DK193881A - Fremgangsmaade til fremstilling af 23-ketoderivater af c-76forbindelser - Google Patents

Fremgangsmaade til fremstilling af 23-ketoderivater af c-76forbindelser

Info

Publication number
DK193881A
DK193881A DK193881A DK193881A DK193881A DK 193881 A DK193881 A DK 193881A DK 193881 A DK193881 A DK 193881A DK 193881 A DK193881 A DK 193881A DK 193881 A DK193881 A DK 193881A
Authority
DK
Denmark
Prior art keywords
compounds
derivatives
chromic acid
oxidized
ketode
Prior art date
Application number
DK193881A
Other languages
Danish (da)
English (en)
Inventor
A J Kempf
J G Macconnell
H H Mrozik
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of DK193881A publication Critical patent/DK193881A/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DK193881A 1980-05-02 1981-05-01 Fremgangsmaade til fremstilling af 23-ketoderivater af c-76forbindelser DK193881A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/146,725 US4289760A (en) 1980-05-02 1980-05-02 23-Keto derivatives of C-076 compounds

Publications (1)

Publication Number Publication Date
DK193881A true DK193881A (da) 1981-11-03

Family

ID=22518711

Family Applications (1)

Application Number Title Priority Date Filing Date
DK193881A DK193881A (da) 1980-05-02 1981-05-01 Fremgangsmaade til fremstilling af 23-ketoderivater af c-76forbindelser

Country Status (13)

Country Link
US (1) US4289760A (pt)
EP (1) EP0040913B1 (pt)
JP (1) JPS5718684A (pt)
AT (1) ATE8637T1 (pt)
AU (1) AU547211B2 (pt)
CA (1) CA1168605A (pt)
DE (1) DE3165016D1 (pt)
DK (1) DK193881A (pt)
ES (1) ES501777A0 (pt)
GR (1) GR74875B (pt)
NZ (1) NZ196897A (pt)
PT (1) PT72915B (pt)
ZA (1) ZA812908B (pt)

Families Citing this family (40)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57139012A (en) * 1981-02-23 1982-08-27 Sankyo Co Ltd Anthelmintic composition
US4333925A (en) * 1981-05-11 1982-06-08 Merck & Co., Inc. Derivatives of C-076 compounds
US4423209A (en) * 1982-02-26 1983-12-27 Merck & Co., Inc. Processes for the interconversion of avermectin compounds
US4510133A (en) * 1982-04-22 1985-04-09 Imperial Chemical Industries Plc Method for combating pests
US4469682A (en) * 1983-01-28 1984-09-04 Merck & Co., Inc. Avermectin and milbemycin phosphate esters, pharmaceutical compositions, and method of use
US4582852A (en) * 1983-11-02 1986-04-15 Ciba-Geigy Corporation 14- and 15-hydroxy milbemycin derivatives for controlling plant and animal parasites
JPS60126289A (ja) * 1983-11-14 1985-07-05 Sankyo Co Ltd ミルベマイシン類の５−カ−ボネ−ト誘導体
US4579864A (en) * 1984-06-11 1986-04-01 Merck & Co., Inc. Avermectin and milbemycin 13-keto, 13-imino and 13-amino derivatives
US4547491A (en) * 1984-07-18 1985-10-15 Merck & Co., Inc. C-8A-Oxo-avermectin and milbemycin derivatives, pharmaceutical compositions and method of use
GB2168345B (en) * 1984-12-14 1988-05-25 Ciba Geigy Ag Pesticidal 13b-substituted milbemycin derivatives
GR861146B (en) * 1985-04-30 1986-08-14 American Cyanamid Co Chemical compounds
AU596586B2 (en) * 1985-04-30 1990-05-10 American Cyanamid Company Chemical derivatives of antibiotics S541
US4789684A (en) * 1985-05-02 1988-12-06 Merck & Co., Inc. Anthelmintic fermentation products of microorganisms
ES8605582A1 (es) * 1985-12-11 1986-03-16 Antibioticos Sa Un procedimiento para la preparacion de avermectinas
CA1301745C (en) * 1986-01-23 1992-05-26 Michael Vincent John Ramsay Macrolide antibiotics and their preparation
AU609032B2 (en) * 1986-03-12 1991-04-26 American Cyanamid Company Macrolide compounds
BR8701118A (pt) * 1986-03-12 1988-01-05 Glaxo Group Ltd Processo para a preparacao de um composto quimico,processo para combater pestes em agricultura,horicultura ou silvicultura,ou em lojas,predios e outros locais publicos e composicao de controle de pestes
GB8606108D0 (en) * 1986-03-12 1986-04-16 Glaxo Group Ltd Chemical compounds
CA1296329C (en) * 1986-06-06 1992-02-25 Derek R. Sutherland Macrolide compounds
US4849446A (en) * 1986-09-12 1989-07-18 American Cyanamid Company 23-imino derivatives of 23-keto compounds
US4886784A (en) * 1986-09-12 1989-12-12 American Cyanamid Company Novel 23-imino derivatives of 23-keto compounds
EP0259779B1 (en) * 1986-09-12 1994-08-10 American Cyanamid Company 23-Oxo (Keto) and 23-imino Derivatives of LL-F28249 Compounds
US4877888A (en) * 1986-09-12 1989-10-31 American Cyanamid Company 13-deoxy-23-imino derivatives of 13-deoxy C-076-aglycone compounds
EP0260537A1 (en) * 1986-09-12 1988-03-23 American Cyanamid Company 13-Deoxy-23-oxo(keto) and 23-imino derivatives of 13-deoxy C-076-aglycone compounds
US4916154A (en) * 1986-09-12 1990-04-10 American Cyanamid Company 23-Imino derivatives of LL-F28249 compounds
US4886829A (en) * 1987-03-06 1989-12-12 American Cyanamid Company 23-Oxo (keto) and 23-imino derivatives of mono- and diepoxy LL-F28249 compounds
US4806527A (en) * 1987-03-16 1989-02-21 Merck & Co., Inc. Avermectin derivatives
US4906619A (en) * 1988-07-22 1990-03-06 Merck & Co., Inc. Alkyl avermectin derivatives
US5428034A (en) * 1988-09-02 1995-06-27 Sankyo Co., Ltd. Milbemycin derivatives, their preparation and their use
US5830875A (en) * 1989-10-30 1998-11-03 Merck & Co., Inc. 24-and 25-substituted avermectin and milbemycin derivatives
JP2622197B2 (ja) * 1990-03-01 1997-06-18 三共株式会社 １３−エーテル置換ミルベマイシン誘導体
US5169839A (en) * 1990-05-11 1992-12-08 Merck & Co., Inc. Derivatives of 3'- and 3"-o-desmethyl avermectin compounds, compositions and methods of treating melmintic and parasitic infections
US5188944A (en) * 1990-06-22 1993-02-23 Merck & Co., Inc. Process for the glycosylation of avermectin agylcones
US5208222A (en) * 1991-03-28 1993-05-04 Merck & Co., Inc. 4"-and 4'-alkylthio avermectin derivatives
US5240915A (en) * 1991-10-15 1993-08-31 Merck & Co., Inc. Avermectin derivatives
EG19869A (en) * 1991-12-18 1996-03-31 Sankyo Co Substituted thio acetoxymilbemycon derivatives their preparation and their agrochemical uses
US5229415A (en) * 1992-03-24 1993-07-20 Merck & Co., Inc. Alkylthio alkyl avermectins are active antiparasitic agents
IL107810A0 (en) * 1992-12-17 1994-02-27 Exxon Chemical Patents Inc Functionalized polymers and processes for the preparation thereof
DE69611773T2 (de) * 1995-09-29 2001-09-13 Sankyo Co., Ltd. 13-Substituierte Milbemycin 5-Oxim Derivate, ihre Herstellung und Verwendung gegen Insekten und andere Schädlinge
AU5261301A (en) 2000-04-27 2001-11-12 Sankyo Co 13-substituted milbemycin derivatives, their preparation and their use against insects and other pests

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE434277B (sv) * 1976-04-19 1984-07-16 Merck & Co Inc Sett att framstella nya antihelmintiskt verkande foreningar genom odling av streptomyces avermitilis
US4134973A (en) * 1977-04-11 1979-01-16 Merck & Co., Inc. Carbohydrate derivatives of milbemycin and processes therefor
NZ188459A (en) * 1977-10-03 1982-09-07 Merck & Co Inc Derivatives of c-076 compounds and pesticidal compositions
US4172940A (en) * 1977-10-03 1979-10-30 Merck & Co., Inc. Purification of C-076 compounds by single column chromatography
US4206205A (en) * 1977-10-03 1980-06-03 Merck & Co., Inc. Monosaccharide and aglycone derivatives of C-076
US4201861A (en) * 1977-10-03 1980-05-06 Merck & Co., Inc. Acyl derivatives of C-076 compounds
US4199569A (en) * 1977-10-03 1980-04-22 Merck & Co., Inc. Selective hydrogenation products of C-076 compounds and derivatives thereof
PH16612A (en) * 1977-12-19 1983-11-28 Merck & Co Inc 13-halo and 13-deoxy derivatives of c-076 compounds
US4171314A (en) * 1977-12-19 1979-10-16 Merck & Co., Inc. 13-Halo and 13-deoxy C-076 compounds
US4203976A (en) * 1978-08-02 1980-05-20 Merck & Co., Inc. Sugar derivatives of C-076 compounds
US4200581A (en) * 1978-08-04 1980-04-29 Merck & Co., Inc. Alkyl derivatives of C-076 compounds

Also Published As

Publication number Publication date
PT72915B (en) 1983-02-16
NZ196897A (en) 1984-09-28
AU547211B2 (en) 1985-10-10
AU6973081A (en) 1981-11-05
JPS5718684A (en) 1982-01-30
ES8207544A1 (es) 1982-09-16
ATE8637T1 (de) 1984-08-15
US4289760A (en) 1981-09-15
EP0040913B1 (en) 1984-07-25
GR74875B (pt) 1984-07-12
ES501777A0 (es) 1982-09-16
DE3165016D1 (en) 1984-08-30
JPH0254358B2 (pt) 1990-11-21
ZA812908B (en) 1982-12-29
EP0040913A1 (en) 1981-12-02
PT72915A (en) 1981-05-01
CA1168605A (en) 1984-06-05

Similar Documents

Publication Publication Date Title
DK193881A (da) Fremgangsmaade til fremstilling af 23-ketoderivater af c-76forbindelser
IE781963L (en) C-076 compounds.
ES8302660A1 (es) "un procedimiento para la preparacion de piridin- y piracin-derivados".
OA08336A (fr) Dérivés de type 13-halogéno-milbémycine et compositions les contenant.
ES464354A1 (es) Procedimiento de preparacion de un complejo insectifugo e insecticida estable.
KR870010002A (ko) 살충성 6-아릴-피리딘 티오세미카르바존, 그의 조성물, 이들 화합물 및 조성물의 제조방법 및 그의 용도
KR870002116A (ko) 피리딘화합물과 살충제로의 사용
JPS5419943A (en) Urea or thiourea compounds, their preparation, and agricultural and horticultural fungicides comprising them as active constituents
JPH0417922B2 (pt)
IE872440L (en) 13-deoxy-23-oxo (keto) and 23-imino derivatives of 13-deoxy¹c-076-aglycone compounds
Bakry et al. Organothiocyanates as insecticides and carbamate synergists
IL44447A (en) N-phenyl-tricyclo(4,2,2,02,4)nonane(or nonene)-6,7-dicarboximides their preparation and their use as insecticides
ATE1422T1 (de) Prostaglandinanaloge imidazolderivate, ein verfahren zu deren herstellung und eine pharmazeutische zusammensetzung, die diese enthaelt.
ES470531A1 (es) Un procedimiento para la preparacion de esteres de acido naftalencarboxilico
IL43739A (en) 1,2,4-triazolyl-thiono and thionothiol phosphoric acid esters,their manufacture and insecticidal and acaricidal compositions containing them
ES481059A1 (es) Procedimiento para la preparacion de compuestos fenilen- o ciclohexilen-bis (2-propinilicos).
DK159130C (da) Herbicide praeparater, oxa- eller dioxa-heterodiaza-2,5-pentalener til anvendelse i praeparatet samt fremgangsmaade til bekaempelse af uoensket plantevaekst
ES420304A1 (es) Un procedimiento para la preparacion de una composicion a- gricola.
DK160733C (da) Synergistisk pesticidt virksomt praeparat og fremgangmsaade til bekaempelse af skadelige organismer
FR2453140A1 (fr) Procede de preparation de pesticides de type ester a l'aide de catalyseurs de transfert de phase
Potvin Studies relating to Ambruticin
JPH0465043B2 (pt)
IE822504L (en) Pyrimidine derivative.
JPS542322A (en) Alkyl n-acylanthranylate derivatives, their preparation, and agricultural and horticultural fungicide containing the same
FR2451161A1 (fr) Melanges synergiques a base d'esters de (s) allethrolone et de (r) allethrolone, doues d'activite contre les arthropodes

Legal Events

Date Code Title Description
ATS Application withdrawn