DK3490988T3 - Ny forbindelse og fremgangsmåde - Google Patents

Ny forbindelse og fremgangsmåde Download PDF

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Publication number
DK3490988T3
DK3490988T3 DK17748880T DK17748880T DK3490988T3 DK 3490988 T3 DK3490988 T3 DK 3490988T3 DK 17748880 T DK17748880 T DK 17748880T DK 17748880 T DK17748880 T DK 17748880T DK 3490988 T3 DK3490988 T3 DK 3490988T3
Authority
DK
Denmark
Prior art keywords
approach
new connection
new
connection
Prior art date
Application number
DK17748880T
Other languages
English (en)
Inventor
Peter Lionel Spargo
Original Assignee
Verona Pharma Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Verona Pharma Plc filed Critical Verona Pharma Plc
Application granted granted Critical
Publication of DK3490988T3 publication Critical patent/DK3490988T3/da

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
DK17748880T 2016-07-28 2017-07-27 Ny forbindelse og fremgangsmåde DK3490988T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB1613054.4A GB201613054D0 (en) 2016-07-28 2016-07-28 New compound and process
PCT/GB2017/052190 WO2018020249A1 (en) 2016-07-28 2017-07-27 New compound and process

Publications (1)

Publication Number Publication Date
DK3490988T3 true DK3490988T3 (da) 2019-10-28

Family

ID=56936838

Family Applications (1)

Application Number Title Priority Date Filing Date
DK17748880T DK3490988T3 (da) 2016-07-28 2017-07-27 Ny forbindelse og fremgangsmåde

Country Status (18)

Country Link
US (1) US10710998B2 (da)
EP (1) EP3490988B1 (da)
JP (1) JP6985367B2 (da)
KR (1) KR102396059B1 (da)
CN (1) CN109641891B (da)
CY (1) CY1122138T1 (da)
DK (1) DK3490988T3 (da)
ES (1) ES2751948T3 (da)
GB (1) GB201613054D0 (da)
HR (1) HRP20192109T1 (da)
HU (1) HUE046509T2 (da)
LT (1) LT3490988T (da)
PL (1) PL3490988T3 (da)
PT (1) PT3490988T (da)
RS (1) RS59566B1 (da)
SI (1) SI3490988T1 (da)
TW (1) TWI739871B (da)
WO (1) WO2018020249A1 (da)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT3231444T (pt) 2014-05-12 2020-03-05 Verona Pharma Plc Novo tratamento
GB201502260D0 (en) 2015-02-11 2015-04-01 Verona Pharma Plc Salt of Pyrimido[6,1-A]Isoquinolin-4-one compound
WO2022228544A1 (zh) 2021-04-29 2022-11-03 苏州盛迪亚生物医药有限公司 异喹啉酮类化合物及其用途
WO2023109802A1 (zh) * 2021-12-14 2023-06-22 海思科医药集团股份有限公司 三环稠杂环类pde3/4双重抑制及其用途

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ185900A (en) 1976-12-10 1981-04-24 Hoechst Ag Pyrimido (6,1-a) isoquinolin-4-ones medicaments intermediate isoquinolines
FI64370C (fi) 1977-05-05 1983-11-10 Hoechst Ag Foerfarande foer framstaellning av terapeutiskt anvaendbara pyimido-(6,1-a)isokinolin-2-imino-4-onderivat
DE2847693A1 (de) 1978-11-03 1980-05-22 Hoechst Ag Verfahren zur herstellung von pyrimido-(6,1-a)-isochinolin-2-onen
DE3135831A1 (de) 1981-09-10 1983-04-28 Hoechst Ag, 6230 Frankfurt 9,10-substituierte 2-mesitylimino-3-alkyl-3,4,6,7-tetrahydro-2h-pyrimido(6,1-a)isochinolin-4-one, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
ZW6284A1 (en) 1983-05-05 1985-10-30 Hoffmann La Roche Novel pyrimidone derivatives
JP4685243B2 (ja) 1999-03-31 2011-05-18 ベローナ・ファーマ・ピーエルシー ピリミド[6,1−a]イソキノリン−4−オン誘導体
SI2603509T1 (sl) 2010-08-09 2014-10-30 Verona Pharma Plc Kristalinična oblika spojine PIRIMIDIO(6,1-A) IZOKINOLIN-4-ENA
CA2902403C (en) 2013-03-15 2021-06-01 Verona Pharma Plc Pde3/pde4 inhibitor/muscarinic receptor antagonist combination
PT3231444T (pt) 2014-05-12 2020-03-05 Verona Pharma Plc Novo tratamento
SI3193835T1 (en) 2014-09-15 2018-06-29 Verona Pharma PLC Bradley Court Liquid inhalation preparation containing rpl554
GB201502260D0 (en) 2015-02-11 2015-04-01 Verona Pharma Plc Salt of Pyrimido[6,1-A]Isoquinolin-4-one compound

Also Published As

Publication number Publication date
TW201806951A (zh) 2018-03-01
LT3490988T (lt) 2019-10-10
PL3490988T3 (pl) 2020-02-28
CN109641891A (zh) 2019-04-16
HUE046509T2 (hu) 2020-03-30
KR102396059B1 (ko) 2022-05-10
JP6985367B2 (ja) 2021-12-22
WO2018020249A1 (en) 2018-02-01
RS59566B1 (sr) 2019-12-31
SI3490988T1 (sl) 2019-11-29
US10710998B2 (en) 2020-07-14
HRP20192109T1 (hr) 2020-02-21
CY1122138T1 (el) 2020-11-25
EP3490988A1 (en) 2019-06-05
CN109641891B (zh) 2021-05-04
EP3490988B1 (en) 2019-08-28
PT3490988T (pt) 2019-10-28
JP2019527228A (ja) 2019-09-26
ES2751948T3 (es) 2020-04-02
KR20190034231A (ko) 2019-04-01
US20190330206A1 (en) 2019-10-31
GB201613054D0 (en) 2016-09-14
TWI739871B (zh) 2021-09-21

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