DK1673370T3 - Krystallingsk form af linezolid - Google Patents
Krystallingsk form af linezolidInfo
- Publication number
- DK1673370T3 DK1673370T3 DK03769887T DK03769887T DK1673370T3 DK 1673370 T3 DK1673370 T3 DK 1673370T3 DK 03769887 T DK03769887 T DK 03769887T DK 03769887 T DK03769887 T DK 03769887T DK 1673370 T3 DK1673370 T3 DK 1673370T3
- Authority
- DK
- Denmark
- Prior art keywords
- linezolid
- crystalline form
- preparation
- relates
- present
- Prior art date
Links
- TYZROVQLWOKYKF-ZDUSSCGKSA-N linezolid Chemical compound O=C1O[C@@H](CNC(=O)C)CN1C(C=C1F)=CC=C1N1CCOCC1 TYZROVQLWOKYKF-ZDUSSCGKSA-N 0.000 title abstract 2
- 229960003907 linezolid Drugs 0.000 title abstract 2
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PCT/IN2003/000336 WO2005035530A1 (fr) | 2003-10-16 | 2003-10-16 | Nouvelle forme cristalline du linezolid |
Publications (1)
Publication Number | Publication Date |
---|---|
DK1673370T3 true DK1673370T3 (da) | 2009-12-07 |
Family
ID=34430675
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK03769887T DK1673370T3 (da) | 2003-10-16 | 2003-10-16 | Krystallingsk form af linezolid |
Country Status (10)
Country | Link |
---|---|
US (4) | US7714128B2 (fr) |
EP (3) | EP2100884A1 (fr) |
AT (1) | ATE442364T1 (fr) |
AU (1) | AU2003278592A1 (fr) |
DE (2) | DE60329237D1 (fr) |
DK (1) | DK1673370T3 (fr) |
ES (3) | ES2331001T3 (fr) |
HU (1) | HUE051230T2 (fr) |
PT (1) | PT1673370E (fr) |
WO (1) | WO2005035530A1 (fr) |
Families Citing this family (36)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2331001T3 (es) | 2003-10-16 | 2009-12-18 | Symed Labs Limited | Forma cristalina de linezolid. |
EP1737850B1 (fr) | 2004-04-19 | 2007-10-03 | Symed Labs Limited | Nouveau procede pour preparer du linezolide et des composes associes |
MX2007000084A (es) * | 2004-06-29 | 2007-06-14 | Teva Pharma | Formas solidas de linezolid y procesos para la preparacion delas mismas. |
JP2007504173A (ja) * | 2004-06-29 | 2007-03-01 | テバ ファーマシューティカル インダストリーズ リミティド | リネゾリドのiv型結晶 |
JP2008530028A (ja) | 2005-02-24 | 2008-08-07 | テバ ファーマシューティカル インダストリーズ リミティド | リネゾリッド中間体の調製方法 |
DE602006001699D1 (de) * | 2005-07-20 | 2008-08-21 | Teva Pharma | Stabile pharmazeutische Zusammensetzung mit Linezolid Form IV |
IT1390957B1 (it) * | 2008-07-07 | 2011-10-27 | Dipharma Francis Srl | Sali di linezolid e loro uso nella preparazione di forme cristalline di linezolid |
EP2033960A3 (fr) | 2007-09-04 | 2009-04-29 | Dipharma Francis S.r.l. | Formule d'hydrate cristalline de linézolide et sels de linézolide |
WO2009032294A2 (fr) * | 2007-09-06 | 2009-03-12 | Teva Pharmaceutical Industries Ltd. | Procédés de préparation d'un intermédiaire du linézolide, hydroxyde de linezolide |
WO2009140466A2 (fr) * | 2008-05-14 | 2009-11-19 | Dr. Reddy's Laboratories Ltd. | Co-cristaux de linézolide |
EP2493867A1 (fr) | 2009-10-28 | 2012-09-05 | Synthon BV | Procédé de fabrication d'une forme cristalline a de linézolide |
WO2011050826A1 (fr) * | 2009-10-28 | 2011-05-05 | Synthon B.V. | Procédé de fabrication d'une forme cristalline de linézolide |
EP2516408A1 (fr) | 2009-12-26 | 2012-10-31 | Alembic Pharmaceuticals Limited | Procédé pour la préparation de linézolide |
EP2603505A1 (fr) | 2010-08-11 | 2013-06-19 | Synthon BV | Procédé pour fabriquer du linézolid |
EP2603506A1 (fr) | 2010-08-11 | 2013-06-19 | Synthon BV | Procédé pour fabriquer du linézolid |
EP2611799A4 (fr) | 2010-09-02 | 2014-01-29 | Hetero Research Foundation | Compositions pharmaceutiques de linézolide |
CN102070548B (zh) * | 2011-01-13 | 2012-12-26 | 浙江新东港药业股份有限公司 | 一种晶型ⅰ型利奈唑胺的蒸发结晶工艺 |
WO2012114354A1 (fr) | 2011-02-24 | 2012-08-30 | Lee Pharma Limited | Forme ii cristalline anhydre de linézolide |
WO2012119653A1 (fr) | 2011-03-09 | 2012-09-13 | Synthon Bv | Procédé de préparation de la forme cristalline a du linézolid |
CN102766106A (zh) * | 2011-05-03 | 2012-11-07 | 江苏豪森医药集团有限公司 | 利奈唑胺的新晶型及其制备方法 |
ITMI20111311A1 (it) * | 2011-07-14 | 2013-01-15 | Dipharma Francis Srl | Sali di linezolid e loro uso nella preparazione di forme cristalline di linezolid |
WO2013072923A1 (fr) | 2011-09-19 | 2013-05-23 | Cadila Healthcare Limited | Procédé de préparation de linézolide cristallin |
WO2013093751A1 (fr) * | 2011-12-24 | 2013-06-27 | Alembic Pharmaceuticals Limited | Conditionnement pour le linézolide |
EP2852580A1 (fr) | 2012-01-24 | 2015-04-01 | Jubilant Life Sciences Ltd. | Procédé amélioré de préparation de la forme cristalline stable i du linézolide, pratiquement exempte de solvant résiduel |
WO2013120496A1 (fr) | 2012-02-14 | 2013-08-22 | Pharmathen S.A. | Procédé pour la préparation de linézolide sous forme cristalline et de sels de celui-ci |
WO2013190559A1 (fr) * | 2012-06-19 | 2013-12-27 | Symed Labs Limited | Procédés perfectionnés pour la préparation de forme cristalline iii du linézolide |
US9492459B2 (en) * | 2012-08-10 | 2016-11-15 | Indoco Remedies Limited | Pharmaceutical composition of linezolid |
EP2917189B1 (fr) | 2012-11-09 | 2016-08-17 | Synthon BV | Procédé de production de linézolide |
WO2014118809A1 (fr) | 2013-01-29 | 2014-08-07 | Actavis Group Ptc Ehf. | Composition pharmaceutique comprenant du linézolide |
WO2015068121A1 (fr) | 2013-11-06 | 2015-05-14 | Unimark Remedies Ltd. | Procédé pour la préparation de la forme cristalline i de linézolide et ses compositions |
CN105254580B (zh) * | 2014-04-22 | 2018-01-02 | 江苏豪森药业集团有限公司 | 利奈唑胺晶型的制备方法 |
WO2016113751A1 (fr) * | 2015-01-13 | 2016-07-21 | Nosch Labs Private Limited | Procédé de préparation de linézolide cristallin de forme iii |
WO2018051360A1 (fr) * | 2016-09-16 | 2018-03-22 | Lee Pharma Limited | Nouveau procédé de préparation de linézolide cristallin de forme iii |
WO2019097242A1 (fr) | 2017-11-16 | 2019-05-23 | Persica Pharmaceuticals Ltd. | Formulations de linézolide |
CN110194750A (zh) * | 2019-06-19 | 2019-09-03 | 四川美大康华康药业有限公司 | 一种利奈唑胺的制备方法及精制方法 |
WO2023062080A1 (fr) | 2021-10-12 | 2023-04-20 | Persica Pharmaceuticals Ltd. | Traitement de la lombalgie |
Family Cites Families (26)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US583870A (en) * | 1897-06-01 | Wrench | ||
DE2810349A1 (de) | 1978-03-10 | 1979-09-20 | Kali Chemie Pharma Gmbh | Verfahren zur herstellung von 3-hydroxy-6-phenyl-1,2,3,4-tetrahydro- 1,5-benzodiazocinen |
FR2506769A2 (fr) | 1978-06-09 | 1982-12-03 | Delalande Sa | Para-((cyano-5 n pentyl-1) phenyl)-3 methoxymethyl-5 oxazolidinone-2, son procede de preparation et ses applications en therapeutique |
US4340606A (en) | 1980-10-23 | 1982-07-20 | E. I. Du Pont De Nemours And Company | 3-(p-Alkylsulfonylphenyl)oxazolidinone derivatives as antibacterial agents |
FR2608604B1 (fr) | 1986-12-19 | 1989-04-28 | Delalande Sa | Derives 5-hydroxyethyles de l'oxazolidinone-2, leurs procedes de preparation et leurs applications en therapeutique |
US5006528A (en) | 1988-10-31 | 1991-04-09 | Otsuka Pharmaceutical Co., Ltd. | Carbostyril derivatives |
DE9310451U1 (de) | 1993-03-05 | 1994-06-30 | Landis & Gyr Business Support | Steuer- bzw. Regeleinrichtung für Gas-Feuerungsautomaten von Heizungsanlagen |
EP0615095B1 (fr) | 1993-03-11 | 1997-05-07 | Landis & Gyr Technology Innovation AG | Commande de brûleur |
US5688792A (en) | 1994-08-16 | 1997-11-18 | Pharmacia & Upjohn Company | Substituted oxazine and thiazine oxazolidinone antimicrobials |
MY115155A (en) | 1993-09-09 | 2003-04-30 | Upjohn Co | Substituted oxazine and thiazine oxazolidinone antimicrobials. |
KR100530297B1 (ko) | 1996-04-11 | 2005-11-22 | 파마시아 앤드 업존 캄파니 엘엘씨 | 옥사졸리디논의 제조 방법 |
EP0890791A1 (fr) | 1997-07-11 | 1999-01-13 | Electrowatt Technology Innovation AG | Dispositif de commande et de régulation pour un brûleur |
EP1028940B1 (fr) * | 1997-11-07 | 2007-04-18 | Pharmacia & Upjohn Company LLC | Procede de production d'oxazolidinones |
US6444813B2 (en) * | 2000-02-02 | 2002-09-03 | Pharmacia & Upjohn Company | Linezolid-crystal form II |
AR027261A1 (es) | 2000-02-02 | 2003-03-19 | Upjohn Co | Linezolid forma cristalina ii |
MY127336A (en) * | 2000-03-22 | 2006-11-30 | Upjohn Co | Container for linezolid iv solution |
DE10037585A1 (de) | 2000-08-02 | 2002-02-14 | Valeo Schalter & Sensoren Gmbh | Rückstellvorrichtung für einen Blinkerschalter in Kraftfahrzeugen |
PL365608A1 (en) | 2000-08-14 | 2005-01-10 | Teva Pharmaceutical Industries Ltd. | Preparation of risperidone |
US20030008012A1 (en) * | 2001-02-05 | 2003-01-09 | Pena Lorraine E. | Composition for rectal delivery of an oxazolidinone antibacterial drug |
WO2002085849A2 (fr) * | 2001-04-20 | 2002-10-31 | Pharmacia & Upjohn Company | Procede de preparation d'oxazolidinones |
CN1155585C (zh) | 2001-12-19 | 2004-06-30 | 中国医学科学院医药生物技术研究所 | 3,5-取代噁唑烷酮衍生物及其制备方法和应用 |
US6992219B2 (en) | 2002-08-09 | 2006-01-31 | Cephalon France | Modafinil polymorphic forms |
ES2331001T3 (es) | 2003-10-16 | 2009-12-18 | Symed Labs Limited | Forma cristalina de linezolid. |
EP1737850B1 (fr) | 2004-04-19 | 2007-10-03 | Symed Labs Limited | Nouveau procede pour preparer du linezolide et des composes associes |
JP2007504173A (ja) | 2004-06-29 | 2007-03-01 | テバ ファーマシューティカル インダストリーズ リミティド | リネゾリドのiv型結晶 |
ATE429423T1 (de) | 2004-07-20 | 2009-05-15 | Symed Labs Ltd | Neue zwischenprodukte für linezolid und verwandte verbindungen |
-
2003
- 2003-10-16 ES ES03769887T patent/ES2331001T3/es not_active Expired - Lifetime
- 2003-10-16 EP EP20090163348 patent/EP2100884A1/fr not_active Withdrawn
- 2003-10-16 ES ES09163348T patent/ES2331454T1/es active Pending
- 2003-10-16 EP EP15155714.7A patent/EP2902386B1/fr not_active Expired - Lifetime
- 2003-10-16 HU HUE15155714A patent/HUE051230T2/hu unknown
- 2003-10-16 PT PT03769887T patent/PT1673370E/pt unknown
- 2003-10-16 DE DE60329237T patent/DE60329237D1/de not_active Expired - Lifetime
- 2003-10-16 EP EP03769887A patent/EP1673370B1/fr not_active Revoked
- 2003-10-16 DK DK03769887T patent/DK1673370T3/da active
- 2003-10-16 AT AT03769887T patent/ATE442364T1/de active
- 2003-10-16 ES ES15155714T patent/ES2803516T3/es not_active Expired - Lifetime
- 2003-10-16 WO PCT/IN2003/000336 patent/WO2005035530A1/fr active Application Filing
- 2003-10-16 AU AU2003278592A patent/AU2003278592A1/en not_active Abandoned
- 2003-10-16 DE DE2009163348 patent/DE09163348T1/de active Pending
- 2003-10-16 US US10/524,478 patent/US7714128B2/en active Active
-
2007
- 2007-09-26 US US11/861,406 patent/US7732597B2/en not_active Expired - Fee Related
- 2007-09-26 US US11/861,340 patent/US7718799B2/en not_active Expired - Fee Related
- 2007-09-26 US US11/861,433 patent/US7718800B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
DE60329237D1 (de) | 2009-10-22 |
US20060128703A1 (en) | 2006-06-15 |
EP1673370B1 (fr) | 2009-09-09 |
WO2005035530A1 (fr) | 2005-04-21 |
ATE442364T1 (de) | 2009-09-15 |
US20080090820A1 (en) | 2008-04-17 |
EP2902386A1 (fr) | 2015-08-05 |
EP2100884A1 (fr) | 2009-09-16 |
US20080090824A1 (en) | 2008-04-17 |
EP1673370A1 (fr) | 2006-06-28 |
US20080091011A1 (en) | 2008-04-17 |
US7718799B2 (en) | 2010-05-18 |
ES2803516T3 (es) | 2021-01-27 |
DE09163348T1 (de) | 2010-01-07 |
HUE051230T2 (hu) | 2021-03-01 |
EP2902386B1 (fr) | 2020-04-08 |
ES2331001T3 (es) | 2009-12-18 |
US7718800B2 (en) | 2010-05-18 |
PT1673370E (pt) | 2009-11-05 |
ES2331454T1 (es) | 2010-01-05 |
US7714128B2 (en) | 2010-05-11 |
US7732597B2 (en) | 2010-06-08 |
AU2003278592A1 (en) | 2005-04-27 |
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