DK275984A - 1-(ethoxy-carbonyloxy)ethyl-6alfa-(aminoethyl)penicillanat-1,1-dioxid, n-benzyloxycarbonylderivater deraf, fremg. til fremst. af carboxylbeskyttet 6alfa-(benzyloxycarbonylaminomethyl)penicillansyre-1,1-dioxid og grignard-reagens som mellemprodukt herved - Google Patents

1-(ethoxy-carbonyloxy)ethyl-6alfa-(aminoethyl)penicillanat-1,1-dioxid, n-benzyloxycarbonylderivater deraf, fremg. til fremst. af carboxylbeskyttet 6alfa-(benzyloxycarbonylaminomethyl)penicillansyre-1,1-dioxid og grignard-reagens som mellemprodukt herved Download PDF

Info

Publication number
DK275984A
DK275984A DK275984A DK275984A DK275984A DK 275984 A DK275984 A DK 275984A DK 275984 A DK275984 A DK 275984A DK 275984 A DK275984 A DK 275984A DK 275984 A DK275984 A DK 275984A
Authority
DK
Denmark
Prior art keywords
dioxide
6alfa
penicillanate
ethyl
benzyloxycarbonylaminomethyl
Prior art date
Application number
DK275984A
Other languages
Danish (da)
English (en)
Other versions
DK275984D0 (da
Inventor
Wayne Ernest Barth
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DK275984D0 publication Critical patent/DK275984D0/da
Publication of DK275984A publication Critical patent/DK275984A/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
DK275984A 1983-06-06 1984-06-04 1-(ethoxy-carbonyloxy)ethyl-6alfa-(aminoethyl)penicillanat-1,1-dioxid, n-benzyloxycarbonylderivater deraf, fremg. til fremst. af carboxylbeskyttet 6alfa-(benzyloxycarbonylaminomethyl)penicillansyre-1,1-dioxid og grignard-reagens som mellemprodukt herved DK275984A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/501,476 US4502990A (en) 1983-06-06 1983-06-06 Process for 6-(aminomethyl)penicillanic acid 1,1-dioxide and derivatives thereof

Publications (2)

Publication Number Publication Date
DK275984D0 DK275984D0 (da) 1984-06-04
DK275984A true DK275984A (da) 1984-12-07

Family

ID=23993716

Family Applications (1)

Application Number Title Priority Date Filing Date
DK275984A DK275984A (da) 1983-06-06 1984-06-04 1-(ethoxy-carbonyloxy)ethyl-6alfa-(aminoethyl)penicillanat-1,1-dioxid, n-benzyloxycarbonylderivater deraf, fremg. til fremst. af carboxylbeskyttet 6alfa-(benzyloxycarbonylaminomethyl)penicillansyre-1,1-dioxid og grignard-reagens som mellemprodukt herved

Country Status (21)

Country Link
US (1) US4502990A (de)
EP (1) EP0128718B1 (de)
JP (1) JPS606692A (de)
KR (1) KR870000313B1 (de)
AT (1) ATE24513T1 (de)
AU (1) AU545506B2 (de)
CA (1) CA1209983A (de)
DE (1) DE3461801D1 (de)
DK (1) DK275984A (de)
ES (1) ES533148A0 (de)
FI (1) FI842252A (de)
GR (1) GR81626B (de)
HU (1) HU191667B (de)
IL (1) IL72002A (de)
NO (1) NO842247L (de)
NZ (1) NZ208380A (de)
PH (1) PH19283A (de)
PL (1) PL144041B1 (de)
PT (1) PT78690A (de)
YU (1) YU97184A (de)
ZA (1) ZA844183B (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4868296A (en) * 1985-10-29 1989-09-19 Pfizer Inc. 6-(1-carbamoyl-1-hydroxymethyl) penicillanic acid derivatives
WO1990006928A1 (en) * 1985-10-29 1990-06-28 Barth Wayne E 6-(1-carbamoyl-1-hydroxymethyl)penicillanic acid derivatives

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4207323A (en) * 1975-11-21 1980-06-10 Merck & Co., Inc. 6-Substituted methyl penicillins, derivatives and analogues thereof
US4234579A (en) * 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
US4237051A (en) * 1979-04-19 1980-12-02 Schering Corporation Stereospecific production of 6- or 7-carbon-substituted-β-lactams
US4309347A (en) * 1979-05-16 1982-01-05 Pfizer Inc. Penicillanoyloxymethyl penicillanate 1,1,1',1'-tetraoxide
DE2927004A1 (de) * 1979-07-04 1981-05-27 Bayer Ag, 5090 Leverkusen Penicillansaeure-1,1-dioxide, ihre herstellung und ihre verwendung als arzneimittel als arzneimittel
US4287181A (en) * 1979-10-22 1981-09-01 Pfizer Inc. Derivatives of 6β-hydroxyalkylpenicillanic acids as β-lactamase inhibitors
RO87705A (ro) * 1982-01-11 1985-10-31 Pfizer Inc,Us Procedeu pentru prepararea unor derivati ai acidului 6-aminoalchilpenicilanic 1,1-dioxid

Also Published As

Publication number Publication date
YU97184A (en) 1986-06-30
PT78690A (en) 1984-07-01
DK275984D0 (da) 1984-06-04
EP0128718B1 (de) 1986-12-30
GR81626B (de) 1984-12-11
JPS606692A (ja) 1985-01-14
PL144041B1 (en) 1988-04-30
AU2907784A (en) 1984-12-13
HU191667B (en) 1987-03-30
IL72002A0 (en) 1984-10-31
PL248045A1 (en) 1985-07-30
ZA844183B (en) 1986-01-29
US4502990A (en) 1985-03-05
DE3461801D1 (en) 1987-02-05
ES8506317A1 (es) 1985-07-01
NZ208380A (en) 1987-05-29
CA1209983A (en) 1986-08-19
FI842252A (fi) 1984-12-07
HUT34203A (en) 1985-02-28
FI842252A0 (fi) 1984-06-05
EP0128718A1 (de) 1984-12-19
KR850000447A (ko) 1985-02-27
NO842247L (no) 1984-12-07
PH19283A (en) 1986-03-04
KR870000313B1 (ko) 1987-02-26
IL72002A (en) 1988-03-31
AU545506B2 (en) 1985-07-18
ATE24513T1 (de) 1987-01-15
ES533148A0 (es) 1985-07-01

Similar Documents

Publication Publication Date Title
FI881978A0 (fi) Menetelmä eperisonia sisältävän farmaseuttisen koostumuksen valmistamiseksi
DE3485546D1 (de) Zwischenprodukte zur herstellung von stickstoff enthaltenden, substituierten, heterocyclischen verbindungen.
IT8120947A0 (it) Processo per la produzione di microcapsule.
DE3485860D1 (de) Cephalosporinverbindungen, verfahren zu ihrer herstellung und pharmazeutishe praeparate.
LU84491A1 (fr) Composition anti-acneique contenant en tant que compose actif un derive d'isothiazolo-(5,4b) pyridine one-3
IT8023163A0 (it) Processo per la preparazione dicomposti organici carbossilati.
DK275984A (da) 1-(ethoxy-carbonyloxy)ethyl-6alfa-(aminoethyl)penicillanat-1,1-dioxid, n-benzyloxycarbonylderivater deraf, fremg. til fremst. af carboxylbeskyttet 6alfa-(benzyloxycarbonylaminomethyl)penicillansyre-1,1-dioxid og grignard-reagens som mellemprodukt herved
DE3870065D1 (de) Zusammensetzungen von polyarylalkanoligomeren, verfahren zu deren herstellung.
IT8221455A0 (it) Processo per la preparazione di un substrato granulare, specialmente per idrocolture, e substrato adatto come fase solida per idrocolture.
NO159658C (no) Mellomprodukt for fremstilling av 1,1-diokso-penicillanoyloksymetyl-6-(2-amino-2-fenyl-acetamido)penicillanat-antibiotika.
IT1227126B (it) Processo per la preparazione di composti penem.
IT8719283A0 (it) Metodo per produrre nastri da imballaggio.
FR2555450B1 (fr) Composition anti-acneique contenant en tant que compose actif un derive d'isothiazolo-(5,4b) pyridine one-3
SU655668A1 (ru) Травильный раствор
DE3778812D1 (de) Pro-arzneimittel von antihypercholesterinaemischen verbindungen.
IT8023364A0 (it) Processo per la produzione di alfa-6-desossi-tetracicline.
BA97155B1 (bs) Postupak za dobivanje penicilanoiloskimetil penicilanat 1,1,1-tetraoksida
IT8022659A0 (it) Processo per la produzione di cimetidina.
IT8221602A0 (it) Processo per la produzione di dl-cisteina.
ES509780A0 (es) Un metodo de produccion de un compuesto 3,5-di-t-butil-4-hidroxifenil-heterociclico sustituido.
ATE33249T1 (de) Verfahren zur herstellung von 6,6dibromopenicillans|ure-1,1-dioxyd.
BA97152B1 (bs) Postupak za proizvodnju supstituisanog piridinsulfonamidnog jedinjenja
ES509779A0 (es) Un metodo de produccion de un compuesto 3,5-dt-t-butil-4-hidroxifenil-heterociclico sustituido.
TH4958EX (th) สารประกอบ b-แลคแทม,วิธีสำหรับการสังเคาะห์สารชนิดผสมที่มีสารชนิดนี้ที่ใช้เป็นยาสำหรับรักษาโรคซึ่งติดเชื่อแบคทีเรียและอินเทอร์มีเดียทต่างๆสำหรับการสังเคราะห์สารชนิดนี้
SU1162187A1 (ru) N-(N-АНИЗИЛ- β -ОКСИЭТИЛ)-4-ЭТОКСИКАРБОНИЛ-1,2,3,6-ТЕТРАГИДРОПИРИДИН В КАЧЕСТВЕ ПОЛУПРОДУКТА ДЛЯ СИНТЕЗА 1,2,3,6-ТЕТРАГИДРОИЗОНИКОТИНОВОЙ КИСЛОТЫ

Legal Events

Date Code Title Description
AHB Application shelved due to non-payment