EA200100515A3 - Диазепиноиндолы для лечения хронического обструктивного заболевания легких - Google Patents

Диазепиноиндолы для лечения хронического обструктивного заболевания легких

Info

Publication number
EA200100515A3
EA200100515A3 EA200100515A EA200100515A EA200100515A3 EA 200100515 A3 EA200100515 A3 EA 200100515A3 EA 200100515 A EA200100515 A EA 200100515A EA 200100515 A EA200100515 A EA 200100515A EA 200100515 A3 EA200100515 A3 EA 200100515A3
Authority
EA
Eurasian Patent Office
Prior art keywords
treatment
chronic obstructive
diazepinoindols
lung diseases
obstructive lung
Prior art date
Application number
EA200100515A
Other languages
English (en)
Other versions
EA200100515A2 (ru
Inventor
Аннетт Доуэрти
Original Assignee
Уорнер-Ламберт Компани
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Уорнер-Ламберт Компани filed Critical Уорнер-Ламберт Компани
Publication of EA200100515A2 publication Critical patent/EA200100515A2/ru
Publication of EA200100515A3 publication Critical patent/EA200100515A3/ru

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A61K31/55131,4-Benzodiazepines, e.g. diazepam or clozapine
    • A61K31/55171,4-Benzodiazepines, e.g. diazepam or clozapine condensed with five-membered rings having nitrogen as a ring hetero atom, e.g. imidazobenzodiazepines, triazolam
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/02Nasal agents, e.g. decongestants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pulmonology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Настоящее изобретение относится к применению диазепиноиндолов формулыв которой А представляет собой азотсодержащий гетероарил, а В представляет собой гидроксильный или аминорадикал, для лечения хронического обструктивного заболевания легких.
EA200100515A 2000-06-09 2001-06-06 Диазепиноиндолы для лечения хронического обструктивного заболевания легких EA200100515A3 (ru)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP00401646A EP1161949A1 (en) 2000-06-09 2000-06-09 Use od diazepinoindoles for the treatment of chronic obstructive pulmonary disease

Publications (2)

Publication Number Publication Date
EA200100515A2 EA200100515A2 (ru) 2001-12-24
EA200100515A3 true EA200100515A3 (ru) 2002-06-27

Family

ID=8173724

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200100515A EA200100515A3 (ru) 2000-06-09 2001-06-06 Диазепиноиндолы для лечения хронического обструктивного заболевания легких

Country Status (19)

Country Link
US (1) US6544983B2 (ru)
EP (1) EP1161949A1 (ru)
JP (1) JP2002138090A (ru)
KR (1) KR20010111457A (ru)
CN (1) CN1345725A (ru)
AR (1) AR030291A1 (ru)
AU (1) AU5181301A (ru)
BR (1) BR0102289A (ru)
CA (1) CA2347337A1 (ru)
CZ (1) CZ20011999A3 (ru)
EA (1) EA200100515A3 (ru)
HU (1) HUP0102388A3 (ru)
IL (1) IL143636A0 (ru)
MX (1) MXPA01005726A (ru)
NO (1) NO20012831L (ru)
NZ (1) NZ512222A (ru)
PL (1) PL347922A1 (ru)
SK (1) SK7832001A3 (ru)
ZA (1) ZA200104616B (ru)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20050085430A1 (en) * 2003-07-31 2005-04-21 Robinson Cynthia B. Combination of dehydroepiandrosterone or dehydroepiandrosterone-sulfate with a PDE-4 inhibitor for treatment of asthma or chronic obstructive pulmonary disease
US20050026883A1 (en) * 2003-07-31 2005-02-03 Robinson Cynthia B. Combination of dehydroepiandrosterone or dehydroepiandrosterone-sulfate with a PDE-4 inhibitor for treatment of asthma or chronic obstructive pulmonary disease
US20090274676A1 (en) * 2003-07-31 2009-11-05 Robinson Cynthia B Combination of dehydroepiandrosterone or dehydroepiandrosterone-sulfate with a pde-4 inhibitor for treatment of asthma or chronic obstructive pulmonary disease
US20050187278A1 (en) * 2003-08-28 2005-08-25 Pharmacia Corporation Treatment or prevention of vascular disorders with Cox-2 inhibitors in combination with cyclic AMP-specific phosphodiesterase inhibitors
CA2544322C (en) * 2003-11-20 2012-05-08 Astellas Pharma Inc. Agent for treating chronic pelvic pain syndrome
DE102004002557A1 (de) * 2004-01-17 2005-08-04 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verwendung von substituierten Pyrimido(5,4-d)pyrimidinen zur Behandlung von Atemwegserkrankungen
KR20090045233A (ko) 2006-07-10 2009-05-07 파이온 유케이 리미티드 속효형 벤조디아제핀 염 및 이의 중합체 형태
US8426673B2 (en) 2008-01-11 2013-04-23 Astellas Pharma, Inc. Pathological animal model for pelvic pain syndrome
EP2450039A1 (en) 2010-11-08 2012-05-09 PAION UK Ltd. Dosing regimen for sedation with CNS 7056 (Remimazolam)
US20150148338A1 (en) * 2012-05-22 2015-05-28 Paion Uk Limited Compositions comprising short-acting benzodiazepines
AR094963A1 (es) 2013-03-04 2015-09-09 Ono Pharmaceutical Co Reacción de oxidación excelente en el índice de conversión

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2652352A1 (fr) 1989-09-28 1991-03-29 Jouveinal Sa Benzodiazepines, leur procede et intermediaires de preparation et leurs applications en therapeutique.
FR2725719B1 (fr) 1994-10-14 1996-12-06 Jouveinal Inst Rech Diazepino-indoles inhibiteurs de phosphodiesterases iv
FR2746800B1 (fr) * 1996-03-29 1998-06-05 Jouveinal Inst Rech Diazepino-indoles inhibiteurs de phosphodiesterases 4
FR2762841B1 (fr) 1997-04-30 1999-07-02 Jouveinal Inst Rech Diazepino-indolones inhibitrices de phosphodiesterases iv

Also Published As

Publication number Publication date
EA200100515A2 (ru) 2001-12-24
AR030291A1 (es) 2003-08-20
US6544983B2 (en) 2003-04-08
SK7832001A3 (en) 2002-05-09
IL143636A0 (en) 2002-04-21
KR20010111457A (ko) 2001-12-19
JP2002138090A (ja) 2002-05-14
CA2347337A1 (en) 2001-12-09
MXPA01005726A (es) 2003-08-20
NZ512222A (en) 2002-10-25
CZ20011999A3 (cs) 2002-04-17
NO20012831D0 (no) 2001-06-08
HUP0102388A2 (hu) 2002-04-29
ZA200104616B (en) 2002-10-30
PL347922A1 (en) 2001-12-17
BR0102289A (pt) 2002-03-12
HU0102388D0 (en) 2001-08-28
AU5181301A (en) 2001-12-13
NO20012831L (no) 2001-12-10
US20020010175A1 (en) 2002-01-24
EP1161949A1 (en) 2001-12-12
CN1345725A (zh) 2002-04-24
HUP0102388A3 (en) 2004-11-29

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