EA200500301A1 - NEW CARBOXAMIDE COMPOUNDS, HAVING ANTAGONISTIC CONCERNING THE SITTING OF SITES, CONTAINING THESE CONNECTIONS MEDICINES AND METHOD OF THEIR PRODUCTION - Google Patents

NEW CARBOXAMIDE COMPOUNDS, HAVING ANTAGONISTIC CONCERNING THE SITTING OF SITES, CONTAINING THESE CONNECTIONS MEDICINES AND METHOD OF THEIR PRODUCTION

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Publication number
EA200500301A1
EA200500301A1 EA200500301A EA200500301A EA200500301A1 EA 200500301 A1 EA200500301 A1 EA 200500301A1 EA 200500301 A EA200500301 A EA 200500301A EA 200500301 A EA200500301 A EA 200500301A EA 200500301 A1 EA200500301 A1 EA 200500301A1
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EA
Eurasian Patent Office
Prior art keywords
carboxamide compounds
antagonistic
sitting
medicines
concerning
Prior art date
Application number
EA200500301A
Other languages
Russian (ru)
Other versions
EA012834B1 (en
Inventor
Торстен Леманн-Линтц
Дирк Штенкамп
Мартин Лентер
Хайке-Андреа Виланд
Клаус Рудольф
Штефан Георг Мюллер
Ральф Р.Х. Лотц
Кирстен Арндт
Филипп Лустенбергер
Original Assignee
Бёрингер Ингельхайм Фарма Гмбх Унд Ко. Кг
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Application filed by Бёрингер Ингельхайм Фарма Гмбх Унд Ко. Кг filed Critical Бёрингер Ингельхайм Фарма Гмбх Унд Ко. Кг
Publication of EA200500301A1 publication Critical patent/EA200500301A1/en
Publication of EA012834B1 publication Critical patent/EA012834B1/en

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Abstract

В заявке описаны карбоксамидные соединения общей формулы (I)в которой группы и остатки A, B, W, X, Y, Z, R, R, Rи k имеют указанные в п.1 формулы изобретения значения. В заявке описаны далее способ получения таких карбоксамидных соединений, а также лекарственные средства, содержащие по меньшей мере одно предлагаемое в изобретении карбоксамидное соединение. Предлагаемые в изобретении лекарственные средства благодаря наличию у них антагонистической в отношении MCH-рецептора активности пригодны для лечения связанных с нарушением обмена веществ расстройств и/или расстройств приема пищи, прежде всего ожирения, булимии, анорексии, гиперфагии и диабета.Международная заявка была опубликована вместе с отчетом о международном поиске.The application describes carboxamide compounds of general formula (I) in which the groups and residues A, B, W, X, Y, Z, R, R, R and k have the meanings indicated in claim 1. The application further describes a method for producing such carboxamide compounds, as well as medicaments containing at least one carboxamide compound according to the invention. Due to their antagonistic activity against the MCH receptor, the drugs according to the invention are suitable for treating metabolic disorders and / or eating disorders, especially obesity, bulimia, anorexia, hyperphagia and diabetes. The international application was published with international search report.

EA200500301A 2002-08-24 2003-08-16 Novel carboxamide compounds having an mch-antagonistic effect, medicaments containing said compounds, and methods for the production thereof EA012834B1 (en)

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AR043046A1 (en) 2005-07-13
HRP20050179A2 (en) 2006-05-31
MXPA05002158A (en) 2005-05-23
EA012834B1 (en) 2009-12-30
RS20050173A (en) 2007-09-21
CN1678591A (en) 2005-10-05
UA82853C2 (en) 2008-05-26
PL375344A1 (en) 2005-11-28
NO20050068L (en) 2005-03-04
WO2004024702A1 (en) 2004-03-25
TW200413332A (en) 2004-08-01
PE20040974A1 (en) 2005-01-12

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