DK602589A - Quinazolinonderivater - Google Patents

Quinazolinonderivater

Info

Publication number
DK602589A
DK602589A DK602589A DK602589A DK602589A DK 602589 A DK602589 A DK 602589A DK 602589 A DK602589 A DK 602589A DK 602589 A DK602589 A DK 602589A DK 602589 A DK602589 A DK 602589A
Authority
DK
Denmark
Prior art keywords
4alkyl
hydrogen
substituted
6alkyl
hydroxy
Prior art date
Application number
DK602589A
Other languages
Danish (da)
English (en)
Other versions
DK602589D0 (da
Inventor
William John Coates
Lawrence Ivan Kruse
Original Assignee
Smith Kline French Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smith Kline French Lab filed Critical Smith Kline French Lab
Publication of DK602589D0 publication Critical patent/DK602589D0/da
Publication of DK602589A publication Critical patent/DK602589A/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88—Oxygen atoms
    • C07D239/91—Oxygen atoms with aryl or aralkyl radicals attached in position 2 or 3
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
    • C07C237/28—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a non-condensed six-membered aromatic ring of the carbon skeleton
    • C07C237/42—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a non-condensed six-membered aromatic ring of the carbon skeleton having nitrogen atoms of amino groups bound to the carbon skeleton of the acid part, further acylated

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Adhesives Or Adhesive Processes (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK602589A 1988-11-30 1989-11-29 Quinazolinonderivater DK602589A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB888827988A GB8827988D0 (en) 1988-11-30 1988-11-30 Chemical compounds

Publications (2)

Publication Number Publication Date
DK602589D0 DK602589D0 (da) 1989-11-29
DK602589A true DK602589A (da) 1990-05-31

Family

ID=10647738

Family Applications (1)

Application Number Title Priority Date Filing Date
DK602589A DK602589A (da) 1988-11-30 1989-11-29 Quinazolinonderivater

Country Status (11)

Country Link
US (1) US5147875A (de)
EP (1) EP0371731B1 (de)
JP (1) JPH02193983A (de)
AT (1) ATE104665T1 (de)
AU (1) AU630638B2 (de)
CA (1) CA2003690A1 (de)
DE (1) DE68914793T2 (de)
DK (1) DK602589A (de)
GB (1) GB8827988D0 (de)
PT (1) PT92437B (de)
ZA (1) ZA899101B (de)

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Family Cites Families (8)

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Publication number Priority date Publication date Assignee Title
US3169129A (en) * 1963-05-10 1965-02-09 American Cyanamid Co 2-ortho-hydroxy-phenyl-4-(3h)-quinazolinones
USRE26565E (en) * 1966-03-02 1969-04-29 Table iii
US3526627A (en) * 1969-06-05 1970-09-01 American Cyanamid Co Method for preparation of quinazolones
US3651061A (en) * 1970-04-20 1972-03-21 Ernst Reif 2 3-dihydro-2-(1-naphthyl)-4(1h)quinazolinone and the 6-chloroanalog
JPS604831B2 (ja) * 1975-10-20 1985-02-06 中外製薬株式会社 ４（３ｈ）−キナゾリノン誘導体の製法
IT1050750B (it) * 1975-12-05 1981-03-20 Erba Carlo Spa Derivati della 3.4 di idro chinazolina
US4159330A (en) * 1976-11-02 1979-06-26 Carlo Erba S.P.A. 2-Disubstituted phenyl-3,4-dihydro-4-oxo-quinazoline derivatives and process for their preparation
US4431440A (en) * 1981-02-20 1984-02-14 American Cyanamid Company Method to alter or control the development and/or the life cycle of various plant species

Also Published As

Publication number Publication date
EP0371731B1 (de) 1994-04-20
JPH02193983A (ja) 1990-07-31
EP0371731A2 (de) 1990-06-06
AU4541689A (en) 1990-06-07
CA2003690A1 (en) 1990-05-31
DE68914793D1 (de) 1994-05-26
ZA899101B (en) 1990-09-26
GB8827988D0 (en) 1989-01-05
PT92437B (pt) 1995-08-09
AU630638B2 (en) 1992-11-05
US5147875A (en) 1992-09-15
DE68914793T2 (de) 1994-08-18
EP0371731A3 (de) 1991-01-02
DK602589D0 (da) 1989-11-29
PT92437A (pt) 1990-05-31
ATE104665T1 (de) 1994-05-15

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