DK2515886T3 - Transdermal therapeutic system for administration of rivastigmine or derivatives thereof - Google Patents
Transdermal therapeutic system for administration of rivastigmine or derivatives thereof Download PDFInfo
- Publication number
- DK2515886T3 DK2515886T3 DK10790565.5T DK10790565T DK2515886T3 DK 2515886 T3 DK2515886 T3 DK 2515886T3 DK 10790565 T DK10790565 T DK 10790565T DK 2515886 T3 DK2515886 T3 DK 2515886T3
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- DK
- Denmark
- Prior art keywords
- reservoir
- transdermal therapeutic
- therapeutic system
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- Prior art date
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- XSVMFMHYUFZWBK-NSHDSACASA-N Rivastigmine Chemical compound CCN(C)C(=O)OC1=CC=CC([C@H](C)N(C)C)=C1 XSVMFMHYUFZWBK-NSHDSACASA-N 0.000 title claims abstract description 59
- 229960004136 rivastigmine Drugs 0.000 title claims abstract description 59
- 230000001225 therapeutic effect Effects 0.000 title claims abstract description 39
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- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 claims abstract description 31
- 150000003839 salts Chemical class 0.000 claims abstract description 15
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- A61F13/00—Bandages or dressings; Absorbent pads
- A61F13/00987—Apparatus or processes for manufacturing non-adhesive dressings or bandages
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- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/27—Esters, e.g. nitroglycerine, selenocyanates of carbamic or thiocarbamic acids, meprobamate, carbachol, neostigmine
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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- A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
- Y10T—TECHNICAL SUBJECTS COVERED BY FORMER US CLASSIFICATION
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Landscapes
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- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Inorganic Chemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Materials For Medical Uses (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP09180413 | 2009-12-22 | ||
| EP10154648 | 2010-02-25 | ||
| PCT/EP2010/069654 WO2011076621A2 (de) | 2009-12-22 | 2010-12-14 | Transdermales therapeutisches system zur verabreichung von rivastigmin oder dessen derivaten |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK2515886T3 true DK2515886T3 (en) | 2018-06-14 |
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| Application Number | Title | Priority Date | Filing Date |
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| DK10790565.5T DK2515886T3 (en) | 2009-12-22 | 2010-12-14 | Transdermal therapeutic system for administration of rivastigmine or derivatives thereof |
Country Status (16)
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| PL3254676T3 (pl) | 2009-10-30 | 2019-06-28 | Ix Biopharma Ltd | Szybko rozpuszczająca się stała postać dawkowana |
| US12186426B2 (en) | 2009-10-30 | 2025-01-07 | Ix Biopharma Ltd. | Solid dosage form |
| DE102010026903A1 (de) | 2010-07-12 | 2012-01-12 | Amw Gmbh | Transdermales therapeutisches System mit Avocadoöl oder Palmöl als Hilfsstoff |
| EP2468274B1 (de) * | 2010-12-14 | 2015-07-01 | Acino AG | Transdermales therapeutisches System zur Verabreichung eines Wirkstoffs |
| EP2711002A4 (en) * | 2011-05-20 | 2014-10-29 | Sk Chemicals Co Ltd | PLASTER WITH RIVASTIGMIN |
| EP2729148A4 (en) | 2011-07-06 | 2015-04-22 | Parkinson S Inst | COMPOSITIONS AND METHOD FOR THE TREATMENT OF SYMPTOMS IN PATIENTS WITH MORBUS PARKINSON |
| WO2013031992A1 (ja) * | 2011-08-31 | 2013-03-07 | 積水メディカル株式会社 | 貼付剤 |
| EP2594261A1 (en) | 2011-11-18 | 2013-05-22 | Labtec GmbH | Composition for transdermal administration of rivastigmine |
| DE102012000369A1 (de) | 2012-01-11 | 2013-07-11 | Alfred E. Tiefenbacher (Gmbh & Co. Kg) | Transdermales therapeutisches System mit Cholinesterase-Hemmer |
| AU2012371935A1 (en) | 2012-02-28 | 2014-09-11 | Nichiban Co., Ltd. | Transdermal patch |
| US20140083878A1 (en) * | 2012-09-21 | 2014-03-27 | Mylan Inc. | Transdermal drug delivery device |
| CN103933018A (zh) * | 2013-01-18 | 2014-07-23 | 江苏康倍得药业有限公司 | 一种透皮给药系统 |
| JPWO2015174502A1 (ja) | 2014-05-15 | 2017-05-25 | ニチバン株式会社 | リバスチグミンを含有する貼付剤のための包装体 |
| WO2016049035A1 (en) * | 2014-09-23 | 2016-03-31 | Equistar Chemicals, Lp | Polyolefin-based compositions, adhesives, and related multi-layered structures prepared therefrom |
| WO2016123406A1 (en) | 2015-01-28 | 2016-08-04 | Chrono Therapeutics Inc. | Drug delivery methods and systems |
| EP3267875A4 (en) | 2015-03-12 | 2018-12-05 | Chrono Therapeutics Inc. | Craving input and support system |
| DE102015119789A1 (de) * | 2015-11-16 | 2017-05-18 | Denso-Holding Gmbh & Co. | Korrosionsschutzzusammensetzung umfassend Polyisobutylene |
| WO2018129304A1 (en) | 2017-01-06 | 2018-07-12 | Chrono Therapeutics Inc. | Transdermal drug delivery devices and methods |
| JP6832456B2 (ja) | 2017-03-24 | 2021-02-24 | イー インク カリフォルニア， エルエルシー | 活性分子の投与率を調整するための荷電または磁気粒子を含むマイクロセル送達システム |
| TWI753284B (zh) | 2017-03-24 | 2022-01-21 | 美商伊英克加利福尼亞有限責任公司 | 活性分子遞送系統 |
| JP6972334B2 (ja) | 2017-11-14 | 2021-11-24 | イー インク カリフォルニア， エルエルシー | 多孔性伝導電極層を含む電気泳動活性分子送達システム |
| ES2983443T3 (es) * | 2018-04-17 | 2024-10-23 | Lts Lohmann Therapie Systeme Ag | Sistema terapéutico transdérmico para la administración transdérmica de solifenacina |
| CA3101966A1 (en) | 2018-05-29 | 2019-12-05 | Morningside Venture Investments Limited | Drug delivery methods and systems |
| JP2022507660A (ja) | 2018-11-16 | 2022-01-18 | モーニングサイド ベンチャー インベストメンツ リミテッド | 温度によって調節される経皮薬剤送達システム |
| CN114728155B (zh) | 2019-11-27 | 2024-04-26 | 伊英克公司 | 包括具有电蚀密封层的微单元的有益剂输送系统 |
| EP4236926A4 (en) | 2020-10-29 | 2024-08-28 | E Ink Corporation | MICROCELL SYSTEMS FOR DELIVERY OF BENEFICIAL AGENTS |
| CN116507322A (zh) | 2020-10-29 | 2023-07-28 | 伊英克加利福尼亚有限责任公司 | 用于递送亲水活性分子的微单元系统 |
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| HU201906B (en) | 1987-03-04 | 1991-01-28 | Sandoz Ag | Process for producing phenyl-carbamate derivative and acid additional salts and pharmaceutical compositions containing them |
| JPS63307818A (ja) * | 1987-06-08 | 1988-12-15 | Sekisui Chem Co Ltd | 経皮吸収貼付剤 |
| JPH07116025B2 (ja) * | 1988-03-11 | 1995-12-13 | 積水化学工業株式会社 | 貼付剤 |
| JP2693212B2 (ja) * | 1989-03-28 | 1997-12-24 | 日東電工株式会社 | 疾患治療用テープ製剤 |
| JPH08193030A (ja) | 1995-01-12 | 1996-07-30 | Nitto Denko Corp | エメダスチン貼付製剤 |
| JPH10152434A (ja) | 1996-09-26 | 1998-06-09 | Nitto Denko Corp | 経皮吸収型製剤 |
| GB9800526D0 (en) | 1998-01-12 | 1998-03-11 | Ciba Geigy Ag | Organic compounds |
| DE19814087A1 (de) * | 1998-03-30 | 1999-10-14 | Lohmann Therapie Syst Lts | Feuchtigkeitsaktivierbares therapeutisches System |
| DE19918106A1 (de) | 1999-04-22 | 2000-10-26 | Lohmann Therapie Syst Lts | Transdermales therapeutisches System mit neutralisierten Acrylathaftklebern |
| DE10033853A1 (de) | 2000-07-12 | 2002-01-31 | Hexal Ag | Transdermales therapeutisches System mit hochdispersem Siliziumdioxid |
| DE10141652B4 (de) | 2001-08-24 | 2011-04-07 | Lts Lohmann Therapie-Systeme Ag | Transdermales therapeutisches System auf der Basis von Polyacrylat-Haftklebern ohne funktionelle Gruppen und seine Verwendung |
| US20040258741A1 (en) * | 2001-10-17 | 2004-12-23 | Takaaki Terahara | Percutaneous absorption preparations |
| JP4478757B2 (ja) * | 2002-04-19 | 2010-06-09 | 日東電工株式会社 | ビソプロロール含有貼付剤 |
| US8481565B2 (en) * | 2004-12-27 | 2013-07-09 | Eisai R&D Management Co., Ltd. | Method for stabilizing anti-dementia drug |
| TWI389709B (zh) * | 2005-12-01 | 2013-03-21 | Novartis Ag | 經皮治療系統 |
| CN1994290B (zh) * | 2006-01-04 | 2011-03-16 | 上海医药工业研究院 | 卡巴拉汀透皮贴剂及其制备方法 |
| ES2466647T3 (es) * | 2006-05-08 | 2014-06-10 | Teikoku Seiyaku Co., Ltd. | Preparación absorbible por vía transdérmica que comprende un agente contra la demencia |
| US9248104B2 (en) | 2006-08-17 | 2016-02-02 | Core Tech Solutions, Inc. | Transdermal methods and systems for treating Alzheimer's disease |
| JP2009022730A (ja) * | 2007-06-18 | 2009-02-05 | Kyoritsu Yakuhin Kogyo Kk | 貼付剤 |
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- 2010-12-14 MX MX2012007214A patent/MX350357B/es active IP Right Grant
- 2010-12-14 ES ES10790565.5T patent/ES2670227T3/es active Active
- 2010-12-14 NO NO10790565A patent/NO2515886T3/no unknown
- 2010-12-14 KR KR1020127017374A patent/KR101674240B1/ko active Active
- 2010-12-14 EP EP10790565.5A patent/EP2515886B1/de active Active
- 2010-12-14 AU AU2010335309A patent/AU2010335309B2/en active Active
- 2010-12-14 US US13/518,006 patent/US8962014B2/en active Active
-
2018
- 2018-05-25 CY CY20181100570T patent/CY1120283T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ES2670227T3 (es) | 2018-05-29 |
| KR101674240B1 (ko) | 2016-11-08 |
| BR112012017168A2 (pt) | 2018-05-02 |
| AU2010335309B2 (en) | 2015-08-20 |
| BR112012017168B1 (pt) | 2022-03-15 |
| PT2515886T (pt) | 2018-05-23 |
| MX350357B (es) | 2017-09-05 |
| AU2010335309A1 (en) | 2012-07-19 |
| CA2785117A1 (en) | 2011-06-30 |
| CY1120283T1 (el) | 2019-07-10 |
| JP2013515025A (ja) | 2013-05-02 |
| MX2012007214A (es) | 2012-09-12 |
| PL2515886T3 (pl) | 2018-08-31 |
| CN102711744B (zh) | 2014-06-25 |
| WO2011076621A3 (de) | 2012-02-09 |
| NO2515886T3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 2018-09-08 |
| US20130261571A1 (en) | 2013-10-03 |
| KR20120128606A (ko) | 2012-11-27 |
| JP6083734B2 (ja) | 2017-02-22 |
| CA2785117C (en) | 2016-12-06 |
| EP2515886A2 (de) | 2012-10-31 |
| EP2515886B1 (de) | 2018-04-11 |
| WO2011076621A2 (de) | 2011-06-30 |
| US8962014B2 (en) | 2015-02-24 |
| CN102711744A (zh) | 2012-10-03 |
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