DK3019499T3 - Polycykliske-carbamoylpyridon-forbindelser og anvendelse deraf til behandling af hiv-infektioner - Google Patents

Polycykliske-carbamoylpyridon-forbindelser og anvendelse deraf til behandling af hiv-infektioner

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Publication number
DK3019499T3
DK3019499T3 DK14745053.0T DK14745053T DK3019499T3 DK 3019499 T3 DK3019499 T3 DK 3019499T3 DK 14745053 T DK14745053 T DK 14745053T DK 3019499 T3 DK3019499 T3 DK 3019499T3
Authority
DK
Denmark
Prior art keywords
carbamoylpyridon
polycyclic
compounds
treating hiv
hiv infections
Prior art date
Application number
DK14745053.0T
Other languages
Danish (da)
English (en)
Inventor
Mingzhe Ji
Teresa Alejandra Trejo Martin
Manoj C Desai
Haolun Jin
Hyung-Jung Pyun
Original Assignee
Gilead Sciences Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gilead Sciences Inc filed Critical Gilead Sciences Inc
Application granted granted Critical
Publication of DK3019499T3 publication Critical patent/DK3019499T3/da

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/18—Bridged systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
DK14745053.0T 2013-07-12 2014-07-11 Polycykliske-carbamoylpyridon-forbindelser og anvendelse deraf til behandling af hiv-infektioner DK3019499T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361845807P 2013-07-12 2013-07-12
PCT/US2014/046415 WO2015006733A1 (en) 2013-07-12 2014-07-11 Polycyclic-carbamoylpyridone compounds and their use for the treatment of hiv infections

Publications (1)

Publication Number Publication Date
DK3019499T3 true DK3019499T3 (da) 2017-11-20

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DK14745053.0T DK3019499T3 (da) 2013-07-12 2014-07-11 Polycykliske-carbamoylpyridon-forbindelser og anvendelse deraf til behandling af hiv-infektioner

Country Status (18)

Country Link
US (6) US9458159B2 (cg-RX-API-DMAC10.html)
EP (2) EP3252053B1 (cg-RX-API-DMAC10.html)
JP (1) JP6411492B2 (cg-RX-API-DMAC10.html)
AU (3) AU2014286995B2 (cg-RX-API-DMAC10.html)
CA (1) CA2918055C (cg-RX-API-DMAC10.html)
CY (1) CY1119545T1 (cg-RX-API-DMAC10.html)
DK (1) DK3019499T3 (cg-RX-API-DMAC10.html)
ES (2) ES2856867T3 (cg-RX-API-DMAC10.html)
HR (1) HRP20171807T1 (cg-RX-API-DMAC10.html)
HU (1) HUE037343T2 (cg-RX-API-DMAC10.html)
LT (1) LT3019499T (cg-RX-API-DMAC10.html)
NO (1) NO2865735T3 (cg-RX-API-DMAC10.html)
PL (1) PL3019499T3 (cg-RX-API-DMAC10.html)
PT (1) PT3019499T (cg-RX-API-DMAC10.html)
RS (1) RS56539B1 (cg-RX-API-DMAC10.html)
SI (2) SI3019499T1 (cg-RX-API-DMAC10.html)
SM (1) SMT201700525T1 (cg-RX-API-DMAC10.html)
WO (1) WO2015006733A1 (cg-RX-API-DMAC10.html)

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