DK258280A - PROCEDURE FOR THE MANUFACTURING OF OXYMORPHONE - Google Patents
PROCEDURE FOR THE MANUFACTURING OF OXYMORPHONEInfo
- Publication number
- DK258280A DK258280A DK258280A DK258280A DK258280A DK 258280 A DK258280 A DK 258280A DK 258280 A DK258280 A DK 258280A DK 258280 A DK258280 A DK 258280A DK 258280 A DK258280 A DK 258280A
- Authority
- DK
- Denmark
- Prior art keywords
- oxymorphone
- procedure
- manufacturing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D489/00—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
- C07D489/06—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: with a hetero atom directly attached in position 14
- C07D489/08—Oxygen atom
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Polarising Elements (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US95305678A | 1978-10-19 | 1978-10-19 | |
PCT/US1979/000862 WO1980000841A1 (en) | 1978-10-19 | 1979-10-18 | Process for producing oxymorphone |
Publications (1)
Publication Number | Publication Date |
---|---|
DK258280A true DK258280A (en) | 1980-06-17 |
Family
ID=25493512
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK258280A DK258280A (en) | 1978-10-19 | 1980-06-17 | PROCEDURE FOR THE MANUFACTURING OF OXYMORPHONE |
Country Status (16)
Country | Link |
---|---|
JP (1) | JPS55501025A (en) |
AU (1) | AU5189779A (en) |
BE (1) | BE879494A (en) |
CA (1) | CA1108132A (en) |
CS (1) | CS211364B2 (en) |
DK (1) | DK258280A (en) |
ES (1) | ES485154A1 (en) |
FI (1) | FI793235A (en) |
FR (1) | FR2439201A1 (en) |
GB (1) | GB2049680A (en) |
IL (1) | IL58489A0 (en) |
IT (1) | IT7969032A0 (en) |
NL (1) | NL7920126A (en) |
NO (1) | NO793297L (en) |
SE (1) | SE8004454L (en) |
WO (1) | WO1980000841A1 (en) |
Families Citing this family (34)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4795813A (en) * | 1981-08-17 | 1989-01-03 | The Florida Board Of Regents On Behalf Of The Florida State University | Synthesis of derivatives of codeine and other 3-O-alkylmorphines |
US5668285A (en) * | 1986-10-31 | 1997-09-16 | The United States Of America As Represented By The Department Of Health And Human Services | Total synthesis of northebaine, normophine, noroxymorphone enantiomers and derivatives via N-Nor intermediates |
FR2636330B1 (en) * | 1988-09-13 | 1990-11-30 | Sanofi Sa | PROCESS FOR THE PREPARATION OF MORPHINANE DERIVATIVES |
ES2129395T3 (en) * | 1989-10-16 | 1999-06-16 | Us Health | TOTAL SYNTHESIS OF NORTEBAINE, NORMORPHINE, NOROXYMORPHONE ENANTIOMERS AND THEIR DERIVATIVES THROUGH N-NOR INTERMEDIATE PRODUCTS. |
WO2003004031A1 (en) | 2001-07-06 | 2003-01-16 | Endo Pharmaceuticals, Inc. | Parenteral administration of 6-hydroxy-oxymorphone for use as an analgesic |
US8329216B2 (en) | 2001-07-06 | 2012-12-11 | Endo Pharmaceuticals Inc. | Oxymorphone controlled release formulations |
US7776314B2 (en) | 2002-06-17 | 2010-08-17 | Grunenthal Gmbh | Abuse-proofed dosage system |
DE10361596A1 (en) | 2003-12-24 | 2005-09-29 | Grünenthal GmbH | Process for producing an anti-abuse dosage form |
US20070048228A1 (en) | 2003-08-06 | 2007-03-01 | Elisabeth Arkenau-Maric | Abuse-proofed dosage form |
DE102005005446A1 (en) | 2005-02-04 | 2006-08-10 | Grünenthal GmbH | Break-resistant dosage forms with sustained release |
DE10336400A1 (en) | 2003-08-06 | 2005-03-24 | Grünenthal GmbH | Anti-abuse dosage form |
DE102004032049A1 (en) | 2004-07-01 | 2006-01-19 | Grünenthal GmbH | Anti-abuse, oral dosage form |
DE102005005449A1 (en) | 2005-02-04 | 2006-08-10 | Grünenthal GmbH | Process for producing an anti-abuse dosage form |
CA2644095A1 (en) | 2006-03-02 | 2007-09-13 | Mallinckrodt Inc. | Processes for preparing morphinan-6-one products with low levels of alpha, beta-unsaturated ketone compounds |
BRPI0906467C1 (en) | 2008-01-25 | 2021-05-25 | Gruenenthal Gmbh | pharmaceutical dosage form with modified tear-resistant outer shape and controlled release |
LT2273983T (en) | 2008-05-09 | 2016-10-25 | Grünenthal GmbH | Process for the preparation of an intermediate powder formulation and a final solid dosage form under usage of a spray congealing step |
AU2010275754B2 (en) | 2009-07-22 | 2014-05-15 | Grünenthal GmbH | Tamper-resistant dosage form for oxidation-sensitive opioids |
EP2456427B1 (en) | 2009-07-22 | 2015-03-04 | Grünenthal GmbH | Hot-melt extruded controlled release dosage form |
MX2013002293A (en) | 2010-09-02 | 2013-05-09 | Gruenenthal Gmbh | Tamper resistant dosage form comprising an anionic polymer. |
WO2012028319A1 (en) | 2010-09-02 | 2012-03-08 | Grünenthal GmbH | Tamper resistant dosage form comprising inorganic salt |
BR112014002022A2 (en) | 2011-07-29 | 2017-02-21 | Gruenenthal Gmbh | tamper-resistant tablet providing immediate drug release |
LT2736497T (en) | 2011-07-29 | 2017-11-10 | Grünenthal GmbH | Tamper-resistant tablet providing immediate drug release |
US20130225697A1 (en) | 2012-02-28 | 2013-08-29 | Grunenthal Gmbh | Tamper-resistant dosage form comprising pharmacologically active compound and anionic polymer |
AU2013248351B2 (en) | 2012-04-18 | 2018-04-26 | Grunenthal Gmbh | Tamper resistant and dose-dumping resistant pharmaceutical dosage form |
US10064945B2 (en) | 2012-05-11 | 2018-09-04 | Gruenenthal Gmbh | Thermoformed, tamper-resistant pharmaceutical dosage form containing zinc |
CA2907950A1 (en) | 2013-05-29 | 2014-12-04 | Grunenthal Gmbh | Tamper-resistant dosage form containing one or more particles |
JP6466417B2 (en) | 2013-05-29 | 2019-02-06 | グリュネンタール・ゲゼルシャフト・ミト・ベシュレンクテル・ハフツング | A tamper-resistant dosage form with a bimodal release profile |
EA032465B1 (en) | 2013-07-12 | 2019-05-31 | Грюненталь Гмбх | Tamper-resistant oral pharmaceutical dosage form containing ethylene-vinyl acetate polymer and process for the production thereof |
AU2014356581C1 (en) | 2013-11-26 | 2020-05-28 | Grunenthal Gmbh | Preparation of a powdery pharmaceutical composition by means of cryo-milling |
CN106572980A (en) | 2014-05-12 | 2017-04-19 | 格吕伦塔尔有限公司 | Tamper resistant immediate release capsule formulation comprising tapentadol |
CN106456550A (en) | 2014-05-26 | 2017-02-22 | 格吕伦塔尔有限公司 | Multiparticles safeguarded against ethanolic dose-dumping |
AU2016251854A1 (en) | 2015-04-24 | 2017-10-19 | Grunenthal Gmbh | Tamper-resistant dosage form with immediate release and resistance against solvent extraction |
JP2018526414A (en) | 2015-09-10 | 2018-09-13 | グリュネンタール・ゲゼルシャフト・ミト・ベシュレンクテル・ハフツング | Protection against oral overdose with abuse-inhibiting immediate release formulations |
ES2701855T3 (en) | 2016-05-31 | 2019-02-26 | Alcaliber Investig Desarrollo E Innovacion Slu | Process for obtaining 3,14-diacetyloxymorphona from oripavine |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3249616A (en) * | 1966-05-03 | Ix-dfflydroxy-g-oxo-n-phenethylmor- phinan (cis) and production thereof | ||
US2806033A (en) * | 1955-08-03 | 1957-09-10 | Lewenstein | Morphine derivative |
US3775414A (en) * | 1972-05-10 | 1973-11-27 | Bristol Myers Co | Process for the preparation of 14-hydroxymorphinan derivatives |
-
1979
- 1979-10-12 NO NO793297A patent/NO793297L/en unknown
- 1979-10-18 BE BE0/197710A patent/BE879494A/en unknown
- 1979-10-18 ES ES485154A patent/ES485154A1/en not_active Expired
- 1979-10-18 WO PCT/US1979/000862 patent/WO1980000841A1/en unknown
- 1979-10-18 GB GB8014422A patent/GB2049680A/en not_active Withdrawn
- 1979-10-18 NL NL7920126A patent/NL7920126A/en unknown
- 1979-10-18 IT IT7969032A patent/IT7969032A0/en unknown
- 1979-10-18 FR FR7925895A patent/FR2439201A1/en not_active Withdrawn
- 1979-10-18 AU AU51897/79A patent/AU5189779A/en not_active Abandoned
- 1979-10-18 FI FI793235A patent/FI793235A/en not_active Application Discontinuation
- 1979-10-18 JP JP50190279A patent/JPS55501025A/ja active Pending
- 1979-10-18 IL IL58489A patent/IL58489A0/en unknown
- 1979-10-18 CA CA337,908A patent/CA1108132A/en not_active Expired
- 1979-10-19 CS CS797115A patent/CS211364B2/en unknown
-
1980
- 1980-06-16 SE SE8004454A patent/SE8004454L/en not_active Application Discontinuation
- 1980-06-17 DK DK258280A patent/DK258280A/en unknown
Also Published As
Publication number | Publication date |
---|---|
WO1980000841A1 (en) | 1980-05-01 |
SE8004454L (en) | 1980-06-16 |
NL7920126A (en) | 1980-08-29 |
ES485154A1 (en) | 1980-06-16 |
AU5189779A (en) | 1980-04-24 |
IT7969032A0 (en) | 1979-10-18 |
GB2049680A (en) | 1980-12-31 |
CS211364B2 (en) | 1982-02-26 |
CA1108132A (en) | 1981-09-01 |
BE879494A (en) | 1980-02-15 |
JPS55501025A (en) | 1980-11-27 |
NO793297L (en) | 1980-04-22 |
IL58489A0 (en) | 1980-01-31 |
FI793235A (en) | 1980-04-20 |
FR2439201A1 (en) | 1980-05-16 |
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