DK226983A - Fremgangsmaade til fremstilling af methylammoniumderivater af 4,4-dioxopenicillansyre - Google Patents
Fremgangsmaade til fremstilling af methylammoniumderivater af 4,4-dioxopenicillansyre Download PDFInfo
- Publication number
- DK226983A DK226983A DK226983A DK226983A DK226983A DK 226983 A DK226983 A DK 226983A DK 226983 A DK226983 A DK 226983A DK 226983 A DK226983 A DK 226983A DK 226983 A DK226983 A DK 226983A
- Authority
- DK
- Denmark
- Prior art keywords
- methylammonium
- derivatives
- preparing
- dioxopenicillanic acid
- dioxopenicillanic
- Prior art date
Links
- BAVYZALUXZFZLV-UHFFFAOYSA-N Methylamine Chemical class NC BAVYZALUXZFZLV-UHFFFAOYSA-N 0.000 title 1
- 239000002253 acid Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/381,104 US4428935A (en) | 1982-05-24 | 1982-05-24 | Penicillanic acid dioxide prodrug |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK226983D0 DK226983D0 (da) | 1983-05-20 |
| DK226983A true DK226983A (da) | 1983-11-25 |
Family
ID=23503664
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK226983A DK226983A (da) | 1982-05-24 | 1983-05-20 | Fremgangsmaade til fremstilling af methylammoniumderivater af 4,4-dioxopenicillansyre |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US4428935A (en:Method) |
| EP (1) | EP0095341B1 (en:Method) |
| JP (1) | JPS58216191A (en:Method) |
| DE (1) | DE3362266D1 (en:Method) |
| DK (1) | DK226983A (en:Method) |
| GR (1) | GR79260B (en:Method) |
| IE (1) | IE55577B1 (en:Method) |
Families Citing this family (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4681943A (en) * | 1984-11-30 | 1987-07-21 | The Dow Chemical Company | 1-acyl-1-(2-pyridinyl)semicarbazides |
| US4946959A (en) * | 1984-11-30 | 1990-08-07 | The Dow Chemical Company | Method of preparing 5-alkyl-1-(2-pyridinyl)-1H-1,2,4-triazol-3-ols |
| JPH06104671B2 (ja) * | 1990-04-13 | 1994-12-21 | ファイザー・インコーポレーテッド | スルタミシリン中間体の製造方法 |
| US7189351B2 (en) * | 2001-10-25 | 2007-03-13 | Spherix Incorporated | D-tagatose as an anti-biofilm agent |
| PA8579701A1 (es) * | 2002-08-23 | 2005-05-24 | Pfizer Prod Inc | Profarmaco inhibidor de beta-lactamasa |
| CA2528065A1 (en) * | 2003-06-05 | 2004-12-16 | Pfizer Products Inc. | Beta-lactamase inhibitor prodrug |
| KR20070058381A (ko) * | 2004-04-27 | 2007-06-08 | 메디시노바, 인크. | 염증성 질환 치료용 페녹시알킬카르복실 산 유도체 |
| PL2121593T3 (pl) | 2006-12-10 | 2015-11-30 | Chongxi Yu | Przezskórne systemy dostarczania antybiotyków beta-laktamowych |
| US9969751B2 (en) | 2009-06-10 | 2018-05-15 | Techfields Pharma Co., Ltd. | High penetration prodrug compositions of antimicrobials and antimicrobial-related compounds |
| JP5916129B2 (ja) * | 2009-06-10 | 2016-05-11 | テックフィールズ バイオケム カンパニー リミテッド | 抗菌薬および抗菌薬関連化合物の高透過性組成物またはプロドラッグ |
| JP5732453B2 (ja) | 2009-06-25 | 2015-06-10 | アルカーメス ファーマ アイルランド リミテッド | Ｎｈ酸性化合物のプロドラッグ |
| US8431576B2 (en) | 2009-06-25 | 2013-04-30 | Alkermes Pharma Ireland Limited | Heterocyclic compounds for the treatment of neurological and psychological disorders |
| US8592427B2 (en) | 2010-06-24 | 2013-11-26 | Alkermes Pharma Ireland Limited | Prodrugs of NH-acidic compounds: ester, carbonate, carbamate and phosphonate derivatives |
| LT2685979T (lt) | 2011-03-18 | 2016-12-12 | Alkermes Pharma Ireland Limited | Injekcinės farmacinės kompozicijos, apimančios vandenyje netirpų antipsichotiką, sorbitano lauratą ir polisorbatą 20 |
| KR20190085184A (ko) * | 2011-07-28 | 2019-07-17 | 켐팜 인코포레이티드 | 메틸페니데이트 프로드러그, 이의 제조 방법 및 사용 방법 |
| AU2012351747B2 (en) | 2011-12-15 | 2016-05-12 | Alkermes Pharma Ireland Limited | Prodrugs of secondary amine compounds |
| CA2867137C (en) | 2012-03-19 | 2020-12-08 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions comprising aripiprazole prodrugs and benzyl alcohol |
| ES2764383T3 (es) | 2012-03-19 | 2020-06-03 | Alkermes Pharma Ireland Ltd | Composiciones farmacéuticas que comprenden ésteres de glicerol |
| WO2013142198A1 (en) | 2012-03-19 | 2013-09-26 | Alkermes Pharma Ireland Limited | Pharmaaceutical compositions comprising fatty acid esters |
| NZ631345A (en) | 2012-09-19 | 2017-06-30 | Alkermes Pharma Ireland Ltd | Pharmaceutical compositions having improved storage stability |
| CN104812388A (zh) * | 2012-10-05 | 2015-07-29 | 斯菲拉制药私人有限公司 | 新型化合物、其合成及其用途 |
| BR112016021535A8 (pt) | 2014-03-20 | 2021-07-20 | Alkermes Pharma Ireland Ltd | kit compreendendo formulações de aripiprazol tendo velocidades de injeção aumentadas útil para o tratamento de uma desordem do sistema nervoso central e uso |
| CA3092335A1 (en) | 2018-03-05 | 2019-09-12 | Alkermes Pharma Ireland Limited | Aripiprazole dosing strategy |
| CN114286811B (zh) * | 2019-04-17 | 2024-03-08 | 伊克斯切尔制药有限责任公司 | 富马酸单甲酯的前药 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1255034A (en) * | 1968-09-06 | 1971-11-24 | Beecham Group Ltd | Penicillin esters |
| NL7401782A (en:Method) * | 1973-02-14 | 1974-08-16 | ||
| US4234579A (en) | 1977-06-07 | 1980-11-18 | Pfizer Inc. | Penicillanic acid 1,1-dioxides as β-lactamase inhibitors |
| JPS6056160B2 (ja) | 1977-06-07 | 1985-12-09 | フアイザ−・インコ−ポレ−テツド | β−ラクタマ−ゼ阻害剤としてのペニシラン酸１，１−ジオキシド |
| US4244951A (en) | 1979-05-16 | 1981-01-13 | Pfizer Inc. | Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide |
| US4376767A (en) * | 1981-01-02 | 1983-03-15 | Merck & Co., Inc. | Pyridylmethyl esters of selected bio-affecting carboxylic acids |
| US4323499A (en) | 1981-01-05 | 1982-04-06 | Pfizer Inc. | 6-(2-Aryl-2-(1,1-dioxopenicillanoyloxy-methoxycarbonyl)acetamido penicillanic acids |
-
1982
- 1982-05-24 US US06/381,104 patent/US4428935A/en not_active Expired - Lifetime
-
1983
- 1983-05-20 DK DK226983A patent/DK226983A/da not_active Application Discontinuation
- 1983-05-20 DE DE8383302891T patent/DE3362266D1/de not_active Expired
- 1983-05-20 EP EP83302891A patent/EP0095341B1/en not_active Expired
- 1983-05-23 IE IE1203/83A patent/IE55577B1/en unknown
- 1983-05-23 GR GR71431A patent/GR79260B/el unknown
- 1983-05-24 JP JP58091409A patent/JPS58216191A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| US4428935A (en) | 1984-01-31 |
| EP0095341B1 (en) | 1986-02-26 |
| GR79260B (en:Method) | 1984-10-22 |
| IE55577B1 (en) | 1990-11-07 |
| EP0095341A1 (en) | 1983-11-30 |
| IE831203L (en) | 1983-11-24 |
| DE3362266D1 (de) | 1986-04-03 |
| DK226983D0 (da) | 1983-05-20 |
| JPS58216191A (ja) | 1983-12-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AHB | Application shelved due to non-payment |