EA200100515A3 - Диазепиноиндолы для лечения хронического обструктивного заболевания легких - Google Patents
Диазепиноиндолы для лечения хронического обструктивного заболевания легкихInfo
- Publication number
- EA200100515A3 EA200100515A3 EA200100515A EA200100515A EA200100515A3 EA 200100515 A3 EA200100515 A3 EA 200100515A3 EA 200100515 A EA200100515 A EA 200100515A EA 200100515 A EA200100515 A EA 200100515A EA 200100515 A3 EA200100515 A3 EA 200100515A3
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- treatment
- chronic obstructive
- diazepinoindols
- lung diseases
- obstructive lung
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
- A61K31/5513—1,4-Benzodiazepines, e.g. diazepam or clozapine
- A61K31/5517—1,4-Benzodiazepines, e.g. diazepam or clozapine condensed with five-membered rings having nitrogen as a ring hetero atom, e.g. imidazobenzodiazepines, triazolam
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Pulmonology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Настоящее изобретение относится к применению диазепиноиндолов формулыв которой А представляет собой азотсодержащий гетероарил, а В представляет собой гидроксильный или аминорадикал, для лечения хронического обструктивного заболевания легких.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP00401646A EP1161949A1 (en) | 2000-06-09 | 2000-06-09 | Use od diazepinoindoles for the treatment of chronic obstructive pulmonary disease |
Publications (2)
Publication Number | Publication Date |
---|---|
EA200100515A2 EA200100515A2 (ru) | 2001-12-24 |
EA200100515A3 true EA200100515A3 (ru) | 2002-06-27 |
Family
ID=8173724
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200100515A EA200100515A3 (ru) | 2000-06-09 | 2001-06-06 | Диазепиноиндолы для лечения хронического обструктивного заболевания легких |
Country Status (19)
Country | Link |
---|---|
US (1) | US6544983B2 (ru) |
EP (1) | EP1161949A1 (ru) |
JP (1) | JP2002138090A (ru) |
KR (1) | KR20010111457A (ru) |
CN (1) | CN1345725A (ru) |
AR (1) | AR030291A1 (ru) |
AU (1) | AU5181301A (ru) |
BR (1) | BR0102289A (ru) |
CA (1) | CA2347337A1 (ru) |
CZ (1) | CZ20011999A3 (ru) |
EA (1) | EA200100515A3 (ru) |
HU (1) | HUP0102388A3 (ru) |
IL (1) | IL143636A0 (ru) |
MX (1) | MXPA01005726A (ru) |
NO (1) | NO20012831L (ru) |
NZ (1) | NZ512222A (ru) |
PL (1) | PL347922A1 (ru) |
SK (1) | SK7832001A3 (ru) |
ZA (1) | ZA200104616B (ru) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20050026883A1 (en) * | 2003-07-31 | 2005-02-03 | Robinson Cynthia B. | Combination of dehydroepiandrosterone or dehydroepiandrosterone-sulfate with a PDE-4 inhibitor for treatment of asthma or chronic obstructive pulmonary disease |
US20050085430A1 (en) * | 2003-07-31 | 2005-04-21 | Robinson Cynthia B. | Combination of dehydroepiandrosterone or dehydroepiandrosterone-sulfate with a PDE-4 inhibitor for treatment of asthma or chronic obstructive pulmonary disease |
US20090274676A1 (en) * | 2003-07-31 | 2009-11-05 | Robinson Cynthia B | Combination of dehydroepiandrosterone or dehydroepiandrosterone-sulfate with a pde-4 inhibitor for treatment of asthma or chronic obstructive pulmonary disease |
US20050187278A1 (en) * | 2003-08-28 | 2005-08-25 | Pharmacia Corporation | Treatment or prevention of vascular disorders with Cox-2 inhibitors in combination with cyclic AMP-specific phosphodiesterase inhibitors |
CA2544322C (en) * | 2003-11-20 | 2012-05-08 | Astellas Pharma Inc. | Agent for treating chronic pelvic pain syndrome |
DE102004002557A1 (de) * | 2004-01-17 | 2005-08-04 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Verwendung von substituierten Pyrimido(5,4-d)pyrimidinen zur Behandlung von Atemwegserkrankungen |
KR20150081370A (ko) | 2006-07-10 | 2015-07-13 | 파이온 유케이 리미티드 | 속효형 벤조디아제핀 염 및 이의 중합체 형태 |
JP5240205B2 (ja) | 2008-01-11 | 2013-07-17 | アステラス製薬株式会社 | 精巣の疼痛又は不快感行動及び頻尿併発モデル動物 |
EP2450039A1 (en) | 2010-11-08 | 2012-05-09 | PAION UK Ltd. | Dosing regimen for sedation with CNS 7056 (Remimazolam) |
MX368854B (es) * | 2012-05-22 | 2019-10-18 | Paion Uk Ltd | Composiciones que comprenden benzodiazepinas de acción corta. |
AR094963A1 (es) | 2013-03-04 | 2015-09-09 | Ono Pharmaceutical Co | Reacción de oxidación excelente en el índice de conversión |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2652352A1 (fr) | 1989-09-28 | 1991-03-29 | Jouveinal Sa | Benzodiazepines, leur procede et intermediaires de preparation et leurs applications en therapeutique. |
FR2725719B1 (fr) | 1994-10-14 | 1996-12-06 | Jouveinal Inst Rech | Diazepino-indoles inhibiteurs de phosphodiesterases iv |
FR2746800B1 (fr) * | 1996-03-29 | 1998-06-05 | Jouveinal Inst Rech | Diazepino-indoles inhibiteurs de phosphodiesterases 4 |
FR2762841B1 (fr) | 1997-04-30 | 1999-07-02 | Jouveinal Inst Rech | Diazepino-indolones inhibitrices de phosphodiesterases iv |
-
2000
- 2000-06-09 EP EP00401646A patent/EP1161949A1/en not_active Withdrawn
-
2001
- 2001-05-11 CA CA002347337A patent/CA2347337A1/en not_active Abandoned
- 2001-06-05 CZ CZ20011999A patent/CZ20011999A3/cs unknown
- 2001-06-06 EA EA200100515A patent/EA200100515A3/ru unknown
- 2001-06-06 PL PL01347922A patent/PL347922A1/xx not_active Application Discontinuation
- 2001-06-06 ZA ZA200104616A patent/ZA200104616B/xx unknown
- 2001-06-07 BR BR0102289-0A patent/BR0102289A/pt not_active IP Right Cessation
- 2001-06-07 US US09/876,719 patent/US6544983B2/en not_active Expired - Fee Related
- 2001-06-07 AU AU51813/01A patent/AU5181301A/en not_active Abandoned
- 2001-06-07 NZ NZ512222A patent/NZ512222A/xx unknown
- 2001-06-07 MX MXPA01005726A patent/MXPA01005726A/es unknown
- 2001-06-07 SK SK783-2001A patent/SK7832001A3/sk unknown
- 2001-06-07 AR ARP010102725A patent/AR030291A1/es not_active Application Discontinuation
- 2001-06-07 IL IL14363601A patent/IL143636A0/xx unknown
- 2001-06-08 NO NO20012831A patent/NO20012831L/no not_active Application Discontinuation
- 2001-06-08 HU HU0102388A patent/HUP0102388A3/hu unknown
- 2001-06-08 CN CN01120850A patent/CN1345725A/zh active Pending
- 2001-06-08 KR KR1020010031887A patent/KR20010111457A/ko not_active Application Discontinuation
- 2001-06-08 JP JP2001174372A patent/JP2002138090A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
NO20012831L (no) | 2001-12-10 |
AR030291A1 (es) | 2003-08-20 |
KR20010111457A (ko) | 2001-12-19 |
CN1345725A (zh) | 2002-04-24 |
HUP0102388A3 (en) | 2004-11-29 |
ZA200104616B (en) | 2002-10-30 |
US6544983B2 (en) | 2003-04-08 |
PL347922A1 (en) | 2001-12-17 |
EA200100515A2 (ru) | 2001-12-24 |
MXPA01005726A (es) | 2003-08-20 |
EP1161949A1 (en) | 2001-12-12 |
HUP0102388A2 (hu) | 2002-04-29 |
HU0102388D0 (en) | 2001-08-28 |
CZ20011999A3 (cs) | 2002-04-17 |
BR0102289A (pt) | 2002-03-12 |
IL143636A0 (en) | 2002-04-21 |
CA2347337A1 (en) | 2001-12-09 |
SK7832001A3 (en) | 2002-05-09 |
JP2002138090A (ja) | 2002-05-14 |
US20020010175A1 (en) | 2002-01-24 |
NO20012831D0 (no) | 2001-06-08 |
NZ512222A (en) | 2002-10-25 |
AU5181301A (en) | 2001-12-13 |
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