ATE37714T1 - Imidazolyl-, triazolyl- und tetrazolylverbindungen. - Google Patents
Imidazolyl-, triazolyl- und tetrazolylverbindungen.Info
- Publication number
- ATE37714T1 ATE37714T1 AT85304235T AT85304235T ATE37714T1 AT E37714 T1 ATE37714 T1 AT E37714T1 AT 85304235 T AT85304235 T AT 85304235T AT 85304235 T AT85304235 T AT 85304235T AT E37714 T1 ATE37714 T1 AT E37714T1
- Authority
- AT
- Austria
- Prior art keywords
- triazolyl
- imidazolyl
- tetrazolyl compounds
- tetrazolyl
- compounds
- Prior art date
Links
- -1 IMIDAZOLYL Chemical class 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
- 102000014654 Aromatase Human genes 0.000 abstract 1
- 108010078554 Aromatase Proteins 0.000 abstract 1
- 230000001419 dependent effect Effects 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 229940011871 estrogen Drugs 0.000 abstract 1
- 239000000262 estrogen Substances 0.000 abstract 1
- 125000002883 imidazolyl group Chemical group 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000003831 tetrazolyl group Chemical group 0.000 abstract 1
- 125000001425 triazolyl group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/621,581 US4659730A (en) | 1984-06-18 | 1984-06-18 | Aromatase inhibiting imidazole derivatives |
| EP85304235A EP0165780B1 (de) | 1984-06-18 | 1985-06-14 | Imidazolyl-, Triazolyl- und Tetrazolyl-Verbindungen |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE37714T1 true ATE37714T1 (de) | 1988-10-15 |
Family
ID=24490759
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT85304235T ATE37714T1 (de) | 1984-06-18 | 1985-06-14 | Imidazolyl-, triazolyl- und tetrazolylverbindungen. |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US4659730A (de) |
| EP (1) | EP0165780B1 (de) |
| JP (1) | JPH0662581B2 (de) |
| AT (1) | ATE37714T1 (de) |
| CA (1) | CA1256112A (de) |
| DE (1) | DE3565403D1 (de) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NZ219311A (en) * | 1986-02-27 | 1989-04-26 | Janssen Pharmaceutica Nv | Imidazoles and herbicidal compositions |
| US4937250A (en) * | 1988-03-07 | 1990-06-26 | Ciba-Geigy Corporation | Alpha-heterocycle substituted tolunitriles |
| US4978672A (en) * | 1986-03-07 | 1990-12-18 | Ciba-Geigy Corporation | Alpha-heterocyclc substituted tolunitriles |
| GB8705174D0 (en) * | 1987-03-05 | 1987-04-08 | Ici Plc | Heterocyclic compounds |
| NZ224714A (en) * | 1987-06-01 | 1990-03-27 | Janssen Pharmaceutica Nv | Substituted benzotriazole derivatives and pharmaceutical compositions |
| EP0457716A1 (de) * | 1990-04-20 | 1991-11-21 | Ciba-Geigy Ag | Naphthalinderivate |
| TW224461B (de) * | 1990-09-18 | 1994-06-01 | Ciba Geigy Ag | |
| GB9520150D0 (en) * | 1995-10-03 | 1995-12-06 | Orion Yhtymae Oy | New imidazole derivatives |
| GB9900078D0 (en) * | 1999-01-05 | 1999-02-24 | Zeneca Ltd | Chemical compounds |
| CN101605777A (zh) * | 2006-12-18 | 2009-12-16 | 诺瓦提斯公司 | 作为醛固酮合酶抑制剂的咪唑类化合物 |
| WO2016031928A1 (ja) * | 2014-08-29 | 2016-03-03 | 東京応化工業株式会社 | イミダゾール化合物、金属表面処理液、金属の表面処理方法、及び積層体の製造方法 |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3636002A (en) * | 1969-12-15 | 1972-01-18 | Janssen Pharmaceutica Nv | 1-(2-halobenzyloxy-1-indanyl)-imidazoles |
| US4115578A (en) * | 1975-12-18 | 1978-09-19 | Rohm And Haas Company | 1-Substituted aralkyl imidazoles |
| US4284641A (en) * | 1977-08-26 | 1981-08-18 | Burroughs Wellcome Co. | Pharmaceutically active imidazole derivatives |
| DE2862340D1 (en) * | 1978-02-01 | 1983-11-24 | Wellcome Found | Imidazole derivatives and salts thereof, their synthesis, and pharmaceutical formulations thereof |
| US4235893A (en) * | 1978-05-08 | 1980-11-25 | Brodie Angela M | Ester derivatives of 4-hydroxy-4-androstene-3,17-dione and a method for inhibiting estrogen biosynthesis |
| US4144347A (en) * | 1978-06-26 | 1979-03-13 | Riker Laboratories, Inc. | 3-(N-Imidazolyl)-2-nitrobenzofurans |
| DE2845254A1 (de) * | 1978-10-18 | 1980-05-08 | Basf Ag | Gamma -azolylverbindungen |
| JPS55129284A (en) * | 1979-03-27 | 1980-10-06 | Shionogi & Co Ltd | 3-(1-imipazolyl)indolin-2-one |
| IL62122A0 (en) * | 1980-03-04 | 1981-03-31 | Erba Farmitalia | N-imidazolyl derivatives of 1-chroman,their preparation and pharmaceutical compositions containing them |
| US4352808A (en) * | 1980-12-12 | 1982-10-05 | Schering Corporation | 3-Aralkyloxy-2,3-dihydro-2-(imidazolylmethyl)benzo(b)thiophenes and related derivatives, their use as antimicrobials and pharmaceutical formulations useful therefore |
| US4468404A (en) * | 1980-12-12 | 1984-08-28 | Schering Corporation | 3-Aralkyloxy-2,3-dihydro-2-(triazolymethyl)benzo(b)thiophenes |
| DE3369131D1 (en) * | 1982-04-22 | 1987-02-19 | Ici Plc | Antifungal azolyl phenyl substituted alicyclic alcohols |
| ES523609A0 (es) * | 1982-07-05 | 1985-03-01 | Erba Farmitalia | Procedimiento para preparar derivados n-imidazolilicos de compuestos biciclicos. |
| GB2122997B (en) * | 1982-07-05 | 1985-08-14 | Erba Farmitalia | Imidazoles |
-
1984
- 1984-06-18 US US06/621,581 patent/US4659730A/en not_active Expired - Fee Related
-
1985
- 1985-06-11 CA CA000483673A patent/CA1256112A/en not_active Expired
- 1985-06-14 AT AT85304235T patent/ATE37714T1/de not_active IP Right Cessation
- 1985-06-14 DE DE8585304235T patent/DE3565403D1/de not_active Expired
- 1985-06-14 EP EP85304235A patent/EP0165780B1/de not_active Expired
- 1985-06-18 JP JP60135223A patent/JPH0662581B2/ja not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| US4659730A (en) | 1987-04-21 |
| JPS6117566A (ja) | 1986-01-25 |
| CA1256112A (en) | 1989-06-20 |
| DE3565403D1 (en) | 1988-11-10 |
| EP0165780A1 (de) | 1985-12-27 |
| EP0165780B1 (de) | 1988-10-05 |
| JPH0662581B2 (ja) | 1994-08-17 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification | ||
| REN | Ceased due to non-payment of the annual fee |