DK226983D0 - Fremgangsmade til fremstilling af methylammoniumderivater af 4,4-dioxopenicillansyre - Google Patents
Fremgangsmade til fremstilling af methylammoniumderivater af 4,4-dioxopenicillansyreInfo
- Publication number
- DK226983D0 DK226983D0 DK2269/83A DK226983A DK226983D0 DK 226983 D0 DK226983 D0 DK 226983D0 DK 2269/83 A DK2269/83 A DK 2269/83A DK 226983 A DK226983 A DK 226983A DK 226983 D0 DK226983 D0 DK 226983D0
- Authority
- DK
- Denmark
- Prior art keywords
- methylammonium
- derivatives
- preparing
- dioxopenicillanic acid
- dioxopenicillanic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US06/381,104 US4428935A (en) | 1982-05-24 | 1982-05-24 | Penicillanic acid dioxide prodrug |
Publications (2)
Publication Number | Publication Date |
---|---|
DK226983D0 true DK226983D0 (da) | 1983-05-20 |
DK226983A DK226983A (da) | 1983-11-25 |
Family
ID=23503664
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK226983A DK226983A (da) | 1982-05-24 | 1983-05-20 | Fremgangsmaade til fremstilling af methylammoniumderivater af 4,4-dioxopenicillansyre |
Country Status (7)
Country | Link |
---|---|
US (1) | US4428935A (da) |
EP (1) | EP0095341B1 (da) |
JP (1) | JPS58216191A (da) |
DE (1) | DE3362266D1 (da) |
DK (1) | DK226983A (da) |
GR (1) | GR79260B (da) |
IE (1) | IE55577B1 (da) |
Families Citing this family (24)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4946959A (en) * | 1984-11-30 | 1990-08-07 | The Dow Chemical Company | Method of preparing 5-alkyl-1-(2-pyridinyl)-1H-1,2,4-triazol-3-ols |
US4681943A (en) * | 1984-11-30 | 1987-07-21 | The Dow Chemical Company | 1-acyl-1-(2-pyridinyl)semicarbazides |
DE69103003T2 (de) * | 1990-04-13 | 1994-11-03 | Pfizer Inc., Groton, Conn. | Verfahren für sultamicillinzwischenprodukt. |
US7189351B2 (en) * | 2001-10-25 | 2007-03-13 | Spherix Incorporated | D-tagatose as an anti-biofilm agent |
PA8579701A1 (es) * | 2002-08-23 | 2005-05-24 | Pfizer Prod Inc | Profarmaco inhibidor de beta-lactamasa |
WO2004108733A1 (en) * | 2003-06-05 | 2004-12-16 | Pfizer Products Inc. | Beta-lactamase inhibitor prodrug |
KR20070058381A (ko) | 2004-04-27 | 2007-06-08 | 메디시노바, 인크. | 염증성 질환 치료용 페녹시알킬카르복실 산 유도체 |
CN101547898B (zh) | 2006-12-10 | 2014-09-24 | 于崇曦 | β-内酰胺类抗生素的透皮给药系统 |
JP5916129B2 (ja) * | 2009-06-10 | 2016-05-11 | テックフィールズ バイオケム カンパニー リミテッド | 抗菌薬および抗菌薬関連化合物の高透過性組成物またはプロドラッグ |
US9969751B2 (en) | 2009-06-10 | 2018-05-15 | Techfields Pharma Co., Ltd. | High penetration prodrug compositions of antimicrobials and antimicrobial-related compounds |
EP2445343B1 (en) | 2009-06-25 | 2021-08-04 | Alkermes Pharma Ireland Limited | Prodrugs of nh-acidic compounds |
AU2010266018B2 (en) | 2009-06-25 | 2014-01-09 | Alkermes Pharma Ireland Limited | Heterocyclic compounds for the treatment of neurological and psychological disorders |
NZ604423A (en) | 2010-06-24 | 2015-01-30 | Alkermes Pharma Ireland Ltd | Prodrugs of nh-acidic compounds: ester, carbonate, carbamate and phosphonate derivatives |
EP4327872A3 (en) | 2011-03-18 | 2024-07-10 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions comprising sorbitan esters |
KR20190085184A (ko) * | 2011-07-28 | 2019-07-17 | 켐팜 인코포레이티드 | 메틸페니데이트 프로드러그, 이의 제조 방법 및 사용 방법 |
US8969337B2 (en) | 2011-12-15 | 2015-03-03 | Alkermes Pharma Ireland Limited | Prodrugs of secondary amine compounds |
NZ630428A (en) | 2012-03-19 | 2017-02-24 | Alkermes Pharma Ireland Ltd | Pharmaceutical compositions comprising benzyl alcohol |
NZ630643A (en) | 2012-03-19 | 2017-08-25 | Alkermes Pharma Ireland Ltd | Pharmaceutical compositions comprising fatty acid esters |
ES2764383T3 (es) | 2012-03-19 | 2020-06-03 | Alkermes Pharma Ireland Ltd | Composiciones farmacéuticas que comprenden ésteres de glicerol |
CA2885196C (en) | 2012-09-19 | 2021-06-22 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions having improved storage stability |
EP2903614B1 (en) * | 2012-10-05 | 2021-09-29 | Sphaera Pharma Pte. Ltd | Novel compounds, their synthesis and their uses |
WO2015143145A1 (en) | 2014-03-20 | 2015-09-24 | Alkermes Pharma Ireland Limited | Aripiprazole formulations having increased injection speeds |
US11273158B2 (en) | 2018-03-05 | 2022-03-15 | Alkermes Pharma Ireland Limited | Aripiprazole dosing strategy |
CN114286811B (zh) * | 2019-04-17 | 2024-03-08 | 伊克斯切尔制药有限责任公司 | 富马酸单甲酯的前药 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1255034A (en) * | 1968-09-06 | 1971-11-24 | Beecham Group Ltd | Penicillin esters |
NL7401782A (da) * | 1973-02-14 | 1974-08-16 | ||
JPS6056160B2 (ja) * | 1977-06-07 | 1985-12-09 | フアイザ−・インコ−ポレ−テツド | β−ラクタマ−ゼ阻害剤としてのペニシラン酸1,1−ジオキシド |
US4234579A (en) | 1977-06-07 | 1980-11-18 | Pfizer Inc. | Penicillanic acid 1,1-dioxides as β-lactamase inhibitors |
US4244951A (en) | 1979-05-16 | 1981-01-13 | Pfizer Inc. | Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide |
US4376767A (en) * | 1981-01-02 | 1983-03-15 | Merck & Co., Inc. | Pyridylmethyl esters of selected bio-affecting carboxylic acids |
US4323499A (en) | 1981-01-05 | 1982-04-06 | Pfizer Inc. | 6-(2-Aryl-2-(1,1-dioxopenicillanoyloxy-methoxycarbonyl)acetamido penicillanic acids |
-
1982
- 1982-05-24 US US06/381,104 patent/US4428935A/en not_active Expired - Lifetime
-
1983
- 1983-05-20 DK DK226983A patent/DK226983A/da not_active Application Discontinuation
- 1983-05-20 EP EP83302891A patent/EP0095341B1/en not_active Expired
- 1983-05-20 DE DE8383302891T patent/DE3362266D1/de not_active Expired
- 1983-05-23 IE IE1203/83A patent/IE55577B1/en unknown
- 1983-05-23 GR GR71431A patent/GR79260B/el unknown
- 1983-05-24 JP JP58091409A patent/JPS58216191A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
JPS58216191A (ja) | 1983-12-15 |
DE3362266D1 (de) | 1986-04-03 |
GR79260B (da) | 1984-10-22 |
US4428935A (en) | 1984-01-31 |
EP0095341B1 (en) | 1986-02-26 |
IE55577B1 (en) | 1990-11-07 |
EP0095341A1 (en) | 1983-11-30 |
DK226983A (da) | 1983-11-25 |
IE831203L (en) | 1983-11-24 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
AHB | Application shelved due to non-payment |