DK528086A - N-substituerede 3-piperidincarboxylsyrer eller n-substituerede 3-pyridincarboxylsyrer og derivater deraf - Google Patents
N-substituerede 3-piperidincarboxylsyrer eller n-substituerede 3-pyridincarboxylsyrer og derivater derafInfo
- Publication number
- DK528086A DK528086A DK528086A DK528086A DK528086A DK 528086 A DK528086 A DK 528086A DK 528086 A DK528086 A DK 528086A DK 528086 A DK528086 A DK 528086A DK 528086 A DK528086 A DK 528086A
- Authority
- DK
- Denmark
- Prior art keywords
- substituted
- acids
- piperidincarboxyl
- derivatives
- pyridine carboxyl
- Prior art date
Links
- 239000002253 acid Substances 0.000 title 2
- -1 3-PYRIDINE CARBOXYL ACIDS Chemical class 0.000 title 1
- 150000007513 acids Chemical class 0.000 title 1
- 206010015037 epilepsy Diseases 0.000 abstract 2
- XJLSEXAGTJCILF-RXMQYKEDSA-N (R)-nipecotic acid zwitterion Chemical compound OC(=O)[C@@H]1CCCNC1 XJLSEXAGTJCILF-RXMQYKEDSA-N 0.000 abstract 1
- 229940091860 GABA uptake inhibitor Drugs 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 239000002843 gaba uptake inhibitor Substances 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
- C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D211/78—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/60—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US79634585A | 1985-11-08 | 1985-11-08 | |
| US79634585 | 1985-11-08 | ||
| US89730886A | 1986-08-21 | 1986-08-21 | |
| US89730886 | 1986-08-21 |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| DK528086D0 DK528086D0 (da) | 1986-11-05 |
| DK528086A true DK528086A (da) | 1987-05-09 |
| DK165919B DK165919B (da) | 1993-02-08 |
| DK165919C DK165919C (da) | 1993-06-28 |
Family
ID=27121724
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK528086A DK165919C (da) | 1985-11-08 | 1986-11-05 | N-substituerede 3-piperidin- eller 3-pyridincarboxylsyrederivater, fremgangsmaade til fremstilling heraf og farmaceutiske praeparater indeholdende forbindelserne |
Country Status (15)
| Country | Link |
|---|---|
| EP (1) | EP0221572B1 (da) |
| KR (1) | KR900005023B1 (da) |
| CN (1) | CN86107695A (da) |
| AT (1) | ATE67756T1 (da) |
| AU (1) | AU590172B2 (da) |
| CA (1) | CA1270818A (da) |
| DE (1) | DE3681690D1 (da) |
| DK (1) | DK165919C (da) |
| ES (1) | ES2040201T3 (da) |
| FI (1) | FI864246A7 (da) |
| GR (1) | GR3002842T3 (da) |
| NO (1) | NO864443L (da) |
| NZ (1) | NZ218170A (da) |
| PH (1) | PH24683A (da) |
| PT (1) | PT83705B (da) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK704488D0 (da) * | 1988-12-19 | 1988-12-19 | Novo Industri As | Nye n-substituerede azaheterocykliske carboxylsyrer |
| US4910312A (en) * | 1985-11-08 | 1990-03-20 | Warner-Lambert Company | Various N-substituted 3-piperidine carboxylic acids or N-substituted 3-pyridinecarboxylic acids and derivatives thereof |
| DK270488D0 (da) * | 1988-05-18 | 1988-05-18 | Novo Industri As | Hidtil ukendte o-substituerede ketoximer |
| DK588189D0 (da) * | 1989-11-22 | 1989-11-22 | Novo Nordisk As | Nye heterocykliske carboxylsyrer |
| DK93791D0 (da) * | 1991-05-17 | 1991-05-17 | Novo Nordisk As | Nye heterocykliske carboxylsyrer |
| DK74593D0 (da) * | 1993-06-23 | 1993-06-23 | Novo Nordisk As | Novel heterocyclic chemistry |
| IL112223A0 (en) * | 1994-01-04 | 1995-03-30 | Novo Nordisk As | Pharmaceutical compositions for the treatment of neurological inflammatory conditions |
| EP0820442A1 (en) * | 1995-04-07 | 1998-01-28 | Novo Nordisk A/S | Novel heterocyclic compounds |
| WO1996031503A1 (en) * | 1995-04-07 | 1996-10-10 | Novo Nordisk A/S | Novel heterocyclic compounds |
| US5952352A (en) * | 1995-04-07 | 1999-09-14 | Novo Nordisk A/S | Heterocyclic compounds |
| JPH11503131A (ja) * | 1995-04-07 | 1999-03-23 | ノボ ノルディスク アクティーゼルスカブ | 新規の複素環化合物 |
| EP0825984A1 (en) * | 1995-04-07 | 1998-03-04 | Novo Nordisk A/S | Novel method |
| US5962449A (en) | 1995-04-07 | 1999-10-05 | Novo Nordisk A/S | Tricyclic compounds in treating hyperalgesic conditions and NIDDM |
| US6191165B1 (en) | 1996-05-31 | 2001-02-20 | Allelix Neuroscience Inc. | Pharmaceutical for treatment of neurological and neuropsychiatric disorders |
| DK1368336T3 (da) | 2001-02-16 | 2006-10-02 | Allelix Neuroscience Inc | Thiophensubstituerede aminderivater som GlyT-1-inhibitorer |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3929813A (en) * | 1973-12-26 | 1975-12-30 | Interx Research Corp | Novel pro-drug derivatives of pyridinium aldoxime type cholinesterase reactivators and process for preparing same |
| AU552050B2 (en) * | 1981-05-26 | 1986-05-22 | Smithkline Beckman Corporation | N-substituted azeheterocyclic carboxylic acids and their esters |
-
1986
- 1986-10-20 FI FI864246A patent/FI864246A7/fi not_active Application Discontinuation
- 1986-10-30 KR KR1019860009111A patent/KR900005023B1/ko not_active Expired
- 1986-11-03 CA CA000522045A patent/CA1270818A/en not_active Expired - Fee Related
- 1986-11-04 AU AU64812/86A patent/AU590172B2/en not_active Ceased
- 1986-11-05 NZ NZ218170A patent/NZ218170A/xx unknown
- 1986-11-05 DK DK528086A patent/DK165919C/da not_active IP Right Cessation
- 1986-11-05 PH PH34437A patent/PH24683A/en unknown
- 1986-11-07 DE DE8686115478T patent/DE3681690D1/de not_active Expired - Fee Related
- 1986-11-07 PT PT83705A patent/PT83705B/pt not_active IP Right Cessation
- 1986-11-07 AT AT86115478T patent/ATE67756T1/de not_active IP Right Cessation
- 1986-11-07 EP EP86115478A patent/EP0221572B1/en not_active Expired - Lifetime
- 1986-11-07 NO NO864443A patent/NO864443L/no unknown
- 1986-11-07 ES ES198686115478T patent/ES2040201T3/es not_active Expired - Lifetime
- 1986-11-07 CN CN198686107695A patent/CN86107695A/zh active Pending
-
1991
- 1991-10-03 GR GR91401476T patent/GR3002842T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CA1270818A (en) | 1990-06-26 |
| EP0221572B1 (en) | 1991-09-25 |
| DE3681690D1 (de) | 1991-10-31 |
| PT83705A (en) | 1986-12-01 |
| NO864443L (no) | 1987-05-11 |
| NZ218170A (en) | 1990-07-26 |
| EP0221572A2 (en) | 1987-05-13 |
| KR870004955A (ko) | 1987-06-02 |
| FI864246A0 (fi) | 1986-10-20 |
| PT83705B (pt) | 1989-05-12 |
| DK165919B (da) | 1993-02-08 |
| KR900005023B1 (ko) | 1990-07-18 |
| NO864443D0 (no) | 1986-11-07 |
| DK165919C (da) | 1993-06-28 |
| ES2040201T3 (es) | 1993-10-16 |
| AU6481286A (en) | 1987-05-14 |
| AU590172B2 (en) | 1989-10-26 |
| ATE67756T1 (de) | 1991-10-15 |
| EP0221572A3 (en) | 1987-07-29 |
| FI864246A7 (fi) | 1987-05-09 |
| CN86107695A (zh) | 1987-05-13 |
| PH24683A (en) | 1990-09-07 |
| DK528086D0 (da) | 1986-11-05 |
| GR3002842T3 (en) | 1993-01-25 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PBP | Patent lapsed |