DK3636640T3 - Krystal af heterocyclidenacetamidderivat - Google Patents

Krystal af heterocyclidenacetamidderivat Download PDF

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Publication number
DK3636640T3
DK3636640T3 DK18810263.6T DK18810263T DK3636640T3 DK 3636640 T3 DK3636640 T3 DK 3636640T3 DK 18810263 T DK18810263 T DK 18810263T DK 3636640 T3 DK3636640 T3 DK 3636640T3
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Prior art keywords
heterocyclidenaaceta
crystal
mid
derivative
mid derivative
Prior art date
Application number
DK18810263.6T
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English (en)
Inventor
Tsutomu Satoh
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Mochida Pharm Co Ltd
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Publication of DK3636640T3 publication Critical patent/DK3636640T3/da

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/58Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/02Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
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    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
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    • AHUMAN NECESSITIES
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    • A61P11/02Nasal agents, e.g. decongestants
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    • A61P11/14Antitussive agents
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    • A61P13/00Drugs for disorders of the urinary system
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    • AHUMAN NECESSITIES
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    • A61P17/02Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
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    • A61P27/02Ophthalmic agents
    • A61P27/14Decongestants or antiallergics
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
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    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
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    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
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    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
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    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
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    • A61P7/10Antioedematous agents; Diuretics
    • AHUMAN NECESSITIES
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    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Pulmonology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Epidemiology (AREA)
  • Otolaryngology (AREA)
  • Hospice & Palliative Care (AREA)
  • Obesity (AREA)
  • Psychiatry (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
DK18810263.6T 2017-05-31 2018-05-30 Krystal af heterocyclidenacetamidderivat DK3636640T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201762512775P 2017-05-31 2017-05-31
JP2017108017A JP6230743B1 (ja) 2017-05-31 2017-05-31 ヘテロシクリデンアセトアミド誘導体の結晶
PCT/JP2018/020634 WO2018221543A1 (ja) 2017-05-31 2018-05-30 ヘテロシクリデンアセトアミド誘導体の結晶

Publications (1)

Publication Number Publication Date
DK3636640T3 true DK3636640T3 (da) 2022-12-19

Family

ID=60321089

Family Applications (1)

Application Number Title Priority Date Filing Date
DK18810263.6T DK3636640T3 (da) 2017-05-31 2018-05-30 Krystal af heterocyclidenacetamidderivat

Country Status (13)

Country Link
US (1) US10208010B2 (da)
EP (1) EP3636640B1 (da)
JP (1) JP6230743B1 (da)
KR (1) KR102576964B1 (da)
CN (1) CN110831930B (da)
CA (1) CA3059483A1 (da)
DK (1) DK3636640T3 (da)
ES (1) ES2934508T3 (da)
HU (1) HUE061363T2 (da)
MX (1) MX2019014216A (da)
PL (1) PL3636640T3 (da)
PT (1) PT3636640T (da)
WO (1) WO2018221543A1 (da)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP6230743B1 (ja) 2017-05-31 2017-11-15 持田製薬株式会社 ヘテロシクリデンアセトアミド誘導体の結晶
US20220204475A1 (en) * 2019-04-30 2022-06-30 Beijing Tide Pharmaceutical Co., Ltd. Solid form of diaminopyrimidine compound or hydrate thereof, preparation method therefor, and application thereof
EP4043014A4 (en) * 2019-10-04 2023-10-11 Senju Pharmaceutical Co., Ltd. PHARMACEUTICAL MEDICINAL PRODUCT CONTAINING HETEROCYCLIDE ACETAMIDE DERIVATIVE
WO2022210784A1 (ja) 2021-03-30 2022-10-06 千寿製薬株式会社 ヘテロシクリデンアセトアミド誘導体含有懸濁液
WO2024071348A1 (ja) * 2022-09-29 2024-04-04 千寿製薬株式会社 滅菌処理したヘテロシクリデンアセトアミド誘導体含有懸濁液

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR101136183B1 (ko) * 2005-07-22 2012-04-17 모찌다 세이야쿠 가부시끼가이샤 신규 헤테로시클리덴 아세트아미드 유도체
ZA200800959B (en) * 2005-07-22 2009-10-28 Mochida Pharmaceutical Company Novel heterocyclidene acetamide derivative
JP2011201777A (ja) * 2008-07-23 2011-10-13 Mochida Pharmaceut Co Ltd 光学活性なヘテロシクリデン−n−アリールアセトアミド誘導体
JP2017108017A (ja) 2015-12-10 2017-06-15 キヤノン株式会社 レーザ装置、及びこれを用いた計測装置
JP6230743B1 (ja) 2017-05-31 2017-11-15 持田製薬株式会社 ヘテロシクリデンアセトアミド誘導体の結晶

Also Published As

Publication number Publication date
JP6230743B1 (ja) 2017-11-15
CN110831930B (zh) 2023-04-28
US20180346436A1 (en) 2018-12-06
EP3636640A4 (en) 2021-03-03
EP3636640A1 (en) 2020-04-15
CA3059483A1 (en) 2018-12-06
US10208010B2 (en) 2019-02-19
PT3636640T (pt) 2022-12-26
WO2018221543A1 (ja) 2018-12-06
RU2019137598A3 (da) 2021-07-07
KR102576964B1 (ko) 2023-09-11
ES2934508T3 (es) 2023-02-22
CN110831930A (zh) 2020-02-21
EP3636640B1 (en) 2022-11-30
KR20200011943A (ko) 2020-02-04
MX2019014216A (es) 2020-01-23
HUE061363T2 (hu) 2023-06-28
JP2018203648A (ja) 2018-12-27
RU2019137598A (ru) 2021-06-30
PL3636640T3 (pl) 2023-02-27

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