DK611987D0 - CEPHALOSPORINE DERIVATIVES AND PROCEDURES FOR PREPARING THEREOF AND PHARMACEUTICAL AGENTS CONTAINING THE DERIVATIVES - Google Patents

CEPHALOSPORINE DERIVATIVES AND PROCEDURES FOR PREPARING THEREOF AND PHARMACEUTICAL AGENTS CONTAINING THE DERIVATIVES

Info

Publication number
DK611987D0
DK611987D0 DK611987A DK611987A DK611987D0 DK 611987 D0 DK611987 D0 DK 611987D0 DK 611987 A DK611987 A DK 611987A DK 611987 A DK611987 A DK 611987A DK 611987 D0 DK611987 D0 DK 611987D0
Authority
DK
Denmark
Prior art keywords
derivatives
procedures
preparing
pharmaceutical agents
agents containing
Prior art date
Application number
DK611987A
Other languages
Danish (da)
Other versions
DK611987A (en
Inventor
Dominique Olliero
Bernard Labeeuw
Gilles Roche
Ali Salhi
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Sa filed Critical Sanofi Sa
Publication of DK611987D0 publication Critical patent/DK611987D0/en
Publication of DK611987A publication Critical patent/DK611987A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/247-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/26Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group
    • C07D501/34Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group with the 7-amino radical acylated by carboxylic acids containing hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Derivatives corresponding to the general formula: <IMAGE> in which: - R1, R2 and R3 denote H, or R1 and R2 denote H or CH3 and R3 = COOH or else <IMAGE> form a cyclobutyl group and R3 = COOH; - A and B are different and occupy the meta and para positions of the benzene nucleus; one denotes a hydroxyl group and the other is chosen from the groups <IMAGE> and the pharmaceutically acceptable salts and esters of the said derivatives. Use in therapeutics.
DK611987A 1986-11-20 1987-11-20 CEPHALOSPORINE DERIVATIVES AND PROCEDURES FOR PREPARING THEREOF AND PHARMACEUTICAL AGENTS CONTAINING THE DERIVATIVES DK611987A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8616175A FR2607135B1 (en) 1986-11-20 1986-11-20 NOVEL CEPHALOSPORINS DERIVATIVES WITH IMPROVED PHARMACOKINETICS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Publications (2)

Publication Number Publication Date
DK611987D0 true DK611987D0 (en) 1987-11-20
DK611987A DK611987A (en) 1988-05-21

Family

ID=9341024

Family Applications (1)

Application Number Title Priority Date Filing Date
DK611987A DK611987A (en) 1986-11-20 1987-11-20 CEPHALOSPORINE DERIVATIVES AND PROCEDURES FOR PREPARING THEREOF AND PHARMACEUTICAL AGENTS CONTAINING THE DERIVATIVES

Country Status (13)

Country Link
EP (1) EP0269512B1 (en)
JP (1) JPS63141985A (en)
KR (1) KR880006251A (en)
AT (1) ATE67208T1 (en)
DE (1) DE3772936D1 (en)
DK (1) DK611987A (en)
ES (1) ES2038997T3 (en)
FR (1) FR2607135B1 (en)
GR (1) GR3002769T3 (en)
IL (1) IL84539A (en)
NZ (1) NZ222593A (en)
PT (1) PT86164B (en)
ZA (1) ZA878710B (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2621589B1 (en) * 1987-10-08 1990-03-02 Sanofi Sa CEPHALOSPORIN DERIVATIVES WITH IMPROVED PHARMACOKINETICS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
US5189157A (en) * 1987-06-16 1993-02-23 Hoffmann La Roche Inc. Antibacterial cephalosporin compounds

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2546520B1 (en) * 1983-05-27 1985-08-30 Sanofi Sa NOVEL ANTIBIOTIC COMPOUNDS DERIVED FROM CEPHALOSPORINS
FR2570702B1 (en) * 1984-09-27 1987-01-09 Sanofi Sa CEPHALOSPORIN DERIVATIVES, PROCESSES FOR OBTAINING THEM AND THEIR APPLICATION AS ANTIBIOTICS

Also Published As

Publication number Publication date
EP0269512A1 (en) 1988-06-01
NZ222593A (en) 1989-04-26
AU8134887A (en) 1988-05-26
ES2038997T3 (en) 1993-08-16
ZA878710B (en) 1988-05-20
EP0269512B1 (en) 1991-09-11
DK611987A (en) 1988-05-21
PT86164B (en) 1990-11-20
FR2607135B1 (en) 1989-04-28
FR2607135A1 (en) 1988-05-27
DE3772936D1 (en) 1991-10-17
GR3002769T3 (en) 1993-01-25
KR880006251A (en) 1988-07-22
JPS63141985A (en) 1988-06-14
PT86164A (en) 1987-12-01
ATE67208T1 (en) 1991-09-15
IL84539A (en) 1992-12-01
IL84539A0 (en) 1988-04-29
AU597748B2 (en) 1990-06-07

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Legal Events

Date Code Title Description
AHB Application shelved due to non-payment