DK170234B1 - Hydrochloridhydrat af Endo-4-amino-5-chlor-2-methoxy-N-(1'-azabicyclo-[3.3.1]-non-4'-yl)-benzamid, fremgangsmåde til fremstilling deraf, farmaceutisk præparat indeholdende forbindelsen samt anvendelse af forbindelsen - Google Patents

Hydrochloridhydrat af Endo-4-amino-5-chlor-2-methoxy-N-(1'-azabicyclo-[3.3.1]-non-4'-yl)-benzamid, fremgangsmåde til fremstilling deraf, farmaceutisk præparat indeholdende forbindelsen samt anvendelse af forbindelsen Download PDF

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Publication number
DK170234B1
DK170234B1 DK145287A DK145287A DK170234B1 DK 170234 B1 DK170234 B1 DK 170234B1 DK 145287 A DK145287 A DK 145287A DK 145287 A DK145287 A DK 145287A DK 170234 B1 DK170234 B1 DK 170234B1
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DK
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Prior art keywords
compound
compound according
azabicyclo
endo
chloro
Prior art date
Application number
DK145287A
Other languages
Danish (da)
English (en)
Other versions
DK145287D0 (da
DK145287A (da
Inventor
Paul Smith
Original Assignee
Beecham Group Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Beecham Group Plc filed Critical Beecham Group Plc
Publication of DK145287D0 publication Critical patent/DK145287D0/da
Publication of DK145287A publication Critical patent/DK145287A/da
Application granted granted Critical
Publication of DK170234B1 publication Critical patent/DK170234B1/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK145287A 1986-03-22 1987-03-20 Hydrochloridhydrat af Endo-4-amino-5-chlor-2-methoxy-N-(1'-azabicyclo-[3.3.1]-non-4'-yl)-benzamid, fremgangsmåde til fremstilling deraf, farmaceutisk præparat indeholdende forbindelsen samt anvendelse af forbindelsen DK170234B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB868607163A GB8607163D0 (en) 1986-03-22 1986-03-22 Chemical compound
GB8607163 1986-03-22

Publications (3)

Publication Number Publication Date
DK145287D0 DK145287D0 (da) 1987-03-20
DK145287A DK145287A (da) 1987-09-23
DK170234B1 true DK170234B1 (da) 1995-07-10

Family

ID=10595084

Family Applications (1)

Application Number Title Priority Date Filing Date
DK145287A DK170234B1 (da) 1986-03-22 1987-03-20 Hydrochloridhydrat af Endo-4-amino-5-chlor-2-methoxy-N-(1'-azabicyclo-[3.3.1]-non-4'-yl)-benzamid, fremgangsmåde til fremstilling deraf, farmaceutisk præparat indeholdende forbindelsen samt anvendelse af forbindelsen

Country Status (14)

Country Link
US (1) US4800225A (es)
EP (1) EP0239321B1 (es)
JP (1) JPH07107062B2 (es)
AU (1) AU600476B2 (es)
CA (1) CA1308104C (es)
DE (1) DE3786187T2 (es)
DK (1) DK170234B1 (es)
ES (1) ES2058107T3 (es)
GB (1) GB8607163D0 (es)
HK (1) HK1004548A1 (es)
IE (1) IE60166B1 (es)
NZ (1) NZ219719A (es)
PT (1) PT84535B (es)
ZA (1) ZA872057B (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5187166A (en) * 1990-07-31 1993-02-16 Nisshin Flour Milling Co., Ltd. Azabicyclo derivatives and their use as antiemetics
US5344831A (en) * 1992-01-31 1994-09-06 Nisshin Flour Milling Co., Ltd. Diazabicyclo derivatives
US6340116B1 (en) * 1999-09-16 2002-01-22 Kenneth B. Cecil Proximity card with incorporated pin code protection
US6875774B2 (en) 2002-08-06 2005-04-05 The University Of North Carolina Aza-bridged bicyclic amine derivatives for use as novel cholinergic receptor ligands
GB0321091D0 (en) * 2003-09-09 2003-10-08 Alizyme Therapeutics Ltd Synthesis
GB0329319D0 (en) * 2003-12-18 2004-01-21 Alizyme Therapeutics Ltd Synthesis

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0067565A1 (en) * 1981-06-16 1982-12-22 Beecham Group Plc Pharmaceutically active compounds
AU563225B2 (en) * 1982-04-14 1987-07-02 Alizyme Therapeutics Limited I-aza bicyclic compounds
US4612319A (en) * 1982-04-14 1986-09-16 Beecham Group P.L.C. Bridged quinolizidinylbenzamides, compositions containing them and methods for their use

Also Published As

Publication number Publication date
IE870740L (en) 1987-09-22
DE3786187T2 (de) 1993-10-14
ES2058107T3 (es) 1994-11-01
NZ219719A (en) 1990-03-27
IE60166B1 (en) 1994-06-15
JPH07107062B2 (ja) 1995-11-15
US4800225A (en) 1989-01-24
JPS62270583A (ja) 1987-11-24
AU7044287A (en) 1987-09-24
HK1004548A1 (en) 1998-11-27
EP0239321A2 (en) 1987-09-30
EP0239321B1 (en) 1993-06-16
PT84535B (pt) 1989-11-10
CA1308104C (en) 1992-09-29
DE3786187D1 (de) 1993-07-22
AU600476B2 (en) 1990-08-16
ZA872057B (en) 1987-12-30
DK145287D0 (da) 1987-03-20
EP0239321A3 (en) 1989-08-30
PT84535A (en) 1987-04-01
GB8607163D0 (en) 1986-04-30
DK145287A (da) 1987-09-23

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Legal Events

Date Code Title Description
B1 Patent granted (law 1993)
PUP Patent expired