DK508985A - Anvendelse af 4-((alfa-metyl)-2,3-dimetylbenzyl)-imidazol til fremstilling af veterinaere praeparater - Google Patents

Anvendelse af 4-((alfa-metyl)-2,3-dimetylbenzyl)-imidazol til fremstilling af veterinaere praeparater Download PDF

Info

Publication number
DK508985A
DK508985A DK508985A DK508985A DK508985A DK 508985 A DK508985 A DK 508985A DK 508985 A DK508985 A DK 508985A DK 508985 A DK508985 A DK 508985A DK 508985 A DK508985 A DK 508985A
Authority
DK
Denmark
Prior art keywords
imidazole
methyl
alfa
preparation
dimethyl benzyl
Prior art date
Application number
DK508985A
Other languages
English (en)
Other versions
DK163960C (da
DK508985D0 (da
DK163960B (da
Inventor
R E Virtanen
A J Karjalainen
K O A Kurkela
A T Vaehae-Vahe
O M Vainio-Kevinen
Original Assignee
Farmos Oy
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farmos Oy filed Critical Farmos Oy
Publication of DK508985D0 publication Critical patent/DK508985D0/da
Publication of DK508985A publication Critical patent/DK508985A/da
Publication of DK163960B publication Critical patent/DK163960B/da
Application granted granted Critical
Publication of DK163960C publication Critical patent/DK163960C/da

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
  • Photoreceptors In Electrophotography (AREA)
  • Stringed Musical Instruments (AREA)
DK508985A 1984-12-04 1985-11-05 Anvendelse af 4-((alfa-metyl)-2,3-dimetylbenzyl)-imidazol til fremstilling af veterinaere praeparater DK163960C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FI844786A FI844786A0 (fi) 1984-12-04 1984-12-04 Terapeutiskt utnyttjbar foerening.
FI844786 1984-12-04

Publications (4)

Publication Number Publication Date
DK508985D0 DK508985D0 (da) 1985-11-05
DK508985A true DK508985A (da) 1986-06-05
DK163960B DK163960B (da) 1992-04-27
DK163960C DK163960C (da) 1992-09-21

Family

ID=8520010

Family Applications (1)

Application Number Title Priority Date Filing Date
DK508985A DK163960C (da) 1984-12-04 1985-11-05 Anvendelse af 4-((alfa-metyl)-2,3-dimetylbenzyl)-imidazol til fremstilling af veterinaere praeparater

Country Status (11)

Country Link
US (1) US4670455A (da)
EP (1) EP0187471B1 (da)
JP (1) JPS61134314A (da)
AT (1) ATE65694T1 (da)
AU (1) AU572364B2 (da)
DE (1) DE3583670D1 (da)
DK (1) DK163960C (da)
FI (1) FI844786A0 (da)
IE (1) IE58269B1 (da)
NZ (1) NZ213604A (da)
ZA (1) ZA858416B (da)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI864570A0 (fi) * 1986-11-11 1986-11-11 Farmos Oy Terapeutiskt anvaendbar foerening.
GB2206880B (en) 1987-07-16 1991-04-24 Farmos Oy Optical isomers of an imidazole derivative
GB2215206B (en) 1988-02-29 1991-07-03 Farmos Oy 4-substituted imidazole derivatives useful in perioperative care
US5344840A (en) * 1988-02-29 1994-09-06 Orion-Yhtyma Oy 4-substituted imidazole derivatives useful in perioperative care
US5124157A (en) * 1989-08-18 1992-06-23 Cygnus Therapeutic Systems Method and device for administering dexmedetomidine transdermally
AR015744A1 (es) * 1998-04-01 2001-05-16 Orion Corp Uso de dexmedetomidina para sedacion en terapia intensiva
FI20041425A0 (fi) * 2004-11-05 2004-11-05 Orion Corp Transmukosaalinen veterinäärinen koostumus
US7795263B2 (en) * 2008-07-08 2010-09-14 Wildlife Laboratories, Inc. Pharmaceutical combination for and method of anesthetizing and immobilizing non-domesticated mammals
EP2370136A4 (en) * 2008-12-01 2015-12-30 Map Pharmaceuticals Inc INHALATIVE RELEASE PROCEDURES AND DEVICES
WO2010074753A1 (en) 2008-12-23 2010-07-01 Map Pharmaceuticals, Inc. Inhalation devices and related methods for administration of sedative hypnotic compounds
US20130096170A1 (en) 2011-10-14 2013-04-18 Hospira, Inc. Methods of treating pediatric patients using dexmedetomidine
WO2013069025A1 (en) 2011-11-11 2013-05-16 Neon Laboratories Ltd. "process for the preparation of dexmedetomidine"
US8242158B1 (en) 2012-01-04 2012-08-14 Hospira, Inc. Dexmedetomidine premix formulation
JP6188933B2 (ja) 2013-10-07 2017-08-30 テイコク ファーマ ユーエスエー インコーポレーテッド 非鎮静量のデクスメデトミジンの経皮送達用方法及び組成物
TWI645866B (zh) 2013-10-07 2019-01-01 美商帝國製藥美國股份有限公司 右美托咪啶經皮輸送裝置及使用其之方法
US20150098997A1 (en) 2013-10-07 2015-04-09 Teikoku Pharma Usa, Inc. Methods and Compositions for Treating Attention Deficit Hyperactivity Disorder, Anxiety and Insomnia Using Dexmedetomidine Transdermal Compositions
US9717796B1 (en) 2016-04-20 2017-08-01 Slypharma, Llc Heat sterilizeable, premixed, ready to use dexmedetomidine solution packaged in a flexible plastic container
RU2723761C1 (ru) 2016-10-31 2020-06-17 ТЕЙКОКУ ФАРМА ЮЭсЭй, ИНК. Способы устранения боли с использованием устройств для трансдермальной доставки дексмедетомидина
CN110337290A (zh) 2016-12-31 2019-10-15 比奥克斯塞尔医疗股份有限公司 舌下右旋美托咪啶用于治疗激越的用途
EP4523752A3 (en) 2018-06-27 2025-05-14 BioXcel Therapeutics, Inc. Film formulations containing dexmedetomidine and methods of producing them
US11160791B2 (en) 2018-11-01 2021-11-02 Medefil, Inc. Dexmedetomidine injection premix formulation in ready to use (RTU) bags
JP7739256B2 (ja) 2019-07-19 2025-09-16 バイオエクセル セラピューティクス,インコーポレイテッド 鎮静作用のないデクスメデトミジン治療レジメン
US11806334B1 (en) 2023-01-12 2023-11-07 Bioxcel Therapeutics, Inc. Non-sedating dexmedetomidine treatment regimens

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2092569B (en) * 1981-02-05 1984-09-19 Farmos Oy Substituted imidazole derivatives and their preparation and use
GB2096987B (en) * 1981-04-22 1984-04-04 Farmos Oy Substituted imidazole and imidazole derivatives and their preparation and use
GB2101114B (en) * 1981-07-10 1985-05-22 Farmos Group Ltd Substituted imidazole derivatives and their preparation and use
EP0106060B1 (en) * 1982-08-14 1988-09-28 The Wellcome Foundation Limited Imidazole derivatives and salts thereof, their synthesis, and pharmaceutical formulations

Also Published As

Publication number Publication date
EP0187471B1 (en) 1991-07-31
DK163960C (da) 1992-09-21
NZ213604A (en) 1988-09-29
IE58269B1 (en) 1993-08-25
IE853024L (en) 1986-06-04
DK508985D0 (da) 1985-11-05
ZA858416B (en) 1986-07-30
AU572364B2 (en) 1988-05-05
AU4997185A (en) 1986-06-12
EP0187471A2 (en) 1986-07-16
JPH0465050B2 (da) 1992-10-16
DE3583670D1 (de) 1991-09-05
FI844786A0 (fi) 1984-12-04
JPS61134314A (ja) 1986-06-21
US4670455A (en) 1987-06-02
DK163960B (da) 1992-04-27
EP0187471A3 (en) 1988-09-14
ATE65694T1 (de) 1991-08-15

Similar Documents

Publication Publication Date Title
DK508985D0 (da) Anvendelse af 4-((alfa-metyl)-2,3-dimetylbenzyl)-imidazol til fremstilling af veterinaere praeparater
TR199801360T2 (xx) Yeni ikameli imidazol bile�imleri.
MX9301783A (es) Derivados de 1-[2-arilsulfonilamino)-etil-1-oxo]-piperidina, su preparacion y su aplicacion en terapeutica.
DK46489A (da) Anvendelse af 4-(1-(2,3-dimetylfenyl)-aetyl)-1h-imidazol til fremstilling af laegemidler til perioperativ anvendelse
DE69724246D1 (de) Neue substituierte imidazolverbindungen
IE790107L (en) Substituted propanolamine and morpholine derivatives
BR9912975A (pt) Composto e composições para liberação de agentes ativos, método para sua obtenção e seu uso
EA199900953A1 (ru) ЗАМЕЩЕННЫЕ ПИРАЗОЛЫ, КАК ИНГИБИТОРЫ p38 КИНАЗЫ
FI882882A7 (fi) Menetelmä terapeuttisesti aktiivisten (substituoitu aralkyyli)triatsoli-, -imidatsoli-, -pyridiini- ja -pyrimidiiniyhdisteiden valmistamiseksi
IS1565B (is) Aðferð við framleiðslu á N1-súbstitúeruðum bensimidasólafleiðum til að nota við lækningar
DK76582A (da) Antimycotiske midler
ATE40822T1 (de) Aromatase-hemmende 1,2,3-triazol-1-yl-, tetrazol- 1-yl- und tetrazol-2-yl-verbindungen.
DK686088D0 (da) 2-phenyl-3-(piperazin-1-yl)-1-(1h-1,2,4-triazol-1-yl) propan-2-ol-forbindelser
ES2074178T3 (es) Preparados de antimicoticos externos de imidazol.
DK157134C (da) Analogifremgangsmaade til fremstilling af 1-(5-chlorpyrid-2-yl)-1-(2,4-dihalogenphenyl)-2-(1,2,4-triazol-1-yl)-ethanol-forbindelser eller deres farmaceutisk acceptable syreadditionssalte
SE430117B (sv) Fungicid beredning innehallande 1-(beta-(allyloxi)-2,4-diklorofenetyl) imidazol och en pyrimidinmetanol
ES535341A0 (es) Procedimiento para la obtencion de 1-(2,4-diclorofenil)-2-(1h-imidazol-1-il)-1-(2,4-diclorobenciloximino)
DE3874361D1 (de) Als analgetika verwendbare 1-((4-morpholinyl)alkyl)-1h-indole und deren herstellung.
IT8222035A0 (it) Procedimento perfezionato per lapreparazione della 2,4-diammino-5-(3',4',5'-trimetossi benzil)-pirimidina.
ES551110A0 (es) Procedimiento para la obtencion de derivados de 1-(2,4-diclorofenil)-2-(1-imidazolil)etanol
ECSP971995A (es) Nuevos imidazoles sustituidos con cicloalquilo
ES533613A0 (es) Procedimiento para la obtencion del 1-(4-fluorofenilmetil)-2-(1-(4-metoxifenetil)-4-piperidinil-amino-bencimidazol
IT1111152B (it) Processo per la preparazione dell'1-(2,4iclorofenil)-1-(4-clorofenil)metosso)-2-(imidazolil-1-etano
ES537071A0 (es) Procedimiento de obtencion del 1-(4-(1, 1-dimetiletil)fenil)-4-(4-hidroxidifenilmetil)-1-piperidin)butanol
YU46750B (sh) Derivati laktama i postupci za njihovo dobijanje

Legal Events

Date Code Title Description
PUP Patent expired