DK226983A - Fremgangsmaade til fremstilling af methylammoniumderivater af 4,4-dioxopenicillansyre - Google Patents
Fremgangsmaade til fremstilling af methylammoniumderivater af 4,4-dioxopenicillansyre Download PDFInfo
- Publication number
- DK226983A DK226983A DK226983A DK226983A DK226983A DK 226983 A DK226983 A DK 226983A DK 226983 A DK226983 A DK 226983A DK 226983 A DK226983 A DK 226983A DK 226983 A DK226983 A DK 226983A
- Authority
- DK
- Denmark
- Prior art keywords
- methylammonium
- derivatives
- preparing
- dioxopenicillanic acid
- dioxopenicillanic
- Prior art date
Links
- BAVYZALUXZFZLV-UHFFFAOYSA-N Methylamine Chemical class NC BAVYZALUXZFZLV-UHFFFAOYSA-N 0.000 title 1
- 239000002253 acid Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/381,104 US4428935A (en) | 1982-05-24 | 1982-05-24 | Penicillanic acid dioxide prodrug |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK226983D0 DK226983D0 (da) | 1983-05-20 |
| DK226983A true DK226983A (da) | 1983-11-25 |
Family
ID=23503664
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK226983A DK226983A (da) | 1982-05-24 | 1983-05-20 | Fremgangsmaade til fremstilling af methylammoniumderivater af 4,4-dioxopenicillansyre |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US4428935A (Sortimente) |
| EP (1) | EP0095341B1 (Sortimente) |
| JP (1) | JPS58216191A (Sortimente) |
| DE (1) | DE3362266D1 (Sortimente) |
| DK (1) | DK226983A (Sortimente) |
| GR (1) | GR79260B (Sortimente) |
| IE (1) | IE55577B1 (Sortimente) |
Families Citing this family (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4681943A (en) * | 1984-11-30 | 1987-07-21 | The Dow Chemical Company | 1-acyl-1-(2-pyridinyl)semicarbazides |
| US4946959A (en) * | 1984-11-30 | 1990-08-07 | The Dow Chemical Company | Method of preparing 5-alkyl-1-(2-pyridinyl)-1H-1,2,4-triazol-3-ols |
| CA2078217C (en) * | 1990-04-13 | 2000-02-22 | Dennis M. Godek | Process for sultamicillin intermediate |
| US7189351B2 (en) * | 2001-10-25 | 2007-03-13 | Spherix Incorporated | D-tagatose as an anti-biofilm agent |
| PA8579701A1 (es) * | 2002-08-23 | 2005-05-24 | Pfizer Prod Inc | Profarmaco inhibidor de beta-lactamasa |
| JP2006526612A (ja) * | 2003-06-05 | 2006-11-24 | ファイザー・プロダクツ・インク | ベータ−ラクタマーゼ阻害剤・プロドラッグ |
| WO2005105073A1 (en) * | 2004-04-27 | 2005-11-10 | Medicinova, Inc. | Phenoxyalkycarboxylic acid derivatives in the treatment of inflammatory diseases |
| ES2547258T3 (es) | 2006-12-10 | 2015-10-02 | Chongxi Yu | Sistemas de administración transdérmica de antibióticos beta-lactama |
| RU2586287C2 (ru) * | 2009-06-10 | 2016-06-10 | Текфилдз Байокем Ко., Лтд. | Композиции или пролекарства противомикробных и родственных противомикробным соединений, обладающие высокой проникающей способностью |
| US9969751B2 (en) | 2009-06-10 | 2018-05-15 | Techfields Pharma Co., Ltd. | High penetration prodrug compositions of antimicrobials and antimicrobial-related compounds |
| ES2885698T3 (es) | 2009-06-25 | 2021-12-15 | Alkermes Pharma Ireland Ltd | Profármacos de compuestos nh-ácidos |
| PL2445502T5 (pl) | 2009-06-25 | 2023-03-13 | Alkermes Pharma Ireland Limited | Związki heterocykliczne do leczenia zaburzeń neurologicznych i psychologicznych |
| US8592427B2 (en) | 2010-06-24 | 2013-11-26 | Alkermes Pharma Ireland Limited | Prodrugs of NH-acidic compounds: ester, carbonate, carbamate and phosphonate derivatives |
| PT2685979T (pt) | 2011-03-18 | 2016-12-02 | Alkermes Pharma Ireland Ltd | Composições farmacêuticas injetáveis compreendendo um antipsicótico solúvel em água, laurato de sorbitano e polissorbato 20 |
| PL2736510T3 (pl) * | 2011-07-28 | 2017-07-31 | Kempharm, Inc. | Proleki metylofenidatu, procesy ich wytwarzania i stosowania |
| NZ722096A (en) | 2011-12-15 | 2016-11-25 | Alkermes Pharma Ireland Ltd | Prodrugs of secondary amine compounds |
| CA2867121C (en) | 2012-03-19 | 2021-05-25 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions comprising fatty acid esters |
| JP6219918B2 (ja) | 2012-03-19 | 2017-10-25 | アルカームス ファーマ アイルランド リミテッド | グリセロールエステルを含む医薬組成物 |
| AU2013235526B2 (en) | 2012-03-19 | 2017-11-30 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions comprising benzyl alcohol |
| US9193685B2 (en) | 2012-09-19 | 2015-11-24 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions having improved storage stability |
| EP2903614B1 (en) * | 2012-10-05 | 2021-09-29 | Sphaera Pharma Pte. Ltd | Novel compounds, their synthesis and their uses |
| WO2015143145A1 (en) | 2014-03-20 | 2015-09-24 | Alkermes Pharma Ireland Limited | Aripiprazole formulations having increased injection speeds |
| EP3761983A1 (en) | 2018-03-05 | 2021-01-13 | Alkermes Pharma Ireland Limited | Aripiprazole dosing strategy |
| JP7406566B2 (ja) * | 2019-04-17 | 2023-12-27 | イクシェル ファーマ エルエルシー | フマル酸モノメチルのプロドラッグ |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1255034A (en) * | 1968-09-06 | 1971-11-24 | Beecham Group Ltd | Penicillin esters |
| NL7401782A (Sortimente) * | 1973-02-14 | 1974-08-16 | ||
| JPS6056160B2 (ja) * | 1977-06-07 | 1985-12-09 | フアイザ−・インコ−ポレ−テツド | β−ラクタマ−ゼ阻害剤としてのペニシラン酸１，１−ジオキシド |
| US4234579A (en) | 1977-06-07 | 1980-11-18 | Pfizer Inc. | Penicillanic acid 1,1-dioxides as β-lactamase inhibitors |
| US4244951A (en) | 1979-05-16 | 1981-01-13 | Pfizer Inc. | Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide |
| US4376767A (en) * | 1981-01-02 | 1983-03-15 | Merck & Co., Inc. | Pyridylmethyl esters of selected bio-affecting carboxylic acids |
| US4323499A (en) | 1981-01-05 | 1982-04-06 | Pfizer Inc. | 6-(2-Aryl-2-(1,1-dioxopenicillanoyloxy-methoxycarbonyl)acetamido penicillanic acids |
-
1982
- 1982-05-24 US US06/381,104 patent/US4428935A/en not_active Expired - Lifetime
-
1983
- 1983-05-20 EP EP83302891A patent/EP0095341B1/en not_active Expired
- 1983-05-20 DE DE8383302891T patent/DE3362266D1/de not_active Expired
- 1983-05-20 DK DK226983A patent/DK226983A/da not_active Application Discontinuation
- 1983-05-23 IE IE1203/83A patent/IE55577B1/en unknown
- 1983-05-23 GR GR71431A patent/GR79260B/el unknown
- 1983-05-24 JP JP58091409A patent/JPS58216191A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| JPS58216191A (ja) | 1983-12-15 |
| EP0095341A1 (en) | 1983-11-30 |
| IE831203L (en) | 1983-11-24 |
| DE3362266D1 (de) | 1986-04-03 |
| DK226983D0 (da) | 1983-05-20 |
| US4428935A (en) | 1984-01-31 |
| IE55577B1 (en) | 1990-11-07 |
| GR79260B (Sortimente) | 1984-10-22 |
| EP0095341B1 (en) | 1986-02-26 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AHB | Application shelved due to non-payment |