DK170051B1 - 14-Chlordaunomycin og syreadditionssalte deraf, fremgangsmåde til fremstilling af (2"R)-4'-O-tetrahydropyranyladriamycin samt (2"R)-14-chlor-4'-O-tetrahydropyranyldaunomycin - Google Patents

14-Chlordaunomycin og syreadditionssalte deraf, fremgangsmåde til fremstilling af (2"R)-4'-O-tetrahydropyranyladriamycin samt (2"R)-14-chlor-4'-O-tetrahydropyranyldaunomycin Download PDF

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Publication number
DK170051B1
DK170051B1 DK317888A DK317888A DK170051B1 DK 170051 B1 DK170051 B1 DK 170051B1 DK 317888 A DK317888 A DK 317888A DK 317888 A DK317888 A DK 317888A DK 170051 B1 DK170051 B1 DK 170051B1
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DK
Denmark
Prior art keywords
formula
chloro
daunomycin
group
compound
Prior art date
Application number
DK317888A
Other languages
Danish (da)
English (en)
Other versions
DK317888A (da
DK317888D0 (da
Inventor
Tomoya Machinami
Takeshi Nakamura
Ken Nishihata
Shinichi Kondo
Tomio Takeuchi
Original Assignee
Zaidan Hojin Biseibutsu
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP14533987A external-priority patent/JPH07103145B2/ja
Priority claimed from JP17392487A external-priority patent/JPH07103146B2/ja
Application filed by Zaidan Hojin Biseibutsu filed Critical Zaidan Hojin Biseibutsu
Publication of DK317888D0 publication Critical patent/DK317888D0/da
Publication of DK317888A publication Critical patent/DK317888A/da
Application granted granted Critical
Publication of DK170051B1 publication Critical patent/DK170051B1/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/24—Condensed ring systems having three or more rings
    • C07H15/252—Naphthacene radicals, e.g. daunomycins, adriamycins

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK317888A 1987-06-12 1988-06-10 14-Chlordaunomycin og syreadditionssalte deraf, fremgangsmåde til fremstilling af (2"R)-4'-O-tetrahydropyranyladriamycin samt (2"R)-14-chlor-4'-O-tetrahydropyranyldaunomycin DK170051B1 (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP14533987A JPH07103145B2 (ja) 1987-06-12 1987-06-12 １４−クロロダウノマイシン及びその製造方法
JP14533987 1987-06-12
JP17392487 1987-07-14
JP17392487A JPH07103146B2 (ja) 1987-07-14 1987-07-14 （２″ｒ）−４′−０−テトラヒドロピラニルアドリアマイシンの製造方法

Publications (3)

Publication Number Publication Date
DK317888D0 DK317888D0 (da) 1988-06-10
DK317888A DK317888A (da) 1988-12-13
DK170051B1 true DK170051B1 (da) 1995-05-08

Family

ID=26476490

Family Applications (2)

Application Number Title Priority Date Filing Date
DK317888A DK170051B1 (da) 1987-06-12 1988-06-10 14-Chlordaunomycin og syreadditionssalte deraf, fremgangsmåde til fremstilling af (2"R)-4'-O-tetrahydropyranyladriamycin samt (2"R)-14-chlor-4'-O-tetrahydropyranyldaunomycin
DK079194A DK170172B1 (da) 1987-06-12 1994-07-01 Fremgangsmåde til fremstilling af 14-chlor-daunomycin eller et syreadditionssalt deraf

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK079194A DK170172B1 (da) 1987-06-12 1994-07-01 Fremgangsmåde til fremstilling af 14-chlor-daunomycin eller et syreadditionssalt deraf

Country Status (7)

Country Link
US (1) US4889926A (de)
EP (1) EP0295119B1 (de)
KR (1) KR950013771B1 (de)
CA (1) CA1303027C (de)
DE (1) DE3886101T2 (de)
DK (2) DK170051B1 (de)
ES (1) ES2060652T3 (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2003250151A1 (en) * 2002-07-24 2004-02-16 Diatos S.A. Method for the synthesis of anthracycline-peptide conjugates
CN111675738A (zh) * 2020-07-10 2020-09-18 苏州赛分科技有限公司 一种吡柔比星的纯化方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK160616C (da) * 1979-02-03 1991-09-02 Zaidan Hojin Biseibutsu Fremgangsmaade til fremstilling af anthracyclinderivater eller syreadditionssalte deraf
JPS56156300A (en) * 1980-04-26 1981-12-02 Microbial Chem Res Found Novel preparative method of anthracyclin derivative
JPS62116591A (ja) * 1985-11-16 1987-05-28 Microbial Chem Res Found ４′−Ｏ−テトラヒドロピラニルアドリアマイシンｂの製造方法

Also Published As

Publication number Publication date
DE3886101D1 (de) 1994-01-20
EP0295119B1 (de) 1993-12-08
DK79194A (de) 1994-07-01
EP0295119A3 (en) 1990-05-16
DK170172B1 (da) 1995-06-06
US4889926A (en) 1989-12-26
KR950013771B1 (ko) 1995-11-15
CA1303027C (en) 1992-06-09
DK317888A (da) 1988-12-13
KR890000509A (ko) 1989-03-15
EP0295119A2 (de) 1988-12-14
DK317888D0 (da) 1988-06-10
DE3886101T2 (de) 1994-04-14
ES2060652T3 (es) 1994-12-01

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PBP Patent lapsed

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