DK1924585T3 - Hidtil ukendt krystallinsk for af et pyridazino[4,5-b]indol-derivat - Google Patents
Hidtil ukendt krystallinsk for af et pyridazino[4,5-b]indol-derivatInfo
- Publication number
- DK1924585T3 DK1924585T3 DK06813757.9T DK06813757T DK1924585T3 DK 1924585 T3 DK1924585 T3 DK 1924585T3 DK 06813757 T DK06813757 T DK 06813757T DK 1924585 T3 DK1924585 T3 DK 1924585T3
- Authority
- DK
- Denmark
- Prior art keywords
- pyridazino
- hitherto
- lining
- crystalline
- indole derivative
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/50—Pyridazines; Hydrogenated pyridazines
- A61K31/5025—Pyridazines; Hydrogenated pyridazines ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hospice & Palliative Care (AREA)
- Pulmonology (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Oncology (AREA)
- Urology & Nephrology (AREA)
- Dermatology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US71215305P | 2005-08-29 | 2005-08-29 | |
PCT/US2006/033254 WO2007027525A1 (en) | 2005-08-29 | 2006-08-24 | Novel crystalline form of a pyridazino [4 , 5-b] indole derivative |
Publications (1)
Publication Number | Publication Date |
---|---|
DK1924585T3 true DK1924585T3 (da) | 2012-02-27 |
Family
ID=37546937
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK06813757.9T DK1924585T3 (da) | 2005-08-29 | 2006-08-24 | Hidtil ukendt krystallinsk for af et pyridazino[4,5-b]indol-derivat |
Country Status (32)
Country | Link |
---|---|
US (1) | US7683062B2 (da) |
EP (1) | EP1924585B1 (da) |
JP (1) | JP5063600B2 (da) |
KR (2) | KR20080050577A (da) |
CN (1) | CN101253176B (da) |
AR (1) | AR057099A1 (da) |
AT (1) | ATE531717T1 (da) |
AU (1) | AU2006285142B2 (da) |
BR (1) | BRPI0615259A2 (da) |
CA (1) | CA2619284C (da) |
CR (1) | CR9723A (da) |
CY (1) | CY1112317T1 (da) |
DK (1) | DK1924585T3 (da) |
EA (1) | EA014164B1 (da) |
EC (1) | ECSP088209A (da) |
ES (1) | ES2375841T3 (da) |
HK (1) | HK1123794A1 (da) |
HR (1) | HRP20120073T1 (da) |
IL (1) | IL189276A (da) |
MA (1) | MA30000B1 (da) |
NO (1) | NO20081365L (da) |
NZ (1) | NZ566087A (da) |
PL (1) | PL1924585T3 (da) |
PT (1) | PT1924585E (da) |
RS (1) | RS52318B (da) |
SI (1) | SI1924585T1 (da) |
TN (1) | TNSN08059A1 (da) |
TW (1) | TW200813060A (da) |
UA (1) | UA91716C2 (da) |
UY (1) | UY29771A1 (da) |
WO (1) | WO2007027525A1 (da) |
ZA (1) | ZA200801890B (da) |
Families Citing this family (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU2004311544A1 (en) * | 2003-11-17 | 2005-07-21 | Merck & Cie | Crystalline forms of (6R) -L-erythro-tetrahydrobiopterin dihydrochloride |
ES2370829T3 (es) * | 2004-06-02 | 2011-12-23 | Sandoz Ag | Producto intermedio de meropenem en forma cristalina. |
EP1928826B1 (en) * | 2005-09-21 | 2013-04-24 | 4Sc Ag | Sulphonylpyrrole hydrochloride salts as histone deacetylases inhibitors |
EA014905B1 (ru) * | 2005-10-31 | 2011-02-28 | Янссен Фармацевтика Н.В. | Новый способ получения пиперазинильных производных бензамида |
MX2008016008A (es) * | 2006-06-16 | 2009-01-16 | Lundbeck & Co As H | Formas cristalinas de 4-[2-(4-metilfenilsulfonil)-fenil] piperidina con inhibicion combinada de la recaptacion de serotonina y norepinefrina para el tratamiento del dolor neuropatico. |
BRPI0717394A2 (pt) * | 2006-10-27 | 2013-10-15 | Signal Pharm Llc | Forma cristalina, composição farmacêutica, forma de dosagem unitária única, método para tratar ou prevenir uma doença ou condição, e, processo para preparar um composto |
EP2085397A1 (en) * | 2008-01-21 | 2009-08-05 | Esteve Quimica, S.A. | Crystalline form of abacavir |
US7935817B2 (en) * | 2008-03-31 | 2011-05-03 | Apotex Pharmachem Inc. | Salt form and cocrystals of adefovir dipivoxil and processes for preparation thereof |
AR071318A1 (es) * | 2008-04-15 | 2010-06-09 | Basilea Pharmaceutica Ag | Benzhidril ester del acido (6r,7r)-7-{2-(5-amino-[1,2,4]tiadiazol-3-il)-2-[(z)-tritiloxiimino]-acetilamino}-3-[(r)-1'-terc-butoxicarbonil-2-oxo-[1,3']bipirrolidinil-(3e)-ilidenometil]-8-oxo-5-tia-1-aza-biciclo[4.2.0]oct-2-eno-2-carboxilico cristalino; su elaboracion y uso |
US8097719B2 (en) * | 2008-07-15 | 2012-01-17 | Genesen Labs | Meropenem intermediate in novel crystalline form and a method of manufacture of meropenem |
BRPI0917519A2 (pt) * | 2008-08-18 | 2015-08-04 | Sanofi Aventis Us Llc | Processo para preparacao de um polimorfo de 7-cloro-n,n,5-trimetil-4-oxo-3-fenil-3,5-di-hidro-4h-pir idazino[4,5-b]indol-1-acetamida |
KR101713453B1 (ko) | 2010-03-12 | 2017-03-07 | 오메로스 코포레이션 | Pde10 억제제 및 관련 조성물 및 방법 |
WO2012030957A2 (en) * | 2010-09-01 | 2012-03-08 | Arena Pharmaceuticals, Inc. | Non-hygroscopic salts of 5-ht2c agonists |
CN103930419B (zh) * | 2011-09-30 | 2016-06-01 | 广东东阳光药业有限公司 | 阿齐沙坦的晶型及其制备方法 |
NZ716462A (en) * | 2014-04-28 | 2017-11-24 | Omeros Corp | Optically active pde10 inhibitor |
NZ630810A (en) | 2014-04-28 | 2016-03-31 | Omeros Corp | Processes and intermediates for the preparation of a pde10 inhibitor |
AU2016250843A1 (en) | 2015-04-24 | 2017-10-12 | Omeros Corporation | PDE10 inhibitors and related compositions and methods |
JP2018535969A (ja) | 2015-11-04 | 2018-12-06 | オメロス コーポレーション | Pde10阻害剤の固体状態形態 |
CN111303230B (zh) * | 2020-03-09 | 2021-07-13 | 中国食品药品检定研究院 | 一种黄体酮共晶物及其制备方法和用途 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2766823B1 (fr) * | 1997-07-30 | 1999-10-08 | Synthelabo | Derives de 4-oxo-3,5-dihydro-4h-pyridazino[4,5-b] indole-1-acetamide, leur preparation et leur application en therapeutique |
FR2788696B1 (fr) * | 1999-01-26 | 2004-03-05 | Synthelabo | Utilisation de derives de pyridazino [4,5-b] indole-1-acetamide pour la preparation de medicaments destines aux maladies du systeme nerveux central |
FR2829939B3 (fr) | 2001-09-21 | 2003-11-28 | Sanofi Synthelabo | Utilisation du 7-chloro-n,n,5-trimethyl-4-oxo-3-phenyl-3,5- dihydro-4h-pyridazino(4,5-b)indole-1-acetamide pour la preparation de medicaments destines au traitement de la polyarthrite rhumatoide |
US20050220881A1 (en) | 2003-10-10 | 2005-10-06 | Bvm Holding Co. | Pharmaceutical composition |
-
2006
- 2006-08-24 PT PT06813757T patent/PT1924585E/pt unknown
- 2006-08-24 WO PCT/US2006/033254 patent/WO2007027525A1/en active Application Filing
- 2006-08-24 AU AU2006285142A patent/AU2006285142B2/en not_active Ceased
- 2006-08-24 CA CA2619284A patent/CA2619284C/en not_active Expired - Fee Related
- 2006-08-24 BR BRPI0615259-7A patent/BRPI0615259A2/pt not_active IP Right Cessation
- 2006-08-24 EP EP06813757A patent/EP1924585B1/en active Active
- 2006-08-24 KR KR1020087004953A patent/KR20080050577A/ko active IP Right Grant
- 2006-08-24 PL PL06813757T patent/PL1924585T3/pl unknown
- 2006-08-24 CN CN2006800314750A patent/CN101253176B/zh not_active Expired - Fee Related
- 2006-08-24 ES ES06813757T patent/ES2375841T3/es active Active
- 2006-08-24 EA EA200800716A patent/EA014164B1/ru not_active IP Right Cessation
- 2006-08-24 UA UAA200803953A patent/UA91716C2/ru unknown
- 2006-08-24 RS RS20120032A patent/RS52318B/en unknown
- 2006-08-24 DK DK06813757.9T patent/DK1924585T3/da active
- 2006-08-24 SI SI200631252T patent/SI1924585T1/sl unknown
- 2006-08-24 NZ NZ566087A patent/NZ566087A/en not_active IP Right Cessation
- 2006-08-24 AT AT06813757T patent/ATE531717T1/de active
- 2006-08-24 JP JP2008529130A patent/JP5063600B2/ja not_active Expired - Fee Related
- 2006-08-24 KR KR1020137018636A patent/KR20130087059A/ko not_active Application Discontinuation
- 2006-08-24 ZA ZA200801890A patent/ZA200801890B/xx unknown
- 2006-08-28 AR ARP060103740A patent/AR057099A1/es not_active Application Discontinuation
- 2006-08-29 UY UY29771A patent/UY29771A1/es unknown
- 2006-08-29 TW TW095131681A patent/TW200813060A/zh unknown
-
2008
- 2008-02-04 IL IL189276A patent/IL189276A/en not_active IP Right Cessation
- 2008-02-06 TN TNP2008000059A patent/TNSN08059A1/en unknown
- 2008-02-11 CR CR9723A patent/CR9723A/es unknown
- 2008-02-14 US US12/031,243 patent/US7683062B2/en not_active Expired - Fee Related
- 2008-02-20 EC EC2008008209A patent/ECSP088209A/es unknown
- 2008-03-14 NO NO20081365A patent/NO20081365L/no not_active Application Discontinuation
- 2008-03-17 MA MA30757A patent/MA30000B1/fr unknown
-
2009
- 2009-02-19 HK HK09101601.0A patent/HK1123794A1/xx not_active IP Right Cessation
-
2012
- 2012-01-23 HR HRP20120073TT patent/HRP20120073T1/hr unknown
- 2012-01-26 CY CY20121100092T patent/CY1112317T1/el unknown
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
DK1924585T3 (da) | Hidtil ukendt krystallinsk for af et pyridazino[4,5-b]indol-derivat | |
HK1100410A1 (en) | Indole derivatives having piperidine rings | |
DK1924151T3 (da) | Oral frigivelsessystem med styret frigivelse | |
DK1883451T3 (da) | Substituerede indolforbindelser med NOS-hæmmende virkning | |
ATE501119T1 (de) | Entzündungshemmende indol-derivate | |
MA28347A1 (fr) | Dérivés de quinoléine substitués | |
DK1737461T3 (da) | Carbolin-derivater til inhibering af angiogenese | |
PL2067108T3 (pl) | Lokalizowanie węzłów odniesienia do pozycjonowania | |
DK1710241T3 (da) | Intermediatforbindelser til fremstilling af trans-5-chlor-2-methyl-2,3,3a,12b-tetrahydro-1h-dibenz[2,3:6,7]oxepino[4,5-c]pyrrol | |
GB0419481D0 (en) | Isoindolin-1-one derivatives | |
DK1756049T3 (da) | Fremgangsmåde til fremstilling af 1,4-diphenylazetidinon-derivater | |
DK1874766T3 (da) | Krystallinsk form af en quinolinon-carboxamid-forbindelse | |
EP1893625A4 (en) | PROCESS FOR THE PREPARATION OF 9-DEAZAPURINE DERIVATIVES | |
DK2213654T3 (da) | Fremgangsmåde til fremstilling af 2-amino-5-brombenzamid derivater | |
DK1838683T3 (da) | Fremgangsmåde til fremstilling af [1,4,5]-oxadiazepinderivater | |
IL190729A0 (en) | Methods for preparing glutamic acid derivatives | |
DK1784183T3 (da) | Fremgangsmåder til fremstilling af isothiazolderivater | |
GB0405334D0 (en) | Method for exchanging signals via nodes | |
EP1919871A4 (en) | PROCESS FOR SYNTHESIS OF CHINOLINE DERIVATIVES | |
DK1682541T3 (da) | Fremgangsmåde til fremstilling af tiotropiumsalte | |
DK1888613T3 (da) | Fremgangsmåde til fremstilling af thiophenglycosidderivater | |
EP1880995A4 (en) | METHOD OF SYNTHESIZING AN INDOLE DERIVATIVE COMPRISING A PIPERIDINE CYCLE | |
EP1849766A4 (en) | BETA-BENZYLOXYASPARTICAL ACID DERIVATIVE HAVING TWO SUBSTITUENTS ON BENZENIC CORE | |
GB0521726D0 (en) | Methods for the preparation of organic compounds | |
GB0521728D0 (en) | Methods for the preparation of organic compounds |