EA029745B9 - Конденсированные соединения имидазобензотиазола - Google Patents
Конденсированные соединения имидазобензотиазолаInfo
- Publication number
- EA029745B9 EA029745B9 EA201691920A EA201691920A EA029745B9 EA 029745 B9 EA029745 B9 EA 029745B9 EA 201691920 A EA201691920 A EA 201691920A EA 201691920 A EA201691920 A EA 201691920A EA 029745 B9 EA029745 B9 EA 029745B9
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- compounds
- pharmaceutically acceptable
- present
- fused imidazobenzothiazole
- fused
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/429—Thiazoles condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Pulmonology (AREA)
- Epidemiology (AREA)
- Immunology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Saccharide Compounds (AREA)
Abstract
Настоящее изобретение относится к новым конденсированным производным имидазобензотиазола, их фармацевтически приемлемым солям и их изомерам, стереоизомерам, атропизомерам, конформерам, таутомерам, полиморфам, гидратам, сольватам и N-оксиду. Настоящее изобретение охватывает также фармацевтически приемлемые композиции указанных соединений и способ получения новых соединений. Кроме того, изобретение относится к применению вышеупомянутых соединений для получения лекарственного препарата для применения в качестве фармацевтических препаратов.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN1089MU2014 | 2014-03-27 | ||
PCT/IB2015/052124 WO2015145336A1 (en) | 2014-03-27 | 2015-03-24 | Novel fused imidazobenzothiazole compounds |
Publications (3)
Publication Number | Publication Date |
---|---|
EA201691920A1 EA201691920A1 (ru) | 2017-01-30 |
EA029745B1 EA029745B1 (ru) | 2018-05-31 |
EA029745B9 true EA029745B9 (ru) | 2018-08-31 |
Family
ID=54194050
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201691920A EA029745B9 (ru) | 2014-03-27 | 2015-03-24 | Конденсированные соединения имидазобензотиазола |
Country Status (29)
Country | Link |
---|---|
US (2) | US9908898B2 (ru) |
EP (1) | EP3122755B1 (ru) |
JP (1) | JP6480949B2 (ru) |
KR (1) | KR102339610B1 (ru) |
CN (1) | CN106414458B (ru) |
AR (1) | AR099867A1 (ru) |
AU (1) | AU2015237840B2 (ru) |
CA (1) | CA2943098C (ru) |
CY (1) | CY1121147T1 (ru) |
DK (1) | DK3122755T3 (ru) |
EA (1) | EA029745B9 (ru) |
ES (1) | ES2707099T3 (ru) |
HR (1) | HRP20190121T1 (ru) |
HU (1) | HUE042493T2 (ru) |
IL (1) | IL247955B (ru) |
LT (1) | LT3122755T (ru) |
MX (1) | MX368985B (ru) |
MY (1) | MY193041A (ru) |
PH (1) | PH12016501903B1 (ru) |
PL (1) | PL3122755T3 (ru) |
PT (1) | PT3122755T (ru) |
RS (1) | RS58324B1 (ru) |
SG (1) | SG11201607793RA (ru) |
SI (1) | SI3122755T1 (ru) |
TR (1) | TR201900735T4 (ru) |
TW (1) | TWI648282B (ru) |
UA (1) | UA121469C2 (ru) |
WO (1) | WO2015145336A1 (ru) |
ZA (1) | ZA201606598B (ru) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN105073728A (zh) | 2013-03-15 | 2015-11-18 | 全球血液疗法股份有限公司 | 化合物及其用于调节血红蛋白的用途 |
EA202092627A1 (ru) | 2013-11-18 | 2021-09-30 | Глобал Блад Терапьютикс, Инк. | Соединения и их применения для модуляции гемоглобина |
TWI648282B (zh) * | 2014-03-27 | 2019-01-21 | 印度商托仁特生技有限公司 | 新熔合咪唑苯并噻唑化合物 |
DE102016209204A1 (de) | 2016-05-27 | 2017-11-30 | Robert Bosch Gmbh | Vorrichtung zur Regelung mindestens eines Fluidstroms in einem Fahrzeug |
KR102630959B1 (ko) * | 2016-10-31 | 2024-01-29 | 엘지디스플레이 주식회사 | 유기 화합물과 이를 이용한 발광다이오드 및 유기발광다이오드 표시장치 |
CN106727538A (zh) * | 2017-02-20 | 2017-05-31 | 潘连香 | 一种治疗2型糖尿病的药物组合物 |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8724566D0 (en) | 1987-10-20 | 1987-11-25 | Roussel Lab Ltd | Chemical compounds |
GB8908845D0 (en) | 1989-04-19 | 1989-06-07 | Roussel Lab Ltd | Chemical compounds |
JPH09512548A (ja) * | 1994-04-29 | 1997-12-16 | ファルマシア・アンド・アップジョン・カンパニー | レトロウイルス感染、特にhiv感染の治療のためのメタノール誘導体 |
WO2002014321A1 (en) * | 2000-08-11 | 2002-02-21 | The Regents Of The University Of California | Use of stat-6 inhibitors as therapeutic agents |
US7601846B2 (en) * | 2001-06-26 | 2009-10-13 | The Regents Of The University Of California | Compounds having activity as inhibitors of apoptosis |
CA2506796A1 (en) * | 2002-11-25 | 2004-06-10 | Pharmacia Corporation | Heteroarylsulfonylmethyl hydroxamic acids and amides and their use as protease inhibitors |
GB0320244D0 (en) * | 2003-05-06 | 2003-10-01 | Aventis Pharma Inc | Pyrazoles as inhibitors of tumour necrosis factor |
CA2642209A1 (en) * | 2006-02-09 | 2007-08-16 | Pfizer Limited | Triazolopyridine compounds |
TWI648282B (zh) * | 2014-03-27 | 2019-01-21 | 印度商托仁特生技有限公司 | 新熔合咪唑苯并噻唑化合物 |
-
2015
- 2015-03-16 TW TW104108329A patent/TWI648282B/zh active
- 2015-03-24 TR TR2019/00735T patent/TR201900735T4/tr unknown
- 2015-03-24 PT PT15717242T patent/PT3122755T/pt unknown
- 2015-03-24 EA EA201691920A patent/EA029745B9/ru not_active IP Right Cessation
- 2015-03-24 CA CA2943098A patent/CA2943098C/en active Active
- 2015-03-24 DK DK15717242.0T patent/DK3122755T3/en active
- 2015-03-24 WO PCT/IB2015/052124 patent/WO2015145336A1/en active Application Filing
- 2015-03-24 SG SG11201607793RA patent/SG11201607793RA/en unknown
- 2015-03-24 JP JP2016559356A patent/JP6480949B2/ja not_active Expired - Fee Related
- 2015-03-24 ES ES15717242T patent/ES2707099T3/es active Active
- 2015-03-24 EP EP15717242.0A patent/EP3122755B1/en active Active
- 2015-03-24 KR KR1020167029134A patent/KR102339610B1/ko active IP Right Grant
- 2015-03-24 UA UAA201610628A patent/UA121469C2/uk unknown
- 2015-03-24 MY MYPI2016703533A patent/MY193041A/en unknown
- 2015-03-24 RS RS20190084A patent/RS58324B1/sr unknown
- 2015-03-24 MX MX2016012535A patent/MX368985B/es active IP Right Grant
- 2015-03-24 CN CN201580024068.6A patent/CN106414458B/zh not_active Expired - Fee Related
- 2015-03-24 SI SI201530555T patent/SI3122755T1/sl unknown
- 2015-03-24 HU HUE15717242A patent/HUE042493T2/hu unknown
- 2015-03-24 AU AU2015237840A patent/AU2015237840B2/en not_active Ceased
- 2015-03-24 US US15/128,886 patent/US9908898B2/en active Active
- 2015-03-24 PL PL15717242T patent/PL3122755T3/pl unknown
- 2015-03-24 LT LTEP15717242.0T patent/LT3122755T/lt unknown
- 2015-03-27 AR ARP150100915A patent/AR099867A1/es not_active Application Discontinuation
-
2016
- 2016-09-21 IL IL247955A patent/IL247955B/en active IP Right Grant
- 2016-09-23 ZA ZA2016/06598A patent/ZA201606598B/en unknown
- 2016-09-27 PH PH12016501903A patent/PH12016501903B1/en unknown
-
2018
- 2018-01-03 US US15/861,399 patent/US10227361B2/en active Active
-
2019
- 2019-01-21 HR HRP20190121TT patent/HRP20190121T1/hr unknown
- 2019-01-21 CY CY20191100076T patent/CY1121147T1/el unknown
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
TH4A | Publication of the corrected specification to eurasian patent | ||
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AM AZ BY KZ KG TJ TM |