EA027350B1 - Способ лечения или предупреждения приливов и ночной потливости у женщин в менопаузе - Google Patents
Способ лечения или предупреждения приливов и ночной потливости у женщин в менопаузе Download PDFInfo
- Publication number
- EA027350B1 EA027350B1 EA201290851A EA201290851A EA027350B1 EA 027350 B1 EA027350 B1 EA 027350B1 EA 201290851 A EA201290851 A EA 201290851A EA 201290851 A EA201290851 A EA 201290851A EA 027350 B1 EA027350 B1 EA 027350B1
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- EA
- Eurasian Patent Office
- Prior art keywords
- dextromethorphan
- dextrorphan
- hot flashes
- microparticles
- night sweats
- Prior art date
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/12—Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
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- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Diabetes (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
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| US30963810P | 2010-03-02 | 2010-03-02 | |
| PCT/US2011/026650 WO2011109367A2 (en) | 2010-03-02 | 2011-03-01 | Methods and compositions for treating or preventing symptoms of hormonal variations |
Publications (2)
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| EA201290851A1 EA201290851A1 (ru) | 2013-04-30 |
| EA027350B1 true EA027350B1 (ru) | 2017-07-31 |
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| EA201290851A EA027350B1 (ru) | 2010-03-02 | 2011-03-01 | Способ лечения или предупреждения приливов и ночной потливости у женщин в менопаузе |
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| EP (1) | EP2542241B1 (enExample) |
| JP (1) | JP5839362B2 (enExample) |
| CN (1) | CN102858343B (enExample) |
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| IL (2) | IL221706A (enExample) |
| PL (1) | PL2542241T3 (enExample) |
| WO (1) | WO2011109367A2 (enExample) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US9616123B1 (en) * | 2012-03-05 | 2017-04-11 | Robert L. Knobler | Method and compound for treatment of menopausal symptoms |
| CN107249615B (zh) * | 2015-04-07 | 2021-02-05 | 株式会社明治 | 潮热抑制剂 |
| US11491120B2 (en) | 2017-11-09 | 2022-11-08 | The Trustees Of Columbia University In The City Of New York | Pharmacological prophylactics against stress-induced affective disorders in females |
| US11622948B2 (en) | 2017-11-09 | 2023-04-11 | The Trustees Of Columbia University In The City Of New York | Biomarkers for efficacy of prophylactic treatments against stress-induced affective disorders |
| WO2020219270A1 (en) * | 2019-04-22 | 2020-10-29 | Knobler Robert L | Non-hormonal treatment of hot flashes |
| WO2021108801A2 (en) * | 2019-11-15 | 2021-06-03 | Consegna Pharma, Inc. | Long acting nmda antagonists |
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| US20040259850A1 (en) * | 2001-10-31 | 2004-12-23 | Alves Stephen E. | Method for treating or preventing symptoms of hormonal variation including hot flashes |
| US20080146541A1 (en) * | 2006-12-13 | 2008-06-19 | Hung-Ming Wu | Methods for treating or preventing sysmptoms of hormonal variations |
| US20090053329A1 (en) * | 2007-03-19 | 2009-02-26 | Acadia Pharmaceuticals, Inc. | Combinations of 5-ht2a inverse agonists and antagonists with antipsychotics |
| US20090111846A1 (en) * | 2006-02-03 | 2009-04-30 | Avanir Pharmaceuticals | Pharmaceutical compositions comprising dextromethorphan and quinidine for the treatment of depression, anxiety, and neurodegenerative disorders |
| US20090111817A1 (en) * | 2005-07-06 | 2009-04-30 | Sepracor Inc. | Combinations of Eszopiclone and an Antidepressant |
| WO2010011767A2 (en) * | 2008-07-22 | 2010-01-28 | Duke Debra M | Compositions and methods for treating symptoms associated with menopause, hormonal variations and arthritis |
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| US5321012A (en) * | 1993-01-28 | 1994-06-14 | Virginia Commonwealth University Medical College | Inhibiting the development of tolerance to and/or dependence on a narcotic addictive substance |
| CA2115792C (en) * | 1993-03-05 | 2005-11-01 | David J. Mayer | Method for the treatment of pain |
| AUPN605795A0 (en) * | 1995-10-19 | 1995-11-09 | F.H. Faulding & Co. Limited | Analgesic pharmaceutical composition |
| DE60034344T2 (de) * | 1999-07-22 | 2008-01-10 | University Of Rochester | Methode zur behandlung der symptome hormoneller veränderungen, einschliesslich hitzewallungen |
| US20040002482A1 (en) * | 2000-08-30 | 2004-01-01 | Dudley Robert E. | Androgen pharmaceutical composition and method for treating depression |
| US6569471B2 (en) * | 2000-09-01 | 2003-05-27 | Natumin Pharma Ab | Method for the treatment of symptoms related to normal hormonal variations in women |
| US20050129783A1 (en) * | 2001-04-19 | 2005-06-16 | Mccleary Edward L. | Composition and method for treatment of neurophysiological conditions and maintenance of neurophysiological health |
| UA81423C2 (en) * | 2002-08-15 | 2008-01-10 | PRODUCT CONTAINING SRI AND AGONIST OF THE 5HT2a RECEPTOR FOR TREATMENT OF THERMOREGULATORY DYSFUNCTION | |
| HUP0303313A2 (hu) * | 2003-10-09 | 2005-07-28 | Richter Gedeon Vegyészeti Gyár Rt. | Transzdermális gyógyszerkészítmények |
| US7855195B2 (en) * | 2003-12-02 | 2010-12-21 | Pharmaneuroboost N.V. | Method of treating mental disorders using D4 and 5-HT2A antagonists, inverse agonists or partial agonists |
| JP2007537232A (ja) * | 2004-05-11 | 2007-12-20 | ファイザー・プロダクツ・インク | 非定型抗精神病薬と５−ｈｔ１ｂ受容体拮抗薬の組合せ |
| WO2005120523A1 (en) * | 2004-06-04 | 2005-12-22 | Mood Management Sciences, Llc | Methods and compositions for treating mood disorder |
| US20060122127A1 (en) * | 2004-11-17 | 2006-06-08 | Cypress Bioscience, Inc. | Methods for reducing the side effects associated with mirtzapine treatment |
| MX2008007589A (es) * | 2005-12-13 | 2009-01-27 | Trinity Lab Inc | Un metodo para tratar eyaculacion prematura en seres humanos. |
-
2011
- 2011-03-01 PL PL11751180.8T patent/PL2542241T3/pl unknown
- 2011-03-01 JP JP2012556166A patent/JP5839362B2/ja active Active
- 2011-03-01 CN CN201180020427.2A patent/CN102858343B/zh active Active
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- 2011-03-01 ES ES11751180.8T patent/ES2574210T3/es active Active
- 2011-03-01 EA EA201290851A patent/EA027350B1/ru unknown
- 2011-03-01 AU AU2011223807A patent/AU2011223807B2/en active Active
- 2011-03-01 US US13/037,728 patent/US20110218213A1/en not_active Abandoned
- 2011-03-01 BR BR112012022052-7A patent/BR112012022052B1/pt active IP Right Grant
- 2011-03-01 WO PCT/US2011/026650 patent/WO2011109367A2/en not_active Ceased
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2012
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2018
- 2018-07-12 AU AU2018205147A patent/AU2018205147A1/en not_active Abandoned
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| US5654008A (en) * | 1993-11-19 | 1997-08-05 | Alkermes Controlled Therapeutics Inc. Ii | Preparation of biodegradable microparticles containing a biologically active agent |
| US20040259850A1 (en) * | 2001-10-31 | 2004-12-23 | Alves Stephen E. | Method for treating or preventing symptoms of hormonal variation including hot flashes |
| US20090111817A1 (en) * | 2005-07-06 | 2009-04-30 | Sepracor Inc. | Combinations of Eszopiclone and an Antidepressant |
| US20090111846A1 (en) * | 2006-02-03 | 2009-04-30 | Avanir Pharmaceuticals | Pharmaceutical compositions comprising dextromethorphan and quinidine for the treatment of depression, anxiety, and neurodegenerative disorders |
| US20080146541A1 (en) * | 2006-12-13 | 2008-06-19 | Hung-Ming Wu | Methods for treating or preventing sysmptoms of hormonal variations |
| US20090053329A1 (en) * | 2007-03-19 | 2009-02-26 | Acadia Pharmaceuticals, Inc. | Combinations of 5-ht2a inverse agonists and antagonists with antipsychotics |
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Also Published As
| Publication number | Publication date |
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| EP2542241B1 (en) | 2016-04-27 |
| PL2542241T3 (pl) | 2016-12-30 |
| US20110218213A1 (en) | 2011-09-08 |
| EP2542241A2 (en) | 2013-01-09 |
| IL253853B (en) | 2019-05-30 |
| AU2011223807B2 (en) | 2016-05-12 |
| IL253853A0 (en) | 2017-09-28 |
| CA2828041C (en) | 2018-04-17 |
| AU2016213776B2 (en) | 2018-04-12 |
| IL221706A (en) | 2017-08-31 |
| CN102858343B (zh) | 2015-11-25 |
| AU2016213776A1 (en) | 2016-09-01 |
| WO2011109367A2 (en) | 2011-09-09 |
| ES2574210T3 (es) | 2016-06-15 |
| AU2018205147A1 (en) | 2018-08-02 |
| AU2011223807A1 (en) | 2012-10-18 |
| JP2013521297A (ja) | 2013-06-10 |
| WO2011109367A3 (en) | 2011-12-29 |
| CN102858343A (zh) | 2013-01-02 |
| WO2011109367A4 (en) | 2012-02-23 |
| BR112012022052A2 (pt) | 2020-07-07 |
| EA201290851A1 (ru) | 2013-04-30 |
| BR112012022052B1 (pt) | 2021-06-29 |
| JP5839362B2 (ja) | 2016-01-06 |
| CA2828041A1 (en) | 2011-09-09 |
| EP2542241A4 (en) | 2013-11-06 |
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