013019522A2 (pt) | dissialil lacto-n-tetraose (dslnt) ou as variantes, os isômeros, os análogos e os derivados da mesma para prevenir ou inibir doença do intestino | |
GB201120067D0 (en) | Phytocannabinoids for use in the treatment of intestinal inflammatory diseases | |
GT200900062A (es) | Nuevos compuestos de diosmetina, un proceso para su preparacion y las composiciones farmaceuticas que los contienen | |
IL283034A (en) | Cannabis plants with a cannabinoid profile enriched for delta-9-tetrahydrocannabinol, cannabigerol and tetrahydrocannabiuria | |
CL2017001275A1 (es) | Análogos ligados de urea sustituidos como moduladores de sirtuina | |
CL2012001031A1 (es) | Compuestos derivados de 2-oxo-1-pirrolidinil-imidazotiadiazol; composición farmacéutica que los comprende; útiles para el tratamiento de la epilepsia, transtornos neurológicos, entre otros. | |
NZ730985A (en) | Use of cannabinoids in the treatment of degenerative skeletal muscle diseases | |
CL2015000434A1 (es) | Metodo para el tratamiento, prevencion o disminucion de la severidad de una condicion o trastorno no neoplasico de la piel que comprende administrar un compuesto derivado de retinoides; composicion dermica que comprende los derivados de retinoide. | |
BR112015000051A2 (pt) | tratamento de distúrbios inflamatórios da pele | |
AR119043A1 (es) | Métodos para acelerar la cicatrización mediante el uso de composiciones cannabinoides | |
BR112015010186A2 (pt) | sulfonamida cíclica contendo derivados como inibidores da via de sinalização de hedgehog | |
BR112014007922A2 (pt) | nanocápsulas de oxoisoaporfinas para o tratamento da depressão | |
MX2022004888A (es) | (-)-cis tetrahidrocannabinol ((-)-cis-thc) para uso como medicamento. | |
TH153696A (th) | การใช้ไฟโตแคนนาบินอยด์หรือสารผสมของสารดังกล่าวในการรักษาโรคลมบ้าหมู |