DK2503882T3 - Amidoacetonitrilforbindelser med pesticid virkning - Google Patents

Amidoacetonitrilforbindelser med pesticid virkning Download PDF

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Publication number
DK2503882T3
DK2503882T3 DK10784495.3T DK10784495T DK2503882T3 DK 2503882 T3 DK2503882 T3 DK 2503882T3 DK 10784495 T DK10784495 T DK 10784495T DK 2503882 T3 DK2503882 T3 DK 2503882T3
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DK
Denmark
Prior art keywords
cyano
formula
compound
phenoxy
compounds
Prior art date
Application number
DK10784495.3T
Other languages
English (en)
Inventor
Thomas Goebel
Heinz Sager
Noa Lle Gauvry
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Application granted granted Critical
Publication of DK2503882T3 publication Critical patent/DK2503882T3/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/49—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C255/54—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and etherified hydroxy groups bound to the carbon skeleton
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N37/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids
    • A01N37/44—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing at least one carboxylic group or a thio analogue, or a derivative thereof, and a nitrogen atom attached to the same carbon skeleton by a single or double bond, this nitrogen atom not being a member of a derivative or of a thio analogue of a carboxylic group, e.g. amino-carboxylic acids
    • A01N37/46—N-acyl derivatives
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/02—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having no bond to a nitrogen atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/44—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/62—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Dentistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Wood Science & Technology (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Claims (11)

1. Forbindelse med formlen
i, hvori Xi er halogen; X2 er CF3, OCF3j SCF3j S(0)CF3j S(02)CF3 eller SF5, 0g Y er O, S, S(O) eller S(02).
2. Forbindelse med formlen I ifølge krav 1, hvori Y er O, s eller S(02).
3. Forbindelse med formlen I ifølge krav 1, hvori Y er O.
4. Forbindelse med formlen I ifølge krav 1, hvori Y erS(02).
5. Forbindelse med formlen I ifølge et hvilket som helst af kravene 1 ti 4, hvori X1 er Cl.
6. Forbindelse med formlen I ifølge et hvilket som helst af kravene 1 til 5, hvori X2 er CF3 eller OCF3.
7. Forbindelse med formlen I ifølge krav 1, hvori Xi er Cl, X2 er OCF3, og Y er O, S, S(O) eller S(02).
8. Forbindelse med formlen I ifølge krav 1, som er N-[1-cyano-2-(5-cyano-2-{2-chlor-4-trifluormethoxyphenoxy}-phenoxy)-1-methylethyl]- 4-trifluormethoxybenzamid; eller N-[1-cyano-2-(5-cyano-2-{2-chlor-4-trifluormethoxyphenoxy}-phenoxy)-1-methylethyl]-4-trifluormethylsulfanylbenzamid; eller N-[1-cyano-2-(5-cyano-2-{2-chlor-4-trifluormethoxyphenoxy}-phenoxy)-1-methylethyl]- 4-trifluormethylsulfinylbenzamid; eller N-[1-cyano-2-(5-cyano-2-{2-chlor-4-trifluormethoxyphenoxy}-phenoxy)-1-methylethyl]- 4-trifluormethylsulfonylbenzamid.
9. Den (IS)-enantiomere af en forbindelse med formlen I ifølge et hvilket som helst af kravene 1 til 8.
10. Sammensætning til bekæmpelse af parasitter, der som aktivt stof indeholder mindst én forbindelse med formlen I ifølge et hvilket som helst af kravene 1 til 9 foruden bærestoffer og/eller dispergeringsmidler.
11. Anvendelse af en forbindelse med formlen I ifølge et hvilket som helst af kravene 1 til 9 ved fremstillingen af en farmaceutisk sammensætning mod parasitter på varmblodede dyr.
DK10784495.3T 2009-11-23 2010-11-22 Amidoacetonitrilforbindelser med pesticid virkning DK2503882T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP09176738 2009-11-23
PCT/EP2010/067924 WO2011061326A1 (en) 2009-11-23 2010-11-22 Amidoacetonitrile compounds having pesticical activity

Publications (1)

Publication Number Publication Date
DK2503882T3 true DK2503882T3 (da) 2014-03-24

Family

ID=42060754

Family Applications (1)

Application Number Title Priority Date Filing Date
DK10784495.3T DK2503882T3 (da) 2009-11-23 2010-11-22 Amidoacetonitrilforbindelser med pesticid virkning

Country Status (18)

Country Link
US (1) US8759564B2 (da)
EP (1) EP2503882B1 (da)
JP (1) JP5802870B2 (da)
CN (1) CN102595891B (da)
AR (1) AR079298A1 (da)
AU (1) AU2010320817B2 (da)
BR (1) BR112012012357B1 (da)
CA (1) CA2779563C (da)
CL (1) CL2012001248A1 (da)
CO (1) CO6460730A2 (da)
DK (1) DK2503882T3 (da)
ES (1) ES2455546T3 (da)
MX (1) MX2012005940A (da)
NZ (1) NZ599722A (da)
RU (1) RU2546871C2 (da)
UY (1) UY32992A (da)
WO (1) WO2011061326A1 (da)
ZA (1) ZA201203193B (da)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103030575B (zh) * 2013-01-04 2014-10-01 中国农业大学 一类双氰基酰胺化合物及其合成方法与应用
AR094961A1 (es) 2013-03-15 2015-09-09 Lilly Co Eli 1-hidroxi-benzooxaboroles como agentes antiparasitarios
JPWO2021177334A1 (da) * 2020-03-04 2021-09-10

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6239077B1 (en) * 1998-05-01 2001-05-29 Nihon Nohyaku Co., Ltd. Aminoacetonitrile derivative agricultural and horticultural insecticide containing the same and use thereof
AR038156A1 (es) * 2002-01-21 2004-12-29 Novartis Ag Compuestos de amidoacetonitrilo, proceso para su preparacion, composicion para controlar los parasitos, y uso de estos compuestos para preparar una composicion farmaceutica
AR040229A1 (es) * 2002-05-22 2005-03-23 Novartis Ag Amidoacetonitrilos
AR039961A1 (es) * 2002-06-06 2005-03-09 Novartis Ag Derivados de amidoacetonitrilo y su uso como pesticida
AR046757A1 (es) * 2003-12-10 2005-12-21 Novartis Ag Amidoacetonitrilos utiles como pesticidas
CN101056849B (zh) * 2004-11-09 2012-10-17 诺瓦提斯公司 从其外消旋体制备酰氨基乙腈化合物的对映体的方法
AU2006278867A1 (en) * 2005-07-25 2007-02-15 Novartis Ag Amidonitrile compounds
NZ592367A (en) * 2008-12-03 2013-05-31 Novartis Ag Amidoacetonitrile compounds and pesticidal composition thereof

Also Published As

Publication number Publication date
CN102595891A (zh) 2012-07-18
BR112012012357B1 (pt) 2019-08-27
ZA201203193B (en) 2013-01-30
EP2503882A1 (en) 2012-10-03
AR079298A1 (es) 2012-01-18
ES2455546T3 (es) 2014-04-16
WO2011061326A1 (en) 2011-05-26
RU2012125841A (ru) 2013-12-27
EP2503882B1 (en) 2014-03-05
US20120232138A1 (en) 2012-09-13
CA2779563C (en) 2018-03-20
MX2012005940A (es) 2012-06-25
AU2010320817B2 (en) 2014-02-06
AU2010320817A1 (en) 2012-05-24
CN102595891B (zh) 2013-11-13
CA2779563A1 (en) 2011-05-26
US8759564B2 (en) 2014-06-24
UY32992A (es) 2011-04-29
JP5802870B2 (ja) 2015-11-04
NZ599722A (en) 2014-02-28
RU2546871C2 (ru) 2015-04-10
CL2012001248A1 (es) 2012-09-28
JP2013511495A (ja) 2013-04-04
CO6460730A2 (es) 2012-06-15
BR112012012357A2 (pt) 2015-09-08

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