DK425487A - Pharmaceutisk aktive derivater af glutamin- og asparginsyre - Google Patents
Pharmaceutisk aktive derivater af glutamin- og asparginsyreInfo
- Publication number
- DK425487A DK425487A DK425487A DK425487A DK425487A DK 425487 A DK425487 A DK 425487A DK 425487 A DK425487 A DK 425487A DK 425487 A DK425487 A DK 425487A DK 425487 A DK425487 A DK 425487A
- Authority
- DK
- Denmark
- Prior art keywords
- group
- glutaminic
- carbon atoms
- pharmaceutical active
- active derivatives
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
- C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C233/30—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by doubly-bound oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
- C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C233/45—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT6806285 | 1985-12-17 | ||
IT8568062A IT1215169B (it) | 1985-12-17 | 1985-12-17 | Derivati alchil ossigenati degli acidi glutammico ed aspartico ad attivita antagonista su polipeptidi bioattivi e procedimento per la loro preparazione |
EP8600724 | 1986-12-08 | ||
PCT/EP1986/000724 WO1987003869A2 (en) | 1985-12-17 | 1986-12-08 | Pharmaceutically active derivatives of glutamic and aspartic acids |
Publications (3)
Publication Number | Publication Date |
---|---|
DK425487D0 DK425487D0 (da) | 1987-08-14 |
DK425487A true DK425487A (da) | 1987-08-14 |
DK169666B1 DK169666B1 (da) | 1995-01-09 |
Family
ID=11307569
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK425487A DK169666B1 (da) | 1985-12-17 | 1987-08-14 | Farmaceutisk aktive derivater af D,L-glutamin- og D,L-asparaginsyre, fremgangsmåde til deres fremstilling samt farmaceutisk sammensætning og sammensætning til anvendelse ved husdyrbrug indeholdende sådanne derivater |
Country Status (13)
Country | Link |
---|---|
US (1) | US4769389A (da) |
EP (1) | EP0286643B1 (da) |
JP (1) | JPS62181246A (da) |
AU (1) | AU595858B2 (da) |
CA (1) | CA1269110A (da) |
DK (1) | DK169666B1 (da) |
ES (1) | ES2081777A6 (da) |
GR (1) | GR862921B (da) |
IE (1) | IE59534B1 (da) |
IT (1) | IT1215169B (da) |
PT (1) | PT83952B (da) |
WO (1) | WO1987003869A2 (da) |
ZA (1) | ZA869460B (da) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4880938A (en) * | 1986-06-16 | 1989-11-14 | Merck & Co., Inc. | Amino acid analogs |
US5089638A (en) * | 1986-06-16 | 1992-02-18 | Merck & Co., Inc. | Amino acid analogs as CCK-antagonists |
IT1196849B (it) * | 1986-12-16 | 1988-11-25 | Rotta Research Lab | Nuovi derivati degli acidi 5 pentilammino 5 oxo pentaoico e 4 pentilammino 4 oxo butanoico ad attivita antagonista della colecistochinina e procedimento per la loro preparazione |
IT1217123B (it) * | 1987-02-05 | 1990-03-14 | Rotta Research Lab | Derivati otticamente attivi dell acido 5 pentilammino 5 oxo pentanoico r ad attivita antagonista della colecistochinina e procedimento per la loro preparazione |
US5105007A (en) * | 1987-10-19 | 1992-04-14 | Abbott Laboratories | Phenylacetylglutamine (PAG) analytical test |
EP0411668B2 (en) * | 1989-08-04 | 1998-11-11 | MERCK SHARP & DOHME LTD. | Central cholecystokinin antagonists for treatment of psychiatric disorders |
US5066828A (en) * | 1990-04-12 | 1991-11-19 | Merrell Dow Pharmaceuticals Inc. | Difluoroglutamic acid conjugates with folates and anti-folates for the treatment of neoplastic diseases |
JPH07507993A (ja) * | 1991-12-20 | 1995-09-07 | メルク シヤープ エンド ドーム リミテツド | 医薬活性を有する中枢神経系コレシストキニンアンタゴニスト |
GB9200420D0 (en) * | 1992-01-09 | 1992-02-26 | James Black Foundation The Lim | Amino acid derivatives |
US5716958A (en) | 1994-10-27 | 1998-02-10 | Tobishi Pharmaceutical Co., Ltd. | Amino acid derivative having anti-CCK activity |
CA2614930A1 (en) * | 2005-07-11 | 2007-01-18 | Wyeth | Glutamate aggrecanase inhibitors |
US7863330B2 (en) | 2006-06-14 | 2011-01-04 | Rottapharm S.P.A. | Deloxiglumide and proton pump inhibitor combination in the treatment of gastrointestinal disorders |
CN108912007B (zh) * | 2018-06-20 | 2021-02-26 | 中国农业科学院兰州畜牧与兽药研究所 | 一种右氯谷胺的制备方法 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1108819A (en) * | 1964-07-31 | 1968-04-03 | Rotta Research Lab | Derivatives of 2-acylaminobicarboxylic acids and method for preparing same |
US3465081A (en) * | 1966-05-13 | 1969-09-02 | Thompson Chem Co Hayward | Method of controlling pestiferous organisms |
AT293368B (de) * | 1969-10-13 | 1971-10-11 | Rotta Research Lab | Verfahren zur Herstellung von N-Benzoyl-L-(D- oder DL)-glutaminsäure-l-amiden |
US3803223A (en) * | 1970-07-20 | 1974-04-09 | Searle & Co | 3-amino-n-substituted succinamic acids and intermediates thereto |
US4243678A (en) * | 1977-12-30 | 1981-01-06 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Acylhydrocarbylaminoalkanoic acids, compositions and uses |
IE57892B1 (en) * | 1984-06-25 | 1993-05-05 | Rotta Research Lab | Glutamic and aspartic acid derivatives |
GB8704671D0 (en) * | 1987-02-27 | 1987-04-01 | Shell Int Research | Glycine compounds |
-
1985
- 1985-12-17 IT IT8568062A patent/IT1215169B/it active
-
1986
- 1986-12-08 EP EP87901263A patent/EP0286643B1/en not_active Expired - Lifetime
- 1986-12-08 WO PCT/EP1986/000724 patent/WO1987003869A2/en active IP Right Grant
- 1986-12-08 AU AU69497/87A patent/AU595858B2/en not_active Ceased
- 1986-12-10 IE IE323386A patent/IE59534B1/en not_active IP Right Cessation
- 1986-12-15 CA CA000525358A patent/CA1269110A/en not_active Expired - Fee Related
- 1986-12-16 JP JP61301132A patent/JPS62181246A/ja active Granted
- 1986-12-16 ES ES08603651A patent/ES2081777A6/es not_active Expired - Fee Related
- 1986-12-17 US US06/942,751 patent/US4769389A/en not_active Expired - Lifetime
- 1986-12-17 GR GR862921A patent/GR862921B/el unknown
- 1986-12-17 PT PT83952A patent/PT83952B/pt not_active IP Right Cessation
- 1986-12-17 ZA ZA869460A patent/ZA869460B/xx unknown
-
1987
- 1987-08-14 DK DK425487A patent/DK169666B1/da not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
AU6949787A (en) | 1987-07-15 |
PT83952B (pt) | 1989-06-30 |
GR862921B (en) | 1987-04-27 |
ES2081777A6 (es) | 1996-03-01 |
DK169666B1 (da) | 1995-01-09 |
WO1987003869A3 (en) | 1987-08-13 |
IT1215169B (it) | 1990-01-31 |
DK425487D0 (da) | 1987-08-14 |
JPH0543698B2 (da) | 1993-07-02 |
IE863233L (en) | 1987-06-17 |
EP0286643A1 (en) | 1988-10-19 |
ZA869460B (en) | 1987-08-26 |
CA1269110A (en) | 1990-05-15 |
IE59534B1 (en) | 1994-03-09 |
IT8568062A0 (it) | 1985-12-17 |
AU595858B2 (en) | 1990-04-12 |
WO1987003869A2 (en) | 1987-07-02 |
EP0286643B1 (en) | 1991-05-15 |
JPS62181246A (ja) | 1987-08-08 |
PT83952A (en) | 1987-01-01 |
US4769389A (en) | 1988-09-06 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B1 | Patent granted (law 1993) | ||
PBP | Patent lapsed |
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