DK226983D0 - Fremgangsmade til fremstilling af methylammoniumderivater af 4,4-dioxopenicillansyre - Google Patents

Fremgangsmade til fremstilling af methylammoniumderivater af 4,4-dioxopenicillansyre

Info

Publication number
DK226983D0
DK226983D0 DK2269/83A DK226983A DK226983D0 DK 226983 D0 DK226983 D0 DK 226983D0 DK 2269/83 A DK2269/83 A DK 2269/83A DK 226983 A DK226983 A DK 226983A DK 226983 D0 DK226983 D0 DK 226983D0
Authority
DK
Denmark
Prior art keywords
methylammonium
derivatives
preparing
dioxopenicillanic acid
dioxopenicillanic
Prior art date
Application number
DK2269/83A
Other languages
English (en)
Other versions
DK226983A (da
Inventor
Robert Fischer Myers
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DK226983D0 publication Critical patent/DK226983D0/da
Publication of DK226983A publication Critical patent/DK226983A/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK226983A 1982-05-24 1983-05-20 Fremgangsmaade til fremstilling af methylammoniumderivater af 4,4-dioxopenicillansyre DK226983A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/381,104 US4428935A (en) 1982-05-24 1982-05-24 Penicillanic acid dioxide prodrug

Publications (2)

Publication Number Publication Date
DK226983D0 true DK226983D0 (da) 1983-05-20
DK226983A DK226983A (da) 1983-11-25

Family

ID=23503664

Family Applications (1)

Application Number Title Priority Date Filing Date
DK226983A DK226983A (da) 1982-05-24 1983-05-20 Fremgangsmaade til fremstilling af methylammoniumderivater af 4,4-dioxopenicillansyre

Country Status (7)

Country Link
US (1) US4428935A (da)
EP (1) EP0095341B1 (da)
JP (1) JPS58216191A (da)
DE (1) DE3362266D1 (da)
DK (1) DK226983A (da)
GR (1) GR79260B (da)
IE (1) IE55577B1 (da)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4946959A (en) * 1984-11-30 1990-08-07 The Dow Chemical Company Method of preparing 5-alkyl-1-(2-pyridinyl)-1H-1,2,4-triazol-3-ols
US4681943A (en) * 1984-11-30 1987-07-21 The Dow Chemical Company 1-acyl-1-(2-pyridinyl)semicarbazides
DE69103003T2 (de) * 1990-04-13 1994-11-03 Pfizer Inc., Groton, Conn. Verfahren für sultamicillinzwischenprodukt.
US7189351B2 (en) * 2001-10-25 2007-03-13 Spherix Incorporated D-tagatose as an anti-biofilm agent
PA8579701A1 (es) * 2002-08-23 2005-05-24 Pfizer Prod Inc Profarmaco inhibidor de beta-lactamasa
WO2004108733A1 (en) * 2003-06-05 2004-12-16 Pfizer Products Inc. Beta-lactamase inhibitor prodrug
KR20070058381A (ko) 2004-04-27 2007-06-08 메디시노바, 인크. 염증성 질환 치료용 페녹시알킬카르복실 산 유도체
CN101547898B (zh) 2006-12-10 2014-09-24 于崇曦 β-内酰胺类抗生素的透皮给药系统
JP5916129B2 (ja) * 2009-06-10 2016-05-11 テックフィールズ バイオケム カンパニー リミテッド 抗菌薬および抗菌薬関連化合物の高透過性組成物またはプロドラッグ
US9969751B2 (en) 2009-06-10 2018-05-15 Techfields Pharma Co., Ltd. High penetration prodrug compositions of antimicrobials and antimicrobial-related compounds
EP2445343B1 (en) 2009-06-25 2021-08-04 Alkermes Pharma Ireland Limited Prodrugs of nh-acidic compounds
AU2010266018B2 (en) 2009-06-25 2014-01-09 Alkermes Pharma Ireland Limited Heterocyclic compounds for the treatment of neurological and psychological disorders
NZ604423A (en) 2010-06-24 2015-01-30 Alkermes Pharma Ireland Ltd Prodrugs of nh-acidic compounds: ester, carbonate, carbamate and phosphonate derivatives
EP4327872A3 (en) 2011-03-18 2024-07-10 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising sorbitan esters
KR20190085184A (ko) * 2011-07-28 2019-07-17 켐팜 인코포레이티드 메틸페니데이트 프로드러그, 이의 제조 방법 및 사용 방법
US8969337B2 (en) 2011-12-15 2015-03-03 Alkermes Pharma Ireland Limited Prodrugs of secondary amine compounds
NZ630428A (en) 2012-03-19 2017-02-24 Alkermes Pharma Ireland Ltd Pharmaceutical compositions comprising benzyl alcohol
NZ630643A (en) 2012-03-19 2017-08-25 Alkermes Pharma Ireland Ltd Pharmaceutical compositions comprising fatty acid esters
ES2764383T3 (es) 2012-03-19 2020-06-03 Alkermes Pharma Ireland Ltd Composiciones farmacéuticas que comprenden ésteres de glicerol
CA2885196C (en) 2012-09-19 2021-06-22 Alkermes Pharma Ireland Limited Pharmaceutical compositions having improved storage stability
EP2903614B1 (en) * 2012-10-05 2021-09-29 Sphaera Pharma Pte. Ltd Novel compounds, their synthesis and their uses
WO2015143145A1 (en) 2014-03-20 2015-09-24 Alkermes Pharma Ireland Limited Aripiprazole formulations having increased injection speeds
US11273158B2 (en) 2018-03-05 2022-03-15 Alkermes Pharma Ireland Limited Aripiprazole dosing strategy
CN114286811B (zh) * 2019-04-17 2024-03-08 伊克斯切尔制药有限责任公司 富马酸单甲酯的前药

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1255034A (en) * 1968-09-06 1971-11-24 Beecham Group Ltd Penicillin esters
NL7401782A (da) * 1973-02-14 1974-08-16
JPS6056160B2 (ja) * 1977-06-07 1985-12-09 フアイザ−・インコ−ポレ−テツド β−ラクタマ−ゼ阻害剤としてのペニシラン酸1,1−ジオキシド
US4234579A (en) 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
US4244951A (en) 1979-05-16 1981-01-13 Pfizer Inc. Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide
US4376767A (en) * 1981-01-02 1983-03-15 Merck & Co., Inc. Pyridylmethyl esters of selected bio-affecting carboxylic acids
US4323499A (en) 1981-01-05 1982-04-06 Pfizer Inc. 6-(2-Aryl-2-(1,1-dioxopenicillanoyloxy-methoxycarbonyl)acetamido penicillanic acids

Also Published As

Publication number Publication date
JPS58216191A (ja) 1983-12-15
DE3362266D1 (de) 1986-04-03
GR79260B (da) 1984-10-22
US4428935A (en) 1984-01-31
EP0095341B1 (en) 1986-02-26
IE55577B1 (en) 1990-11-07
EP0095341A1 (en) 1983-11-30
DK226983A (da) 1983-11-25
IE831203L (en) 1983-11-24

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Legal Events

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AHB Application shelved due to non-payment